ATE466579T1 - Verfahren zur herstellung von benzimidazolen - Google Patents
Verfahren zur herstellung von benzimidazolenInfo
- Publication number
- ATE466579T1 ATE466579T1 AT04820975T AT04820975T ATE466579T1 AT E466579 T1 ATE466579 T1 AT E466579T1 AT 04820975 T AT04820975 T AT 04820975T AT 04820975 T AT04820975 T AT 04820975T AT E466579 T1 ATE466579 T1 AT E466579T1
- Authority
- AT
- Austria
- Prior art keywords
- benzimidazoles
- producing
- salts
- reconstitutable
- discloses
- Prior art date
Links
- 150000001556 benzimidazoles Chemical class 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title 1
- 150000003839 salts Chemical class 0.000 abstract 2
- 238000012377 drug delivery Methods 0.000 abstract 1
- 229940102223 injectable solution Drugs 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
- 239000000843 powder Substances 0.000 abstract 1
- 229940126409 proton pump inhibitor Drugs 0.000 abstract 1
- 239000000612 proton pump inhibitor Substances 0.000 abstract 1
- YREYEVIYCVEVJK-UHFFFAOYSA-N rabeprazole Chemical compound COCCCOC1=CC=NC(CS(=O)C=2NC3=CC=CC=C3N=2)=C1C YREYEVIYCVEVJK-UHFFFAOYSA-N 0.000 abstract 1
- 229960004157 rabeprazole Drugs 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Dermatology (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Steroid Compounds (AREA)
- Preventing Corrosion Or Incrustation Of Metals (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN1164MU2003 | 2003-11-05 | ||
| PCT/IN2004/000342 WO2005065682A2 (en) | 2003-11-05 | 2004-11-03 | Rabeprazole containing formulation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE466579T1 true ATE466579T1 (de) | 2010-05-15 |
Family
ID=34746668
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT04820975T ATE466579T1 (de) | 2003-11-05 | 2004-11-03 | Verfahren zur herstellung von benzimidazolen |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20070014875A1 (de) |
| EP (1) | EP1713476B1 (de) |
| AT (1) | ATE466579T1 (de) |
| BR (1) | BRPI0416027A (de) |
| CY (1) | CY1110717T1 (de) |
| DE (1) | DE602004027088D1 (de) |
| DK (1) | DK1713476T3 (de) |
| ES (1) | ES2344905T3 (de) |
| PL (1) | PL1713476T3 (de) |
| PT (1) | PT1713476E (de) |
| WO (1) | WO2005065682A2 (de) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2649946A1 (en) * | 2006-05-09 | 2007-11-15 | Astrazeneca Ab | New sterilized parenteral formulation |
| CN102138907A (zh) * | 2010-02-02 | 2011-08-03 | 南京长澳医药科技有限公司 | 一种稳定的雷贝拉唑钠冻干制剂及其制备方法 |
| CN103463636B (zh) * | 2013-09-17 | 2015-05-27 | 天津市嵩锐医药科技有限公司 | 一种供注射用的泮托拉唑钠药物组合物 |
| MA41623A (fr) * | 2015-11-26 | 2018-01-09 | Verano Ilac Sanayi Ve Ticaret A S | Composition lyophilisée de composé de benzimidazole |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH07509214A (ja) * | 1992-07-20 | 1995-10-12 | ユニリーバー・ナームローゼ・ベンノートシャープ | 気体水化物の製造 |
| RU2126252C1 (ru) * | 1992-07-28 | 1999-02-20 | Астра Актиеболаг | Препарат для инъекций и набор для инъекций, содержащие омепразол и его аналоги |
| TW280770B (de) * | 1993-10-15 | 1996-07-11 | Takeda Pharm Industry Co Ltd | |
| AU2001278755A1 (en) | 2000-08-18 | 2002-03-04 | Takeda Chemical Industries Ltd. | Injections |
-
2004
- 2004-11-03 EP EP04820975A patent/EP1713476B1/de not_active Revoked
- 2004-11-03 AT AT04820975T patent/ATE466579T1/de active
- 2004-11-03 BR BRPI0416027-4A patent/BRPI0416027A/pt not_active IP Right Cessation
- 2004-11-03 DE DE602004027088T patent/DE602004027088D1/de not_active Expired - Lifetime
- 2004-11-03 DK DK04820975.3T patent/DK1713476T3/da active
- 2004-11-03 PT PT04820975T patent/PT1713476E/pt unknown
- 2004-11-03 ES ES04820975T patent/ES2344905T3/es not_active Expired - Lifetime
- 2004-11-03 PL PL04820975T patent/PL1713476T3/pl unknown
- 2004-11-03 WO PCT/IN2004/000342 patent/WO2005065682A2/en not_active Ceased
- 2004-11-03 US US10/574,666 patent/US20070014875A1/en not_active Abandoned
-
2010
- 2010-07-27 CY CY20101100704T patent/CY1110717T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BRPI0416027A (pt) | 2007-01-02 |
| CY1110717T1 (el) | 2015-06-10 |
| WO2005065682A2 (en) | 2005-07-21 |
| DK1713476T3 (da) | 2010-08-09 |
| EP1713476A2 (de) | 2006-10-25 |
| DE602004027088D1 (de) | 2010-06-17 |
| PT1713476E (pt) | 2010-08-04 |
| EP1713476B1 (de) | 2010-05-05 |
| ES2344905T3 (es) | 2010-09-09 |
| US20070014875A1 (en) | 2007-01-18 |
| WO2005065682A3 (en) | 2005-09-01 |
| PL1713476T3 (pl) | 2010-10-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
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