AU2003296414A1 - Method of using aminocyanopyridine compounds as mitogen activated protein kinase-activated protein kinase-2 inhibitors - Google Patents

Method of using aminocyanopyridine compounds as mitogen activated protein kinase-activated protein kinase-2 inhibitors

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Publication number
AU2003296414A1
AU2003296414A1 AU2003296414A AU2003296414A AU2003296414A1 AU 2003296414 A1 AU2003296414 A1 AU 2003296414A1 AU 2003296414 A AU2003296414 A AU 2003296414A AU 2003296414 A AU2003296414 A AU 2003296414A AU 2003296414 A1 AU2003296414 A1 AU 2003296414A1
Authority
AU
Australia
Prior art keywords
protein kinase
activated protein
inhibitors
mitogen
aminocyanopyridine compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003296414A
Other languages
English (en)
Other versions
AU2003296414A8 (en
Inventor
David R. Anderson
Shridhar G. Hegde
Stephen A. Kolodziej
Len F. Lee
Emily J. Reinhard
Nathan W. Stehle
William F. Vernier
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia LLC
Original Assignee
Pharmacia LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia LLC filed Critical Pharmacia LLC
Publication of AU2003296414A8 publication Critical patent/AU2003296414A8/xx
Publication of AU2003296414A1 publication Critical patent/AU2003296414A1/en
Abandoned legal-status Critical Current

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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  • Health & Medical Sciences (AREA)
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  • Veterinary Medicine (AREA)
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  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Molecular Biology (AREA)
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  • Reproductive Health (AREA)
  • Psychiatry (AREA)
  • AIDS & HIV (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
AU2003296414A 2002-12-12 2003-12-09 Method of using aminocyanopyridine compounds as mitogen activated protein kinase-activated protein kinase-2 inhibitors Abandoned AU2003296414A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US43280702P 2002-12-12 2002-12-12
US60/432,807 2002-12-12
PCT/US2003/039166 WO2004054505A2 (fr) 2002-12-12 2003-12-09 Procede d'utilisation de composes d'aminocyanopyridine en tant qu'inhibiteurs de la proteine mapkap kinase-2

Publications (2)

Publication Number Publication Date
AU2003296414A8 AU2003296414A8 (en) 2004-07-09
AU2003296414A1 true AU2003296414A1 (en) 2004-07-09

Family

ID=32595087

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003296414A Abandoned AU2003296414A1 (en) 2002-12-12 2003-12-09 Method of using aminocyanopyridine compounds as mitogen activated protein kinase-activated protein kinase-2 inhibitors

Country Status (7)

Country Link
EP (1) EP1569645A2 (fr)
JP (1) JP2006512338A (fr)
AU (1) AU2003296414A1 (fr)
BR (1) BR0317183A (fr)
CA (1) CA2508780A1 (fr)
MX (1) MXPA05006367A (fr)
WO (1) WO2004054505A2 (fr)

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CN102762206A (zh) * 2009-12-15 2012-10-31 诺华有限公司 免疫增强化合物的均匀悬液及其用途
HRP20211752T1 (hr) 2010-04-07 2022-02-18 Vertex Pharmaceuticals Incorporated Farmaceutski pripravci 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioksol-5-il)ciklopropankarboksamido)-3-metilpiridin-2-il)benzojeve kiseline i njihova primjena
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