AU2003271117A1 - Novel pyrazole compounds having antifungal activity - Google Patents
Novel pyrazole compounds having antifungal activityInfo
- Publication number
- AU2003271117A1 AU2003271117A1 AU2003271117A AU2003271117A AU2003271117A1 AU 2003271117 A1 AU2003271117 A1 AU 2003271117A1 AU 2003271117 A AU2003271117 A AU 2003271117A AU 2003271117 A AU2003271117 A AU 2003271117A AU 2003271117 A1 AU2003271117 A1 AU 2003271117A1
- Authority
- AU
- Australia
- Prior art keywords
- antifungal activity
- pyrazole compounds
- novel pyrazole
- novel
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2002296127 | 2002-10-09 | ||
| JP2002-296127 | 2002-10-09 | ||
| PCT/JP2003/012856 WO2004033432A1 (ja) | 2002-10-09 | 2003-10-08 | 抗真菌活性を有する新規ピラゾール化合物 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2003271117A1 true AU2003271117A1 (en) | 2004-05-04 |
Family
ID=32089230
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2003271117A Abandoned AU2003271117A1 (en) | 2002-10-09 | 2003-10-08 | Novel pyrazole compounds having antifungal activity |
Country Status (4)
| Country | Link |
|---|---|
| JP (1) | JP4537855B2 (ja) |
| AU (1) | AU2003271117A1 (ja) |
| TW (1) | TW200418804A (ja) |
| WO (1) | WO2004033432A1 (ja) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8829198B2 (en) * | 2007-10-31 | 2014-09-09 | Proteotech Inc | Compounds, compositions and methods for the treatment of beta-amyloid diseases and synucleinopathies |
| US7932272B2 (en) | 2003-09-30 | 2011-04-26 | Eisai R&D Management Co., Ltd. | Antifungal agent containing heterocyclic compound |
| WO2006044528A1 (en) * | 2004-10-15 | 2006-04-27 | Memory Pharmaceuticals Corporation | Pyrazole derivatives as phosphodiesterase 4 inhibitors |
| US7829585B2 (en) | 2005-03-30 | 2010-11-09 | Eisai R&D Management Co., Ltd. | Antifungal agent containing pyridine derivative |
| CA2613522A1 (en) | 2005-06-27 | 2007-01-04 | Exelixis, Inc. | Imidazole based lxr modulators |
| WO2007052615A1 (ja) | 2005-10-31 | 2007-05-10 | Eisai R & D Management Co., Ltd. | ヘテロ環置換ピリジン誘導体およびそれらを含有する抗真菌剤 |
| TWI385169B (zh) | 2005-10-31 | 2013-02-11 | Eisai R&D Man Co Ltd | 經雜環取代之吡啶衍生物及含有彼之抗真菌劑 |
| US8183264B2 (en) | 2006-09-21 | 2012-05-22 | Eisai R&D Managment Co., Ltd. | Pyridine derivative substituted by heteroaryl ring, and antifungal agent comprising the same |
| US20100105729A1 (en) * | 2006-10-06 | 2010-04-29 | Kalypsys, Inc. | Aryl-substituted heterocyclic pde4 inhibitors as anti-inflammatory agents |
| CN101679297B (zh) | 2006-12-08 | 2012-01-11 | 埃克塞利希斯股份有限公司 | Lxr和fxr调节剂 |
| TW200841879A (en) | 2007-04-27 | 2008-11-01 | Eisai R&D Man Co Ltd | Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same |
| CN102702185A (zh) | 2007-04-27 | 2012-10-03 | 卫材R&D管理有限公司 | 杂环取代吡啶衍生物的盐的结晶 |
| US8513287B2 (en) | 2007-12-27 | 2013-08-20 | Eisai R&D Management Co., Ltd. | Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same |
| ES2714453T3 (es) * | 2008-06-09 | 2019-05-28 | Univ Muenchen Ludwig Maximilians | Fármacos para inhibir la agregación de proteínas implicadas en enfermedades relacionadas con enfermedades neurodegenerativas y/o agregación de proteínas |
