AU2019415174B2 - Method for producing amide - Google Patents

Method for producing amide Download PDF

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Publication number
AU2019415174B2
AU2019415174B2 AU2019415174A AU2019415174A AU2019415174B2 AU 2019415174 B2 AU2019415174 B2 AU 2019415174B2 AU 2019415174 A AU2019415174 A AU 2019415174A AU 2019415174 A AU2019415174 A AU 2019415174A AU 2019415174 B2 AU2019415174 B2 AU 2019415174B2
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AU
Australia
Prior art keywords
acid
reaction
producing
group
amide
Prior art date
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AU2019415174A
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English (en)
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AU2019415174A1 (en
Inventor
Shinichiro Fuse
Hiroyuki Nakamura
Yuma OTAKE
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Tokyo Institute of Technology NUC
Yokogawa Electric Corp
Original Assignee
Tokyo Institute of Technology NUC
Yokogawa Electric Corp
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Publication of AU2019415174A1 publication Critical patent/AU2019415174A1/en
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/02—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length in solution
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/02—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length in solution
    • C07K1/023—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length in solution using racemisation inhibiting agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Health & Medical Sciences (AREA)
  • Analytical Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Peptides Or Proteins (AREA)
AU2019415174A 2018-12-25 2019-12-11 Method for producing amide Active AU2019415174B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2018241598 2018-12-25
JP2018-241598 2018-12-25
PCT/JP2019/048458 WO2020137545A1 (ja) 2018-12-25 2019-12-11 アミドの製造方法

Publications (2)

Publication Number Publication Date
AU2019415174A1 AU2019415174A1 (en) 2021-07-29
AU2019415174B2 true AU2019415174B2 (en) 2022-08-11

Family

ID=71127982

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2019415174A Active AU2019415174B2 (en) 2018-12-25 2019-12-11 Method for producing amide

Country Status (6)

Country Link
US (1) US20220055984A1 (ja)
EP (1) EP3904317A4 (ja)
JP (1) JPWO2020137545A1 (ja)
CN (1) CN113227019A (ja)
AU (1) AU2019415174B2 (ja)
WO (1) WO2020137545A1 (ja)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023171671A1 (ja) * 2022-03-08 2023-09-14 国立大学法人東海国立大学機構 環状アミドの製造方法

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS62149699A (ja) * 1985-12-24 1987-07-03 Ajinomoto Co Inc Ｎ―ホルミル―α―Ｌ―アスパルチル―Ｌ―フェニルアラニンメチルエステルの製造法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZW6189A1 (en) * 1988-05-09 1990-05-09 Smithkline Beckman Corp Anti-aggregatory peptides
DE4242945A1 (de) * 1992-12-18 1994-06-23 Bayer Ag Neue acyclische, schwefelhaltige Peptide
DE10234422A1 (de) * 2002-07-29 2004-02-12 Bayer Ag Antibakterielle Ester-Makrozyklen

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS62149699A (ja) * 1985-12-24 1987-07-03 Ajinomoto Co Inc Ｎ―ホルミル―α―Ｌ―アスパルチル―Ｌ―フェニルアラニンメチルエステルの製造法

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
DUNETZ, J. R. et al., 'General and Scalable Amide Bond Formation with Epimerization-Prone Substrates Using T3P and Pyridine', Organic Letters. 2011, vol. 13, pages 5048–5051. *
Shinichiro Fuse , Yuto Mifune , Hiroyuki Nakamura , Hiroshi Tanaka, "Total synthesis of feglymycin based on a linear/convergent hybrid approach using micro-flow amide bond formation", Nature Communications, (2016-11-28), vol. 7, pages 1 - 7 *

Also Published As

Publication number Publication date
JPWO2020137545A1 (ja) 2021-11-04
WO2020137545A1 (ja) 2020-07-02
AU2019415174A1 (en) 2021-07-29
CN113227019A (zh) 2021-08-06
EP3904317A4 (en) 2022-09-21
US20220055984A1 (en) 2022-02-24
EP3904317A1 (en) 2021-11-03

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