AU2004203983A1 - Process for the preparation of aryl fused polycyclic lactams - Google Patents

Process for the preparation of aryl fused polycyclic lactams Download PDF

Info

Publication number
AU2004203983A1
AU2004203983A1 AU2004203983A AU2004203983A AU2004203983A1 AU 2004203983 A1 AU2004203983 A1 AU 2004203983A1 AU 2004203983 A AU2004203983 A AU 2004203983A AU 2004203983 A AU2004203983 A AU 2004203983A AU 2004203983 A1 AU2004203983 A1 AU 2004203983A1
Authority
AU
Australia
Prior art keywords
formula
triene
aza
dodeca
tricyclo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2004203983A
Other languages
English (en)
Inventor
Jr. Robert Eugene Handfield
Timothy James Norman Watson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of AU2004203983A1 publication Critical patent/AU2004203983A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22—Bridged ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22—Bridged ring systems
    • C07D221/26—Benzomorphans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
AU2004203983A 2003-01-15 2004-01-08 Process for the preparation of aryl fused polycyclic lactams Abandoned AU2004203983A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US44026603P 2003-01-15 2003-01-15
US60/440,266 2003-01-15
PCT/IB2004/000152 WO2004063164A1 (en) 2003-01-15 2004-01-08 Process for the preparation of aryl fused polycyclic lactams

Publications (1)

Publication Number Publication Date
AU2004203983A1 true AU2004203983A1 (en) 2004-07-29

Family

ID=32713537

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2004203983A Abandoned AU2004203983A1 (en) 2003-01-15 2004-01-08 Process for the preparation of aryl fused polycyclic lactams

Country Status (18)

Country Link
US (1) US20070066827A1 (enExample)
EP (1) EP1587794A1 (enExample)
JP (1) JP2006517202A (enExample)
KR (2) KR20050101177A (enExample)
CN (1) CN100363350C (enExample)
AR (1) AR042855A1 (enExample)
AU (1) AU2004203983A1 (enExample)
BR (1) BRPI0406670A (enExample)
CA (1) CA2513293A1 (enExample)
CL (1) CL2004000041A1 (enExample)
IL (1) IL169479A0 (enExample)
MX (1) MXPA05007565A (enExample)
PL (1) PL379373A1 (enExample)
RS (1) RS20050513A (enExample)
RU (1) RU2291862C2 (enExample)
TW (1) TW200420286A (enExample)
WO (1) WO2004063164A1 (enExample)
ZA (1) ZA200505103B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2284319C2 (ru) 2002-11-25 2006-09-27 Пфайзер Продактс Инк. Усовершенствованный способ получения 1,3-замещенных инденов
RU2372323C1 (ru) * 2008-04-15 2009-11-10 Открытое акционерное общество Научно-производственное предприятие НИИПАВ (ОАО НПП НИИПАВ) Способ получения высокомолекулярных аминов
US8039620B2 (en) * 2008-05-22 2011-10-18 Teva Pharmaceutical Industries Ltd. Varenicline tosylate, an intermediate in the preparation process of varenicline L-tartrate
US20090318695A1 (en) * 2008-06-19 2009-12-24 Vinod Kumar Kansal Processes for the preparation of varenicline and intermediates thereof
US8178537B2 (en) * 2009-06-22 2012-05-15 Teva Pharmaceutical Industries Ltd. Solid state forms of varenicline salts and processes for preparation thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ271765A (en) * 1993-08-05 1996-11-26 Syntex Inc Bridged [1,3]indolo macrocyclic lactam compounds and pharmaceutical compositions
ATE386024T1 (de) * 1997-12-31 2008-03-15 Pfizer Prod Inc Arylkondensierte azapolycyclische derivate
US6605610B1 (en) * 1997-12-31 2003-08-12 Pfizer Inc Aryl fused azapolycyclic compounds
DK1383733T3 (da) * 2001-04-20 2008-06-09 Pfizer Prod Inc Fremgangsmåde til fremstilling af 1,3-substituerede indener og aryl-sammenföjede azapolycykliske forbindelser

Also Published As

Publication number Publication date
CA2513293A1 (en) 2004-07-29
MXPA05007565A (es) 2005-09-21
ZA200505103B (en) 2006-11-29
CL2004000041A1 (es) 2005-04-22
JP2006517202A (ja) 2006-07-20
CN1738803A (zh) 2006-02-22
IL169479A0 (en) 2007-07-04
RU2005122406A (ru) 2006-01-27
WO2004063164A8 (en) 2005-05-26
AR042855A1 (es) 2005-07-06
WO2004063164A1 (en) 2004-07-29
HK1085204A1 (zh) 2006-08-18
KR20070087258A (ko) 2007-08-27
KR20050101177A (ko) 2005-10-20
EP1587794A1 (en) 2005-10-26
PL379373A1 (pl) 2006-08-21
TW200420286A (en) 2004-10-16
RU2291862C2 (ru) 2007-01-20
RS20050513A (sr) 2007-11-15
US20070066827A1 (en) 2007-03-22
CN100363350C (zh) 2008-01-23
BRPI0406670A (pt) 2005-12-20

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Legal Events

Date Code Title Description
MK4 Application lapsed section 142(2)(d) - no continuation fee paid for the application