| AU2009272033B2 (en) | 2008-07-17 | 2011-10-13 | Asahi Kasei Pharma Corporation | Nitrogenated heterocyclic compound |
| US8188119B2 (en) | 2008-10-24 | 2012-05-29 | Eisai R&D Management Co., Ltd | Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same |
| CN101928246B (zh) * | 2009-10-16 | 2013-02-27 | 天津理工大学 | N-[(1-芳基-3-取代苯基-吡唑-4-基)次甲基]-2-羟基苯甲酰肼类化合物或其可药用盐及制备 |
| SG192582A1 (en) * | 2011-01-30 | 2013-09-30 | Meiji Seika Pharma Co Ltd | Topical antifungal agent |
| JP6132842B2 (ja) * | 2012-07-30 | 2017-05-24 | Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 | 抗白癬菌症外用液剤 |
| WO2014021284A1 (ja) | 2012-07-30 | 2014-02-06 | Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 | 抗白癬菌症貼付剤 |
| EP2885293B1 (en) * | 2012-08-16 | 2016-07-27 | Janssen Pharmaceutica, N.V. | Substituted pyrazoles as n-type calcium channel blockers |
| US9453002B2 (en) | 2013-08-16 | 2016-09-27 | Janssen Pharmaceutica Nv | Substituted imidazoles as N-type calcium channel blockers |
| AU2015302633B2 (en) | 2014-08-13 | 2020-01-16 | Meiji Seika Pharma Co., Ltd. | Crystalline anti-trichophyton agents and preparation process thereof |
| CN104313064A (zh) * | 2014-10-01 | 2015-01-28 | 青岛科技大学 | 一种细胞法生产手性溴苯基丙酸甲酯的方法 |
| WO2019220962A1 (ja) | 2018-05-18 | 2019-11-21 | 富士フイルム株式会社 | ３－ジフルオロメチルピラゾール化合物の製造方法及び３－ジフルオロメチルピラゾール－４－カルボン酸化合物の製造方法、並びに、ピラゾリジン化合物 |
| CN110938062B (zh) * | 2019-12-25 | 2021-01-19 | 西华大学 | 3-(4-氯苯基)-4,5-二氢吡唑衍生物及其在农药中的应用 |
| CN111018845B (zh) * | 2019-12-25 | 2020-12-15 | 西华大学 | 3-(4-甲氧苯基)吡唑类化合物及其在农药中的应用 |
| CN111072643B (zh) * | 2019-12-25 | 2021-01-19 | 西华大学 | 4,5-二氢吡唑类化合物及其在农药中的应用 |
| CN111018848B (zh) * | 2019-12-25 | 2020-12-15 | 西华大学 | 1,3,5-三取代-4,5-二氢吡唑衍生物及其在农药中的应用 |
| CN111039933B (zh) * | 2019-12-25 | 2021-03-02 | 西华大学 | 5-杂环取代的吡唑类化合物及其在农药中的应用 |
| CN110981864B (zh) * | 2019-12-25 | 2021-01-29 | 西华大学 | N-(4-氟苯基)-4,5-二氢吡唑类化合物及其在农药中的应用 |
| CN112778208A (zh) * | 2021-01-08 | 2021-05-11 | 中南民族大学 | 一类二氢吡唑类MurA酶抑制剂分子及其制备方法和应用 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2104932A1 (en) * | 1970-09-08 | 1972-04-28 | Ferlux | O-hydroxyphenyl pyrazoles - hypocholesterolemics anti inflammatories analgesics etc |
| US4170464A (en) * | 1974-10-25 | 1979-10-09 | American Cyanamid Company | Herbicidal combinations |
| IL91418A (en) * | 1988-09-01 | 1997-11-20 | Rhone Poulenc Agrochimie | (hetero) cyclic amide derivatives, process for their preparation and fungicidal compositions containing them |
| JP3929700B2 (ja) * | 1998-01-28 | 2007-06-13 | 塩野義製薬株式会社 | 新規三環式化合物 |
-
2003
- 2003-10-08 WO PCT/JP2003/012856 patent/WO2004033432A1/ja active Application Filing
- 2003-10-08 AU AU2003271117A patent/AU2003271117A1/en not_active Abandoned
- 2003-10-08 JP JP2004542837A patent/JP4537855B2/ja not_active Expired - Fee Related
- 2003-10-09 TW TW092128120A patent/TW200418804A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| TW200418804A (en) | 2004-10-01 |
| WO2004033432A1 (ja) | 2004-04-22 |
| JPWO2004033432A1 (ja) | 2006-02-09 |
| JP4537855B2 (ja) | 2010-09-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |