ATE482954T1 - Thiazolidinderivate und ihre verwendung als fungizide - Google Patents
Thiazolidinderivate und ihre verwendung als fungizideInfo
- Publication number
- ATE482954T1 ATE482954T1 AT01963155T AT01963155T ATE482954T1 AT E482954 T1 ATE482954 T1 AT E482954T1 AT 01963155 T AT01963155 T AT 01963155T AT 01963155 T AT01963155 T AT 01963155T AT E482954 T1 ATE482954 T1 AT E482954T1
- Authority
- AT
- Austria
- Prior art keywords
- fungicides
- thiazolidine derivatives
- nr3r4
- thiazolidine
- derivatives
- Prior art date
Links
- OGYGFUAIIOPWQD-UHFFFAOYSA-N 1,3-thiazolidine Chemical class C1CSCN1 OGYGFUAIIOPWQD-UHFFFAOYSA-N 0.000 title 1
- 239000000417 fungicide Substances 0.000 title 1
- 101100516568 Caenorhabditis elegans nhr-7 gene Proteins 0.000 abstract 1
- 206010017533 Fungal infection Diseases 0.000 abstract 1
- 208000031888 Mycoses Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 238000011321 prophylaxis Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0021419.7A GB0021419D0 (en) | 2000-08-31 | 2000-08-31 | Compounds |
| PCT/GB2001/003860 WO2002022612A1 (en) | 2000-08-31 | 2001-08-30 | Thiazolidine derivatives and its use as antifungal agent |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE482954T1 true ATE482954T1 (de) | 2010-10-15 |
Family
ID=9898614
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT01963155T ATE482954T1 (de) | 2000-08-31 | 2001-08-30 | Thiazolidinderivate und ihre verwendung als fungizide |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US6740670B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP1313731B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP2004509121A (cg-RX-API-DMAC7.html) |
| AT (1) | ATE482954T1 (cg-RX-API-DMAC7.html) |
| AU (1) | AU2001284188A1 (cg-RX-API-DMAC7.html) |
| DE (1) | DE60143165D1 (cg-RX-API-DMAC7.html) |
| ES (1) | ES2353685T3 (cg-RX-API-DMAC7.html) |
| GB (1) | GB0021419D0 (cg-RX-API-DMAC7.html) |
| WO (1) | WO2002022612A1 (cg-RX-API-DMAC7.html) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005014563A1 (en) | 2003-08-11 | 2005-02-17 | F. Hoffmann-La Roche Ag | Piperazine with or-substituted phenyl group and their use as glyt1 inhibitors |
| LT2653465T (lt) | 2004-03-15 | 2016-09-12 | Janssen Pharmaceutica Nv | Opioidinio receptoriaus moduliatoriai |
| CN101072762B (zh) | 2004-12-09 | 2010-06-23 | 弗·哈夫曼-拉罗切有限公司 | 苯基-哌嗪甲酮衍生物 |
| WO2006063709A1 (en) | 2004-12-15 | 2006-06-22 | F.Hoffmann-La Roche Ag | Bi- and tricyclic substituted phenyl methanones as glycine transporter i (glyt-1) inhibitors for the treatment of alzheimer’s disease |
| US7485637B2 (en) | 2005-01-04 | 2009-02-03 | Hoffmann-La Roche Inc. | Benzoyl-tetrahydropiperidine derivatives |
| JP5006799B2 (ja) | 2005-01-07 | 2012-08-22 | エフ．ホフマン−ラ ロシュ アーゲー | 神経疾患及び精神神経疾患の処置用のグリシントランスポーター１（ｇｌｙｔ−１）阻害剤としての［４−（ヘテロアリール）ピペラジン−１−イル］−（２，５−置換フェニル）−メタノン誘導体 |
| KR100935256B1 (ko) | 2005-01-18 | 2010-01-06 | 에프. 호프만-라 로슈 아게 | 신경 질환 및 신경정신 질환의 치료를 위한 글라이신트랜스포터 1(ｇｌｙｔ-1) 억제제로서의 2,5-이치환된 페닐메탄온 유도체 |
| ES2332529T3 (es) | 2005-01-26 | 2010-02-08 | F. Hoffmann-La Roche Ag | Derivados de fenil-metanona y su empleo como inhibidores del transportador 1 de glicina. |
| NZ556434A (en) | 2005-02-07 | 2010-05-28 | Hoffmann La Roche | Heterocyclic substituted phenyl methanones as inhibitors of the glycine transporter 1 |
