AU2003299472A1 - Thiadiazoles or oxadiazoles and their use as inhibitors of JAK kinase - Google Patents
Thiadiazoles or oxadiazoles and their use as inhibitors of JAK kinase Download PDFInfo
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- AU2003299472A1 AU2003299472A1 AU2003299472A AU2003299472A AU2003299472A1 AU 2003299472 A1 AU2003299472 A1 AU 2003299472A1 AU 2003299472 A AU2003299472 A AU 2003299472A AU 2003299472 A AU2003299472 A AU 2003299472A AU 2003299472 A1 AU2003299472 A1 AU 2003299472A1
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Classifications
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
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Landscapes
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Applications Claiming Priority (3)
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| DE102004009933A1 (de) * | 2004-02-26 | 2005-09-15 | Merck Patent Gmbh | Verwendung von Thiadiazolharnstoffderivaten |
| US7550499B2 (en) | 2004-05-12 | 2009-06-23 | Bristol-Myers Squibb Company | Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions |
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| CN108148058B (zh) * | 2018-02-08 | 2021-03-16 | 中国人民解放军第四军医大学 | 一种4-(2-巯基噻二唑)取代的嘧啶衍生物其制备方法及应用 |
| EA202192575A1 (ru) | 2019-03-21 | 2022-01-14 | Онксео | Соединения dbait в сочетании с ингибиторами киназ для лечения рака |
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| CN114761006A (zh) | 2019-11-08 | 2022-07-15 | Inserm(法国国家健康医学研究院) | 对激酶抑制剂产生耐药性的癌症的治疗方法 |
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| WO2000075145A1 (en) * | 1999-06-03 | 2000-12-14 | Abbott Laboratories | Cell adhesion-inhibiting antiinflammatory compounds |
| JP2001354658A (ja) * | 2000-06-15 | 2001-12-25 | Taisho Pharmaceut Co Ltd | ヒドロキシホルムアミジン化合物及びその塩並びにそれらを含む医薬 |
| IL153246A0 (en) * | 2000-06-28 | 2003-07-06 | Astrazeneca Ab | Substituted quinazoline derivatives and their use as inhibitors |
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2003
- 2003-05-06 RU RU2004135386/04A patent/RU2004135386A/ru not_active Application Discontinuation
- 2003-05-06 KR KR10-2004-7017933A patent/KR20050006237A/ko not_active Withdrawn
- 2003-05-06 WO PCT/US2003/014223 patent/WO2004058753A1/en not_active Ceased
- 2003-05-06 US US10/430,805 patent/US7271179B2/en not_active Expired - Fee Related
- 2003-05-06 CA CA002485429A patent/CA2485429A1/en not_active Abandoned
- 2003-05-06 AU AU2003299472A patent/AU2003299472A1/en not_active Withdrawn
- 2003-05-06 EP EP10182153A patent/EP2316834A1/en not_active Withdrawn
- 2003-05-06 EP EP03799762A patent/EP1501829B1/en not_active Expired - Lifetime
- 2003-05-06 CN CN038159546A patent/CN1665808A/zh active Pending
- 2003-05-06 AT AT03799762T patent/ATE489384T1/de not_active IP Right Cessation
- 2003-05-06 DE DE60335099T patent/DE60335099D1/de not_active Expired - Lifetime
- 2003-05-06 MX MXPA04011048A patent/MXPA04011048A/es unknown
- 2003-05-06 JP JP2004563181A patent/JP4681302B2/ja not_active Expired - Fee Related
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2004
- 2004-11-07 IL IL16506704A patent/IL165067A0/xx unknown
- 2004-12-02 NO NO20045282A patent/NO20045282L/no not_active Application Discontinuation
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- 2010-04-26 JP JP2010101525A patent/JP2010159306A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004058753A8 (en) | 2005-06-16 |
| CN1665808A (zh) | 2005-09-07 |
| JP2006513192A (ja) | 2006-04-20 |
| CA2485429A1 (en) | 2004-07-15 |
| WO2004058753A1 (en) | 2004-07-15 |
| DE60335099D1 (de) | 2011-01-05 |
| IL165067A0 (en) | 2005-12-18 |
| US20040038992A1 (en) | 2004-02-26 |
| KR20050006237A (ko) | 2005-01-15 |
| EP2316834A1 (en) | 2011-05-04 |
| NO20045282L (no) | 2005-02-07 |
| EP1501829B1 (en) | 2010-11-24 |
| ATE489384T1 (de) | 2010-12-15 |
| MXPA04011048A (es) | 2005-02-17 |
| JP4681302B2 (ja) | 2011-05-11 |
| US7271179B2 (en) | 2007-09-18 |
| EP1501829A1 (en) | 2005-02-02 |
| RU2004135386A (ru) | 2005-07-20 |
| JP2010159306A (ja) | 2010-07-22 |
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