AU2002362443B2 - 2-propynyl adenosine analogs having A2A agonist activity and compositions thereof - Google Patents

2-propynyl adenosine analogs having A2A agonist activity and compositions thereof Download PDF

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Publication number
AU2002362443B2
AU2002362443B2 AU2002362443A AU2002362443A AU2002362443B2 AU 2002362443 B2 AU2002362443 B2 AU 2002362443B2 AU 2002362443 A AU2002362443 A AU 2002362443A AU 2002362443 A AU2002362443 A AU 2002362443A AU 2002362443 B2 AU2002362443 B2 AU 2002362443B2
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compound
carboxylic acid
piperidine
aryl
alkylene
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AU2002362443A1 (en
Inventor
Robert Alan Figler
Joel M. Linden
Timothy L. Macdonald
Lauren Jean Murphree
Jayson M. Rieger
Gail W. Sullivan
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UVA Licensing and Ventures Group
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University of Virginia Patent Foundation
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    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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  • Organic Chemistry (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Biotechnology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biochemistry (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Genetics & Genomics (AREA)
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  • Neurosurgery (AREA)
  • Neurology (AREA)
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AU2002362443A 2001-10-01 2002-10-01 2-propynyl adenosine analogs having A2A agonist activity and compositions thereof Ceased AU2002362443B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US32651701P 2001-10-01 2001-10-01
US60/326,517 2001-10-01
US38320002P 2002-05-24 2002-05-24
US60/383,200 2002-05-24
PCT/US2002/031383 WO2003029264A2 (en) 2001-10-01 2002-10-01 2-propynyl adenosine analogs having a2a agonist activity and compositions thereof

Publications (2)

Publication Number Publication Date
AU2002362443A1 AU2002362443A1 (en) 2003-06-26
AU2002362443B2 true AU2002362443B2 (en) 2008-05-15

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AU2002362443A Ceased AU2002362443B2 (en) 2001-10-01 2002-10-01 2-propynyl adenosine analogs having A2A agonist activity and compositions thereof

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US (3) US7214665B2 (enExample)
EP (1) EP1434782A2 (enExample)
JP (2) JP4514452B2 (enExample)
AU (1) AU2002362443B2 (enExample)
CA (1) CA2460911C (enExample)
NZ (3) NZ556354A (enExample)
SG (1) SG176313A1 (enExample)
WO (1) WO2003029264A2 (enExample)

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