| MX2010012626A (es) | 2008-05-20 | 2011-02-22 | Merck Sharp & Dohme | Produccion eficiente de proteinas heterologas utilizando inhibidores de manosil transferasa. |
| US8957066B2 (en) | 2011-02-28 | 2015-02-17 | Biomarin Pharmaceutical Inc. | Histone deacetylase inhibitors |
| US10059723B2 (en) | 2011-02-28 | 2018-08-28 | Biomarin Pharmaceutical Inc. | Histone deacetylase inhibitors |
| RU2662153C1 (ru) * | 2017-04-20 | 2018-07-24 | Общество С Ограниченной Ответственностью "Дермавитал Групп" | Гибридные эфиры на основе производных тиазолидин-2,4-диона и азолов (1н-1,3-имидазола и 1н-1,3,4-триазола) и их применение |
| RU2690161C1 (ru) * | 2018-06-28 | 2019-05-31 | Общество С Ограниченной Ответственностью "Дермавитал Групп" | 3,5-Замещенные производные тиазолидин-2,4-диона, обладающие противомикробной активностью |
| RU2703997C1 (ru) * | 2018-12-13 | 2019-10-23 | Общество с ограниченной ответственностью "Л-Био" | Гибридные амиды на основе триазола и тиазолидина, обладающие антимикробной активностью |
| US11292776B2 (en) | 2019-12-12 | 2022-04-05 | University Of Sharjah | Small molecule inhibitors of fungal hyphae and biofilm formation |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US47109A (en) * | 1865-04-04 | Improvement in governors | ||
| FR1604530A (cg-RX-API-DMAC7.html) * | 1967-06-06 | 1971-11-29 | ||
| JPS5740478A (en) * | 1980-08-22 | 1982-03-06 | Ono Pharmaceut Co Ltd | Rhodanine derivative, its preparation and aldose reductase inhibitor containing rhodanine derivative |
| DE4318550A1 (de) * | 1993-06-04 | 1994-12-08 | Boehringer Mannheim Gmbh | Aryliden-4-oxo-2-thioxo-3- thiazolidincarbonsäuren, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
| DE19835316A1 (de) * | 1998-08-05 | 2000-02-10 | Bosch Gmbh Robert | Gesteuerte Gleichrichterbrücke mit Überspannungsschutz |
| WO2000018747A1 (en) * | 1998-09-30 | 2000-04-06 | Roche Diagnostics Gmbh | Rhodanine carboxylic acid derivatives for the treatment and prevention of metabolic bone disorders |
-
2000
- 2000-08-31 GB GBGB0021419.7A patent/GB0021419D0/en not_active Ceased
-
2001
- 2001-08-30 ES ES01963155T patent/ES2353685T3/es not_active Expired - Lifetime
- 2001-08-30 DE DE60143165T patent/DE60143165D1/de not_active Expired - Lifetime
- 2001-08-30 AU AU2001284188A patent/AU2001284188A1/en not_active Abandoned
- 2001-08-30 WO PCT/GB2001/003860 patent/WO2002022612A1/en not_active Ceased
- 2001-08-30 EP EP01963155A patent/EP1313731B1/en not_active Expired - Lifetime
- 2001-08-30 AT AT01963155T patent/ATE482954T1/de active
- 2001-08-30 JP JP2002526865A patent/JP2004509121A/ja active Pending
-
2003
- 2003-02-21 US US10/371,979 patent/US6740670B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| ES2353685T3 (es) | 2011-03-04 |
| GB0021419D0 (en) | 2000-10-18 |
| US6740670B2 (en) | 2004-05-25 |
| US20030216453A1 (en) | 2003-11-20 |
| DE60143165D1 (de) | 2010-11-11 |
| WO2002022612A1 (en) | 2002-03-21 |
| WO2002022612A8 (en) | 2002-05-23 |
| EP1313731B1 (en) | 2010-09-29 |
| JP2004509121A (ja) | 2004-03-25 |
| AU2001284188A1 (en) | 2002-03-26 |
| EP1313731A1 (en) | 2003-05-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
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