AU2008230710B2 - The use of PDE7 inhibitors for the treatment of movement disorders - Google Patents
The use of PDE7 inhibitors for the treatment of movement disorders Download PDFInfo
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- AU2008230710B2 AU2008230710B2 AU2008230710A AU2008230710A AU2008230710B2 AU 2008230710 B2 AU2008230710 B2 AU 2008230710B2 AU 2008230710 A AU2008230710 A AU 2008230710A AU 2008230710 A AU2008230710 A AU 2008230710A AU 2008230710 B2 AU2008230710 B2 AU 2008230710B2
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- pde7
- alkyl
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- inhibiting
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Classifications
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/527—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim spiro-condensed
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- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
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- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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Landscapes
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Investigating Or Analysing Biological Materials (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
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| AU2013202067A AU2013202067B2 (en) | 2007-03-27 | 2013-03-22 | The use of PDE7 inhibitors for the treatment of movement disorders |
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| US92049607P | 2007-03-27 | 2007-03-27 | |
| US60/920,496 | 2007-03-27 | ||
| PCT/US2008/058530 WO2008119057A2 (en) | 2007-03-27 | 2008-03-27 | The use of pde7 inhibitors for the treatment of movement disorders |
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| EP (1) | EP2139475B1 (OSRAM) |
| JP (2) | JP5580192B2 (OSRAM) |
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| US8637528B2 (en) | 2007-03-27 | 2014-01-28 | Omeros Corporation | Use of PDE7 inhibitors for the treatment of movement disorders |
| WO2010111060A1 (en) * | 2009-03-23 | 2010-09-30 | Merck Sharp & Dohme Corp. | P2x3, receptor antagonists for treatment of pain |
| FR2943673B1 (fr) * | 2009-03-27 | 2013-03-29 | Sanofi Aventis | Applications therapeutiques de derives de quinazolinedione |
| FR2944282B1 (fr) | 2009-04-09 | 2013-05-03 | Sanofi Aventis | Derives de quinazolinedione, leur preparation et leurs diverses applications therapeutiques |
| FR2944206B1 (fr) | 2009-04-09 | 2012-12-28 | Sanofi Aventis | Applications therapeutiques dans le domaine cardiovasculaire de derives de quinazolinedione |
| AU2013202493B2 (en) * | 2009-05-04 | 2016-03-10 | Omeros Corporation | Use of PDE7 inhibitors for the treatment of movement disorders |
| ES2353093B1 (es) | 2009-05-20 | 2012-01-03 | Consejo Superior De Investigaciones Científicas (Csic) | Uso de derivados de quinazolinas y sus composiciones farmacéuticas en enfermedades neurodegenerativas. |
| ES2360783B1 (es) | 2009-10-02 | 2012-07-04 | Consejo Superior De Investigaciones Científicas (Csic) | 1,2,4-tiadiazoles-5-imino sustituidos utiles en el tratamiento de enfermedades neurodegenerativas |
| US9220715B2 (en) | 2010-11-08 | 2015-12-29 | Omeros Corporation | Treatment of addiction and impulse-control disorders using PDE7 inhibitors |
| MX2013004943A (es) | 2010-11-08 | 2013-09-02 | Omeros Corp | Tratamiento de trastornos de adicion y control de impulsos usando inhibidores de pde7. |
| HRP20190279T1 (hr) * | 2012-05-07 | 2019-04-05 | Omeros Corporation | Liječenje ovisnosti i poremećaja nagona pomoću pde7 inhibitora |
| EP2846805B1 (en) * | 2012-05-07 | 2018-11-21 | Omeros Corporation | Treatment of addiction and impulse-control disorders using pde7 inhibitors |
| US20190185479A1 (en) * | 2016-08-26 | 2019-06-20 | Mitsubishi Tanabe Pharma Corporation | Bicyclic nitrogenated heterocyclic compound |
| JP2021535180A (ja) * | 2018-09-05 | 2021-12-16 | ユニベルシテイト ファン アムステルダム | パーキンソン病の処置の為のｐｄｅ１１又はｐｄｅ２阻害剤の使用 |
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| WO2024259383A2 (en) * | 2023-06-14 | 2024-12-19 | President And Fellows Of Harvard College | Ion channel binders and uses thereof |
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2008
- 2008-03-27 NZ NZ580413A patent/NZ580413A/xx unknown
- 2008-03-27 CN CN200880017058XA patent/CN101917992A/zh active Pending
- 2008-03-27 RU RU2009138966/15A patent/RU2449790C2/ru active
- 2008-03-27 CN CN201510082785.6A patent/CN104758291B/zh active Active
- 2008-03-27 JP JP2010501232A patent/JP5580192B2/ja active Active
- 2008-03-27 EP EP08744515.1A patent/EP2139475B1/en active Active
- 2008-03-27 MX MX2009010450A patent/MX2009010450A/es active IP Right Grant
- 2008-03-27 AU AU2008230710A patent/AU2008230710B2/en active Active
- 2008-03-27 WO PCT/US2008/058530 patent/WO2008119057A2/en not_active Ceased
- 2008-03-27 US US12/057,368 patent/US20080260643A1/en not_active Abandoned
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- 2008-03-27 ES ES08744515.1T patent/ES2533206T3/es active Active
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2010
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2014
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2018
- 2018-12-06 US US16/212,064 patent/US20190183824A1/en not_active Abandoned
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| US20030069169A1 (en) * | 2001-03-02 | 2003-04-10 | Macor John E. | Co-administration of melanocortin receptor agonist and phosphodiesterase inhibitor for treatment of cyclic-AMP associated disorders |
Also Published As
| Publication number | Publication date |
|---|---|
| NZ580413A (en) | 2012-11-30 |
| RU2009138966A (ru) | 2011-05-10 |
| CN104758291B (zh) | 2020-03-03 |
| US20080260643A1 (en) | 2008-10-23 |
| MX2009010450A (es) | 2009-11-23 |
| RU2449790C2 (ru) | 2012-05-10 |
| ES2533206T3 (es) | 2015-04-08 |
| US20110091388A1 (en) | 2011-04-21 |
| WO2008119057A3 (en) | 2008-11-20 |
| JP5580192B2 (ja) | 2014-08-27 |
| AU2008230710A1 (en) | 2008-10-02 |
| CA2681650A1 (en) | 2008-10-02 |
| CN101917992A (zh) | 2010-12-15 |
| HK1139861A1 (en) | 2010-09-30 |
| JP2014198718A (ja) | 2014-10-23 |
| US20190183824A1 (en) | 2019-06-20 |
| EP2139475A2 (en) | 2010-01-06 |
| BRPI0809244A2 (pt) | 2014-09-23 |
| EP2139475A4 (en) | 2012-03-07 |
| CN104758291A (zh) | 2015-07-08 |
| JP5943964B2 (ja) | 2016-07-05 |
| JP2010522768A (ja) | 2010-07-08 |
| CA2681650C (en) | 2016-11-22 |
| WO2008119057A2 (en) | 2008-10-02 |
| EP2139475B1 (en) | 2014-12-17 |
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