AU2003287077B2 - Methylene-bridged selective androgen receptor modulators and methods of use thereof - Google Patents
Methylene-bridged selective androgen receptor modulators and methods of use thereof Download PDFInfo
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- AU2003287077B2 AU2003287077B2 AU2003287077A AU2003287077A AU2003287077B2 AU 2003287077 B2 AU2003287077 B2 AU 2003287077B2 AU 2003287077 A AU2003287077 A AU 2003287077A AU 2003287077 A AU2003287077 A AU 2003287077A AU 2003287077 B2 AU2003287077 B2 AU 2003287077B2
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- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
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- C07C235/32—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
- C07C235/38—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
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Landscapes
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- Dermatology (AREA)
- Biomedical Technology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
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| US41816602P | 2002-10-15 | 2002-10-15 | |
| US60/418,166 | 2002-10-15 | ||
| PCT/US2003/032511 WO2004035738A2 (en) | 2002-10-15 | 2003-10-14 | Methylene-bridged selective androgen receptor modulators and methods of use thereof |
Publications (2)
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| AU2003287077A1 AU2003287077A1 (en) | 2004-05-04 |
| AU2003287077B2 true AU2003287077B2 (en) | 2007-09-20 |
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| EP (1) | EP1562594A4 (enExample) |
| JP (1) | JP2006506369A (enExample) |
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| CA (1) | CA2502209A1 (enExample) |
| TW (1) | TW200503711A (enExample) |
| WO (1) | WO2004035738A2 (enExample) |
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| US8445534B2 (en) | 2000-08-24 | 2013-05-21 | University Of Tennessee Research Foundation | Treating androgen decline in aging male (ADAM)-associated conditions with SARMs |
| US7622503B2 (en) | 2000-08-24 | 2009-11-24 | University Of Tennessee Research Foundation | Selective androgen receptor modulators and methods of use thereof |
| AU2006200749A1 (en) * | 2000-08-24 | 2006-03-16 | University Of Tennessee Research Foundation | Halogenated selective androgen receptor modulators and methods of use thereof |
| US7919647B2 (en) | 2000-08-24 | 2011-04-05 | University Of Tennessee Research Foundation | Selective androgen receptor modulators and methods of use thereof |
| US7855229B2 (en) | 2000-08-24 | 2010-12-21 | University Of Tennessee Research Foundation | Treating wasting disorders with selective androgen receptor modulators |
| US7645898B2 (en) | 2000-08-24 | 2010-01-12 | University Of Tennessee Research Foundation | Selective androgen receptor modulators and method of use thereof |
| US8853266B2 (en) | 2001-12-06 | 2014-10-07 | University Of Tennessee Research Foundation | Selective androgen receptor modulators for treating diabetes |
| WO2004034978A2 (en) * | 2002-10-15 | 2004-04-29 | Gtx, Inc. | Treating obesity with selective androgen receptor modulators |
| CA2514024A1 (en) * | 2003-01-22 | 2004-08-05 | Gtx Inc. | Treating androgen deficiency in female (adif)-associated conditions with sarms |
| US9884038B2 (en) | 2004-06-07 | 2018-02-06 | University Of Tennessee Research Foundation | Selective androgen receptor modulator and methods of use thereof |
| US9889110B2 (en) | 2004-06-07 | 2018-02-13 | University Of Tennessee Research Foundation | Selective androgen receptor modulator for treating hormone-related conditions |
| US9492400B2 (en) | 2004-11-04 | 2016-11-15 | Massachusetts Institute Of Technology | Coated controlled release polymer particles as efficient oral delivery vehicles for biopharmaceuticals |
| CN101146535A (zh) * | 2005-03-25 | 2008-03-19 | 默克公司 | 用睾酮补充剂和5α-还原酶抑制剂治疗男性病人的方法 |
| US9267937B2 (en) | 2005-12-15 | 2016-02-23 | Massachusetts Institute Of Technology | System for screening particles |
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- 2003-10-14 AU AU2003287077A patent/AU2003287077B2/en not_active Ceased
- 2003-10-14 JP JP2004544890A patent/JP2006506369A/ja active Pending
- 2003-10-14 CN CNA2003801061426A patent/CN1726034A/zh active Pending
- 2003-10-14 US US10/683,157 patent/US7253210B2/en not_active Expired - Lifetime
- 2003-10-14 WO PCT/US2003/032511 patent/WO2004035738A2/en not_active Ceased
- 2003-10-14 CA CA002502209A patent/CA2502209A1/en not_active Abandoned
- 2003-10-14 EP EP03777598A patent/EP1562594A4/en not_active Withdrawn
- 2003-10-15 TW TW092128551A patent/TW200503711A/zh unknown
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2007
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| EP0253503A2 (en) * | 1986-07-18 | 1988-01-20 | Imperial Chemical Industries Plc | Substituted anilides having antiandrogenic properties |
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| WO2004035738A2 (en) | 2004-04-29 |
| EP1562594A2 (en) | 2005-08-17 |
| CN1726034A (zh) | 2006-01-25 |
| TW200503711A (en) | 2005-02-01 |
| US20080319009A1 (en) | 2008-12-25 |
| EP1562594A4 (en) | 2008-12-17 |
| JP2006506369A (ja) | 2006-02-23 |
| US20040147550A1 (en) | 2004-07-29 |
| CA2502209A1 (en) | 2004-04-29 |
| WO2004035738A3 (en) | 2004-07-15 |
| US7253210B2 (en) | 2007-08-07 |
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