AU2003234637B2 - Methods and compositions for inhibiting HIV replication - Google Patents
Methods and compositions for inhibiting HIV replication Download PDFInfo
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- AU2003234637B2 AU2003234637B2 AU2003234637A AU2003234637A AU2003234637B2 AU 2003234637 B2 AU2003234637 B2 AU 2003234637B2 AU 2003234637 A AU2003234637 A AU 2003234637A AU 2003234637 A AU2003234637 A AU 2003234637A AU 2003234637 B2 AU2003234637 B2 AU 2003234637B2
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
- A61K31/569—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone substituted in position 17 alpha, e.g. ethisterone
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
- A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
- A61K31/704—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin attached to a condensed carbocyclic ring system, e.g. sennosides, thiocolchicosides, escin, daunorubicin
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
- A61K31/7072—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
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- Tropical Medicine & Parasitology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38340902P | 2002-05-24 | 2002-05-24 | |
| US60/383,409 | 2002-05-24 | ||
| PCT/US2003/016524 WO2003099851A2 (en) | 2002-05-24 | 2003-05-23 | Methods and compositions for inhibiting hiv replication |
Publications (2)
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| AU2003234637A1 AU2003234637A1 (en) | 2003-12-12 |
| AU2003234637B2 true AU2003234637B2 (en) | 2009-04-30 |
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| Application Number | Title | Priority Date | Filing Date |
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| AU2003234637A Ceased AU2003234637B2 (en) | 2002-05-24 | 2003-05-23 | Methods and compositions for inhibiting HIV replication |
Country Status (6)
| Country | Link |
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| US (1) | US20060068389A1 (enExample) |
| EP (1) | EP1523328A4 (enExample) |
| JP (1) | JP2005531589A (enExample) |
| AU (1) | AU2003234637B2 (enExample) |
| CA (1) | CA2487655A1 (enExample) |
| WO (1) | WO2003099851A2 (enExample) |
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| US8192709B2 (en) * | 2008-02-21 | 2012-06-05 | Exxonmobil Research And Engineering Company | Separation of methane from higher carbon number hydrocarbons utilizing zeolitic imidazolate framework materials |
Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0474374A1 (en) * | 1990-08-10 | 1992-03-11 | Ortho Pharmaceutical Corporation | Method for treatment of bone wasting diseases using a progestin |
| JPH08239306A (ja) * | 1995-03-03 | 1996-09-17 | Sunstar Inc | 忌避剤 |
| EP0791356A1 (en) * | 1996-02-28 | 1997-08-27 | Pfizer Inc. | Combinations of droloxifene with progestins for the treatment of osteoporosis |
| US5780220A (en) * | 1994-05-19 | 1998-07-14 | Trustees Of The University Of Pennsylvania | Methods and compositions for inhibiting HIV replication |
| US6113920A (en) * | 1996-10-31 | 2000-09-05 | Glaxo Wellcome Inc. | Pharmaceutical compositions |
| WO2001001996A1 (en) * | 1999-06-29 | 2001-01-11 | University Of Western Australia | Compositions and methods for treating or preventing osteoporosis |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS62201819A (ja) * | 1985-11-13 | 1987-09-05 | Res Dev Corp Of Japan | 免疫不全症処置剤 |
| US5874225A (en) * | 1993-02-19 | 1999-02-23 | Trustees Of The University Of Pennsylvania | Identification of compounds that modulate HIV-1 vpr protein activity |
| AU1373395A (en) * | 1993-12-15 | 1995-07-03 | Trustees Of The University Of Pennsylvania, The | Vpr receptor protein |
| US5639598A (en) * | 1994-05-19 | 1997-06-17 | The Trustees Of The University Of Pennsylvania | Method and kit for identification of antiviral agents capable of abrogating HIV Vpr-Rip-1 binding interactions |
| US5763190A (en) * | 1994-09-21 | 1998-06-09 | The Trustees Of The University Of Pennsylvania | Methods for the identification of compounds capable of inducing the nuclear translocation of a receptor complex comprising the glucocoticoid receptor type II and viral protein R interacting protein |
| US6117446A (en) * | 1999-01-26 | 2000-09-12 | Place; Virgil A. | Drug dosage unit for buccal administration of steroidal active agents |
-
2003
- 2003-05-23 CA CA002487655A patent/CA2487655A1/en not_active Abandoned
- 2003-05-23 WO PCT/US2003/016524 patent/WO2003099851A2/en not_active Ceased
- 2003-05-23 EP EP03729137A patent/EP1523328A4/en not_active Withdrawn
- 2003-05-23 AU AU2003234637A patent/AU2003234637B2/en not_active Ceased
- 2003-05-23 JP JP2004508106A patent/JP2005531589A/ja active Pending
- 2003-05-23 US US10/515,327 patent/US20060068389A1/en not_active Abandoned
Patent Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0474374A1 (en) * | 1990-08-10 | 1992-03-11 | Ortho Pharmaceutical Corporation | Method for treatment of bone wasting diseases using a progestin |
| US5780220A (en) * | 1994-05-19 | 1998-07-14 | Trustees Of The University Of Pennsylvania | Methods and compositions for inhibiting HIV replication |
| JPH08239306A (ja) * | 1995-03-03 | 1996-09-17 | Sunstar Inc | 忌避剤 |
| EP0791356A1 (en) * | 1996-02-28 | 1997-08-27 | Pfizer Inc. | Combinations of droloxifene with progestins for the treatment of osteoporosis |
| US6113920A (en) * | 1996-10-31 | 2000-09-05 | Glaxo Wellcome Inc. | Pharmaceutical compositions |
| WO2001001996A1 (en) * | 1999-06-29 | 2001-01-11 | University Of Western Australia | Compositions and methods for treating or preventing osteoporosis |
Non-Patent Citations (2)
| Title |
|---|
| Derwent Abstract Accession No.1996-472220 & JP 08 239306 A (SUNSTAR CHEM IND CO LTD) 17 September 1996. * |
| Hill, R et al. Dictionary of Steroids. CRC Press. 1991 * |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2003234637A1 (en) | 2003-12-12 |
| EP1523328A4 (en) | 2007-10-31 |
| US20060068389A1 (en) | 2006-03-30 |
| JP2005531589A (ja) | 2005-10-20 |
| WO2003099851A3 (en) | 2005-02-24 |
| EP1523328A2 (en) | 2005-04-20 |
| WO2003099851A2 (en) | 2003-12-04 |
| CA2487655A1 (en) | 2003-12-04 |
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| FGA | Letters patent sealed or granted (standard patent) | ||
| MK14 | Patent ceased section 143(a) (annual fees not paid) or expired |