AU2013340345B2 - Bruton's tyrosine kinase inhibitors - Google Patents

Bruton's tyrosine kinase inhibitors Download PDF

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Publication number
AU2013340345B2
AU2013340345B2 AU2013340345A AU2013340345A AU2013340345B2 AU 2013340345 B2 AU2013340345 B2 AU 2013340345B2 AU 2013340345 A AU2013340345 A AU 2013340345A AU 2013340345 A AU2013340345 A AU 2013340345A AU 2013340345 B2 AU2013340345 B2 AU 2013340345B2
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Australia
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halo
alkyl
alkoxy
compound
independently selected
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Ceased
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AU2013340345A
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AU2013340345A1 (en
Inventor
Balekudru Devadas
Danny James GARLAND
Margaret Lanahan Grapperhaus
Seungil Han
Susan Landis Hockerman
Robert Owen Hughes
Eddine Saiah
Michelle Ann Schmidt
Mark Edward SCHNUTE
Shaun Raj Selness
John Robert Springer
Daniel Patrick Walker
Zhao-Kui Wan
Li Xing
Christoph Wolfgang ZAPF
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Pfizer Inc
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Pfizer Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49596360&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2013340345(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of AU2013340345A1 publication Critical patent/AU2013340345A1/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epidemiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU2013340345A 2012-11-02 2013-11-01 Bruton's tyrosine kinase inhibitors Ceased AU2013340345B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261721920P 2012-11-02 2012-11-02
US61/721,920 2012-11-02
US201361772028P 2013-03-04 2013-03-04
US61/772,028 2013-03-04
PCT/IB2013/059846 WO2014068527A1 (en) 2012-11-02 2013-11-01 Bruton's tyrosine kinase inhibitors

Publications (2)

Publication Number Publication Date
AU2013340345A1 AU2013340345A1 (en) 2015-04-30
AU2013340345B2 true AU2013340345B2 (en) 2016-10-27

Family

ID=49596360

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2013340345A Ceased AU2013340345B2 (en) 2012-11-02 2013-11-01 Bruton's tyrosine kinase inhibitors

Country Status (27)

Country Link
US (4) US20150291554A1 (enExample)
EP (1) EP2914586B1 (enExample)
JP (1) JP6178861B2 (enExample)
KR (1) KR101668574B1 (enExample)
CN (1) CN105008344B (enExample)
AP (1) AP2015008381A0 (enExample)
AU (1) AU2013340345B2 (enExample)
BR (1) BR112015009624A2 (enExample)
CA (1) CA2888960C (enExample)
CL (1) CL2015001168A1 (enExample)
CO (1) CO7350624A2 (enExample)
CR (1) CR20150228A (enExample)
DO (1) DOP2015000100A (enExample)
EA (1) EA201500393A1 (enExample)
ES (1) ES2625944T3 (enExample)
GE (1) GEP201606597B (enExample)
HK (1) HK1211293A1 (enExample)
IL (1) IL238571A0 (enExample)
MD (1) MD20150035A2 (enExample)
MX (1) MX2015005422A (enExample)
NI (1) NI201500059A (enExample)
PE (1) PE20151070A1 (enExample)
PH (1) PH12015500940A1 (enExample)
SG (1) SG11201502893WA (enExample)
TN (1) TN2015000168A1 (enExample)
TW (1) TWI518080B (enExample)
WO (1) WO2014068527A1 (enExample)

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JP2015535277A (ja) 2015-12-10
EP2914586B1 (en) 2017-04-05
US10266513B2 (en) 2019-04-23
IL238571A0 (en) 2015-06-30
ES2625944T3 (es) 2017-07-21
TW201431851A (zh) 2014-08-16
TWI518080B (zh) 2016-01-21
JP6178861B2 (ja) 2017-08-09
HK1211293A1 (en) 2016-05-20
PH12015500940A1 (en) 2015-06-29
CR20150228A (es) 2015-09-14
CL2015001168A1 (es) 2015-07-10
US20170283393A1 (en) 2017-10-05
CA2888960C (en) 2017-08-15
CO7350624A2 (es) 2015-08-10
EP2914586A1 (en) 2015-09-09
MX2015005422A (es) 2015-08-05
CN105008344A (zh) 2015-10-28
AP2015008381A0 (en) 2015-04-30
DOP2015000100A (es) 2015-12-31
CN105008344B (zh) 2017-07-25
KR101668574B1 (ko) 2016-10-24
CA2888960A1 (en) 2014-05-08
PE20151070A1 (es) 2015-08-01
WO2014068527A1 (en) 2014-05-08
US20190202798A1 (en) 2019-07-04
MD20150035A2 (ro) 2015-10-31
SG11201502893WA (en) 2015-05-28
AU2013340345A1 (en) 2015-04-30
EA201500393A1 (ru) 2016-05-31
GEP201606597B (en) 2017-01-10
NI201500059A (es) 2015-06-05
TN2015000168A1 (fr) 2016-10-03
US20210002251A1 (en) 2021-01-07
US20150291554A1 (en) 2015-10-15
US10815213B2 (en) 2020-10-27
BR112015009624A2 (pt) 2017-11-14
KR20150075114A (ko) 2015-07-02

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