AU2016360245B2 - Octahydropyrrolo [3, 4-c] pyrrole derivatives and uses thereof - Google Patents

Octahydropyrrolo [3, 4-c] pyrrole derivatives and uses thereof Download PDF

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AU2016360245B2
AU2016360245B2 AU2016360245A AU2016360245A AU2016360245B2 AU 2016360245 B2 AU2016360245 B2 AU 2016360245B2 AU 2016360245 A AU2016360245 A AU 2016360245A AU 2016360245 A AU2016360245 A AU 2016360245A AU 2016360245 B2 AU2016360245 B2 AU 2016360245B2
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compound
alkyl
alkoxy
disorder
alkylamino
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AU2016360245A1 (en
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Chuanfei JIN
Ji Zhang
Yingjun Zhang
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Sunshine Lake Pharma Co Ltd
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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AU2016360245A 2015-11-23 2016-11-23 Octahydropyrrolo [3, 4-c] pyrrole derivatives and uses thereof Active AU2016360245B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201510823712 2015-11-23
CN201510823712.8 2015-11-23
PCT/CN2016/106937 WO2017088759A1 (en) 2015-11-23 2016-11-23 OCTAHYDROPYRROLO [3, 4-c] PYRROLE DERIVATIVES AND USES THEREOF

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AU2016360245A1 AU2016360245A1 (en) 2018-06-07
AU2016360245B2 true AU2016360245B2 (en) 2020-07-09

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US (1) US10370380B2 (https=)
EP (1) EP3380475A4 (https=)
JP (1) JP6936224B2 (https=)
CN (1) CN106749269B (https=)
AU (1) AU2016360245B2 (https=)
CA (1) CA3005918C (https=)
SG (1) SG11201804223TA (https=)
WO (1) WO2017088759A1 (https=)

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CN109988171A (zh) * 2017-12-29 2019-07-09 广东东阳光药业有限公司 八氢吡咯并[3,4-c]吡咯衍生物及其用途
WO2020158415A1 (ja) * 2019-01-28 2020-08-06 サントリーホールディングス株式会社 オレキシン受容体拮抗阻害用組成物
WO2021104294A1 (en) * 2019-11-29 2021-06-03 Sunshine Lake Pharma Co., Ltd. CRYSTAL FORMS OF OCTAHYDROPYRROLO [3,4-c] PYRROLE DERIVATIVES
CN112876479B (zh) * 2019-11-29 2022-07-26 广东东阳光药业有限公司 八氢吡咯并[3,4-c]吡咯衍生物的晶型
CN112876481B (zh) * 2019-11-29 2022-07-26 广东东阳光药业有限公司 八氢吡咯并[3,4-c]吡咯衍生物的晶型
CN112876480B (zh) * 2019-11-29 2022-07-26 广东东阳光药业有限公司 八氢吡咯并[3,4-c]吡咯衍生物的晶型
CN112876478B (zh) * 2019-11-29 2022-07-26 广东东阳光药业有限公司 八氢吡咯并[3,4-c]吡咯衍生物的晶型
WO2022194122A1 (zh) * 2021-03-16 2022-09-22 上海翰森生物医药科技有限公司 含氮杂环的多环化合物及其制备方法和应用
CN116217593B (zh) * 2021-12-02 2025-05-09 江苏恩华药业股份有限公司 一种八氢吡咯并[3,4-c]吡咯甲基酮衍生物及其应用
KR20250065855A (ko) * 2022-09-14 2025-05-13 장쑤 한서 파마슈티칼 그룹 캄파니 리미티드 질소 함유 헤테로고리의 다환식 화합물의 유리 염기 결정형 및 이의 제조 방법
TW202428580A (zh) 2022-10-31 2024-07-16 日商武田藥品工業股份有限公司 雜環化合物
WO2024125395A1 (zh) * 2022-12-12 2024-06-20 江苏恩华药业股份有限公司 一种取代四氢环戊基[c]吡咯衍生物、制备方法、中间体及其应用
CN118580243B (zh) * 2024-08-07 2025-01-03 艾斯拓康生物医药(天津)有限公司 一类含氮并环化合物及其制备方法和应用

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