ATE493413T1 - Wasserfreie kristalline formen von n-ä1,2- ethoxyethyl)-5-(n-ethyl-n-methylaminoü-7-(4- methylpyridin-2-yl-aminoü-1h-pyrazoloä4,3- - Google Patents

Wasserfreie kristalline formen von n-ä1,2- ethoxyethyl)-5-(n-ethyl-n-methylaminoü-7-(4- methylpyridin-2-yl-aminoü-1h-pyrazoloä4,3-

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Publication number
ATE493413T1
ATE493413T1 AT06744689T AT06744689T ATE493413T1 AT E493413 T1 ATE493413 T1 AT E493413T1 AT 06744689 T AT06744689 T AT 06744689T AT 06744689 T AT06744689 T AT 06744689T AT E493413 T1 ATE493413 T1 AT E493413T1
Authority
AT
Austria
Prior art keywords
ethoxyethyl
ethyl
crystalline forms
anhydrous crystalline
methylaminoü
Prior art date
Application number
AT06744689T
Other languages
German (de)
English (en)
Inventor
David Andrew Entwistle
Peter Vallance Marshall
Stefan Colin John Taylor
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE493413T1 publication Critical patent/ATE493413T1/de

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A61P3/06—Antihyperlipidemics
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AT06744689T 2005-05-12 2006-05-03 Wasserfreie kristalline formen von n-ä1,2- ethoxyethyl)-5-(n-ethyl-n-methylaminoü-7-(4- methylpyridin-2-yl-aminoü-1h-pyrazoloä4,3- ATE493413T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US68044505P 2005-05-12 2005-05-12
US68171105P 2005-05-17 2005-05-17
PCT/IB2006/001233 WO2006120552A2 (en) 2005-05-12 2006-05-03 ANHYDROUS CRYSTALLINE FORMS OF N-[1-(2-ETHOXYETHYL)-5-(N-ETHYL-N-METHYLAMINO)-7-(4-METHYLPYRIDIN-2-yl-AMINO)-1H-PYRAZOLO[4,3-d]PYRIMIDINE-3-CARBONYL]METHANESULFONAMIDE

Publications (1)

Publication Number Publication Date
ATE493413T1 true ATE493413T1 (de) 2011-01-15

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AT06744689T ATE493413T1 (de) 2005-05-12 2006-05-03 Wasserfreie kristalline formen von n-ä1,2- ethoxyethyl)-5-(n-ethyl-n-methylaminoü-7-(4- methylpyridin-2-yl-aminoü-1h-pyrazoloä4,3-

Country Status (23)

Country Link
US (3) US8227475B2 (pl)
EP (1) EP1881985B1 (pl)
JP (2) JP4271695B2 (pl)
KR (1) KR100939890B1 (pl)
AT (1) ATE493413T1 (pl)
AU (1) AU2006245416B2 (pl)
BR (1) BRPI0609225A2 (pl)
CA (1) CA2608018C (pl)
CR (1) CR9505A (pl)
CY (1) CY1111171T1 (pl)
DE (1) DE602006019231D1 (pl)
DK (1) DK1881985T3 (pl)
EA (1) EA012577B1 (pl)
IL (1) IL186693A (pl)
MA (1) MA29447B1 (pl)
MX (1) MX2007013215A (pl)
NO (1) NO20075258L (pl)
NZ (1) NZ564187A (pl)
PL (1) PL1881985T3 (pl)
PT (1) PT1881985E (pl)
TN (1) TNSN07414A1 (pl)
TW (1) TWI380986B (pl)
WO (1) WO2006120552A2 (pl)

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MX2007013215A (es) 2007-12-12
AU2006245416A1 (en) 2006-11-16
PT1881985E (pt) 2011-02-01
US8796287B2 (en) 2014-08-05
PL1881985T3 (pl) 2011-05-31
IL186693A (en) 2012-07-31
TWI380986B (zh) 2013-01-01
US8796288B2 (en) 2014-08-05
AU2006245416B2 (en) 2012-02-23
CA2608018A1 (en) 2006-11-16
NO20075258L (no) 2007-11-15
US20120208830A1 (en) 2012-08-16
TNSN07414A1 (fr) 2009-03-17
JP2006316058A (ja) 2006-11-24
US8227475B2 (en) 2012-07-24
JP4996631B2 (ja) 2012-08-08
EA200702217A1 (ru) 2008-04-28
MA29447B1 (fr) 2008-05-02
EA012577B1 (ru) 2009-10-30
IL186693A0 (en) 2008-02-09
EP1881985A2 (en) 2008-01-30
WO2006120552A3 (en) 2007-01-18
KR20080004593A (ko) 2008-01-09
CR9505A (es) 2008-01-02
NZ564187A (en) 2010-03-26
BRPI0609225A2 (pt) 2010-03-09
US20120214827A1 (en) 2012-08-23
KR100939890B1 (ko) 2010-01-29
US20080194591A1 (en) 2008-08-14
CA2608018C (en) 2010-07-13
CY1111171T1 (el) 2015-06-11
DK1881985T3 (da) 2011-02-14
EP1881985B1 (en) 2010-12-29
TW200716641A (en) 2007-05-01
WO2006120552A2 (en) 2006-11-16
JP2009137987A (ja) 2009-06-25
HK1116485A1 (en) 2008-12-24
JP4271695B2 (ja) 2009-06-03
DE602006019231D1 (en) 2011-02-10

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