AU2420195A - Pharmaceutical composition for treating glaucoma containing terazosin - Google Patents
Pharmaceutical composition for treating glaucoma containing terazosinInfo
- Publication number
- AU2420195A AU2420195A AU24201/95A AU2420195A AU2420195A AU 2420195 A AU2420195 A AU 2420195A AU 24201/95 A AU24201/95 A AU 24201/95A AU 2420195 A AU2420195 A AU 2420195A AU 2420195 A AU2420195 A AU 2420195A
- Authority
- AU
- Australia
- Prior art keywords
- pharmaceutical composition
- intraocular pressure
- terazosin
- glaucoma
- terazosin hydrochloride
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- VCKUSRYTPJJLNI-UHFFFAOYSA-N terazosin Chemical compound N=1C(N)=C2C=C(OC)C(OC)=CC2=NC=1N(CC1)CCN1C(=O)C1CCCO1 VCKUSRYTPJJLNI-UHFFFAOYSA-N 0.000 title claims description 51
- 208000010412 Glaucoma Diseases 0.000 title claims description 28
- 239000008194 pharmaceutical composition Substances 0.000 title claims description 24
- 229960001693 terazosin Drugs 0.000 title description 15
- 239000002997 ophthalmic solution Substances 0.000 claims description 27
- 229940054534 ophthalmic solution Drugs 0.000 claims description 24
- 150000003839 salts Chemical class 0.000 claims description 16
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- 238000000034 method Methods 0.000 claims description 4
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- 238000004519 manufacturing process Methods 0.000 claims description 3
- 230000004410 intraocular pressure Effects 0.000 description 42
- 238000012360 testing method Methods 0.000 description 34
- 239000003814 drug Substances 0.000 description 32
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- 229960001909 terazosin hydrochloride Drugs 0.000 description 31
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Ophthalmology & Optometry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP10367694 | 1994-05-18 | ||
| JP6-103676 | 1994-05-18 | ||
| PCT/JP1995/000920 WO1995031200A1 (en) | 1994-05-18 | 1995-05-15 | Pharmaceutical composition for treating glaucoma containing terazosin |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2420195A true AU2420195A (en) | 1995-12-05 |
Family
ID=14360400
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU24201/95A Abandoned AU2420195A (en) | 1994-05-18 | 1995-05-15 | Pharmaceutical composition for treating glaucoma containing terazosin |
Country Status (10)
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2454544A1 (en) * | 2001-07-02 | 2003-01-16 | Santen Pharmaceutical Co., Ltd. | Optic nerve protecting agents containing .alpha.1 receptor blocker as active ingredient |
| US20040235932A1 (en) * | 2001-07-13 | 2004-11-25 | Kenji Yamazaki | Ophthalmic pharmaceutical compositions |
| CN104840436B (zh) * | 2015-06-11 | 2017-12-05 | 刘磊 | 药物组合物 |
| WO2017002846A1 (ja) * | 2015-06-30 | 2017-01-05 | 株式会社ニデック | 視機能測定装置、および視機能測定プログラム |
| CN112439071B (zh) * | 2019-09-04 | 2022-05-20 | 武汉科福新药有限责任公司 | 透皮促渗组合物及其在噻吗洛尔制剂中的应用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2824863B2 (ja) * | 1989-07-12 | 1998-11-18 | エーザイ株式会社 | α▲下１▼―ブロッカー点眼剤 |
| DE436726T1 (de) * | 1989-08-03 | 1992-02-06 | Eisai Co., Ltd., Tokio/Tokyo | Verfahren zur photostabilisierung von augenspuelloesungen sowie photostabilisierte augenspuelloesung. |
| US5256667A (en) * | 1991-09-25 | 1993-10-26 | Merck & Co., Inc. | Quinazolinones and pyridopyrimidinones |
-
1995
- 1995-05-15 WO PCT/JP1995/000920 patent/WO1995031200A1/en not_active Application Discontinuation
- 1995-05-15 HU HU9603158A patent/HUT76468A/hu unknown
- 1995-05-15 JP JP7529508A patent/JPH10500130A/ja active Pending
- 1995-05-15 CA CA002187361A patent/CA2187361A1/en not_active Abandoned
- 1995-05-15 PL PL95317190A patent/PL317190A1/xx unknown
- 1995-05-15 CN CN95193130A patent/CN1148810A/zh active Pending
- 1995-05-15 BR BR9507732A patent/BR9507732A/pt not_active Application Discontinuation
- 1995-05-15 EP EP95918186A patent/EP0759756A1/en not_active Withdrawn
- 1995-05-15 AU AU24201/95A patent/AU2420195A/en not_active Abandoned
- 1995-05-18 TW TW084104919A patent/TW304879B/zh active
Also Published As
| Publication number | Publication date |
|---|---|
| WO1995031200A1 (en) | 1995-11-23 |
| HUT76468A (en) | 1997-09-29 |
| CA2187361A1 (en) | 1995-11-23 |
| BR9507732A (pt) | 1997-08-19 |
| HU9603158D0 (en) | 1997-01-28 |
| EP0759756A1 (en) | 1997-03-05 |
| JPH10500130A (ja) | 1998-01-06 |
| PL317190A1 (en) | 1997-03-17 |
| TW304879B (enrdf_load_stackoverflow) | 1997-05-11 |
| CN1148810A (zh) | 1997-04-30 |
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