AU2014249233A1 - Compositions comprising thienopyrimidine and thienopyridine compounds and methods of use thereof - Google Patents

Compositions comprising thienopyrimidine and thienopyridine compounds and methods of use thereof Download PDF

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Publication number
AU2014249233A1
AU2014249233A1 AU2014249233A AU2014249233A AU2014249233A1 AU 2014249233 A1 AU2014249233 A1 AU 2014249233A1 AU 2014249233 A AU2014249233 A AU 2014249233A AU 2014249233 A AU2014249233 A AU 2014249233A AU 2014249233 A1 AU2014249233 A1 AU 2014249233A1
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Australia
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substituted
alkyl
group
pct
aromatic ring
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Abandoned
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AU2014249233A
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English (en)
Inventor
Dmitry Borkin
Tomasz Cierpicki
Jolanta Grembecka
Jay Hess
Xiaoqin LI
Duxin Sun
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University of Michigan System
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University of Michigan System
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/16—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Emergency Medicine (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Epidemiology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU2014249233A 2013-03-13 2014-03-10 Compositions comprising thienopyrimidine and thienopyridine compounds and methods of use thereof Abandoned AU2014249233A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361780099P 2013-03-13 2013-03-13
US61/780,099 2013-03-13
PCT/US2014/022750 WO2014164543A1 (en) 2013-03-13 2014-03-10 Compositions comprising thienopyrimidine and thienopyridine compounds and methods of use thereof

Publications (1)

Publication Number Publication Date
AU2014249233A1 true AU2014249233A1 (en) 2015-09-24

Family

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Family Applications (1)

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AU2014249233A Abandoned AU2014249233A1 (en) 2013-03-13 2014-03-10 Compositions comprising thienopyrimidine and thienopyridine compounds and methods of use thereof

Country Status (11)

Country Link
US (4) US9216993B2 (enExample)
EP (1) EP2968342B1 (enExample)
JP (2) JP2016512514A (enExample)
KR (1) KR20150130389A (enExample)
CN (1) CN105188705A (enExample)
AU (1) AU2014249233A1 (enExample)
BR (1) BR112015022602A2 (enExample)
CA (1) CA2904612A1 (enExample)
IL (1) IL241193A0 (enExample)
MX (1) MX2015011576A (enExample)
WO (1) WO2014164543A1 (enExample)

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Also Published As

Publication number Publication date
EP2968342A4 (en) 2016-07-27
US10160769B2 (en) 2018-12-25
US9505782B2 (en) 2016-11-29
US9505781B2 (en) 2016-11-29
US20140275070A1 (en) 2014-09-18
JP2018115214A (ja) 2018-07-26
KR20150130389A (ko) 2015-11-23
US9216993B2 (en) 2015-12-22
CN105188705A (zh) 2015-12-23
US20170253611A1 (en) 2017-09-07
US20160046647A1 (en) 2016-02-18
BR112015022602A2 (pt) 2017-07-18
CA2904612A1 (en) 2014-10-09
WO2014164543A1 (en) 2014-10-09
MX2015011576A (es) 2016-05-16
IL241193A0 (en) 2015-11-30
JP6670885B2 (ja) 2020-03-25
EP2968342A1 (en) 2016-01-20
US20160137665A1 (en) 2016-05-19
JP2016512514A (ja) 2016-04-28
EP2968342B1 (en) 2018-10-03

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