ATE443061T1 - Benzoxazinon- und benzoxazepinonoxazolidinone als antibakterielle mittel - Google Patents

Benzoxazinon- und benzoxazepinonoxazolidinone als antibakterielle mittel

Info

Publication number
ATE443061T1
ATE443061T1 AT07705605T AT07705605T ATE443061T1 AT E443061 T1 ATE443061 T1 AT E443061T1 AT 07705605 T AT07705605 T AT 07705605T AT 07705605 T AT07705605 T AT 07705605T AT E443061 T1 ATE443061 T1 AT E443061T1
Authority
AT
Austria
Prior art keywords
antibacterial agents
benzoxazepinonoxazolidinone
benzoxazinone
het
present
Prior art date
Application number
AT07705605T
Other languages
German (de)
English (en)
Inventor
Hongwu Gao
Mikhail Gordeev
Gary Luehr
Nagendra Josyula Vara Venkata
Adam Renslo
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of ATE443061T1 publication Critical patent/ATE443061T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Oncology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
AT07705605T 2006-02-14 2007-02-05 Benzoxazinon- und benzoxazepinonoxazolidinone als antibakterielle mittel ATE443061T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US77307106P 2006-02-14 2006-02-14
PCT/IB2007/000377 WO2007093904A1 (en) 2006-02-14 2007-02-05 Benzoxazinone and benzoxazepinone oxazolidinones as antibacterial agents

Publications (1)

Publication Number Publication Date
ATE443061T1 true ATE443061T1 (de) 2009-10-15

Family

ID=38068038

Family Applications (1)

Application Number Title Priority Date Filing Date
AT07705605T ATE443061T1 (de) 2006-02-14 2007-02-05 Benzoxazinon- und benzoxazepinonoxazolidinone als antibakterielle mittel

Country Status (9)

Country Link
US (1) US20090318431A1 (enExample)
EP (1) EP1987025B1 (enExample)
JP (1) JP2009526832A (enExample)
AT (1) ATE443061T1 (enExample)
CA (1) CA2642406A1 (enExample)
DE (1) DE602007002476D1 (enExample)
DK (1) DK1987025T3 (enExample)
ES (1) ES2331930T3 (enExample)
WO (1) WO2007093904A1 (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2010008922A (es) * 2008-02-20 2010-09-07 Actelion Pharmaceuticals Ltd Compuestos antibioticos azatriciclicos.
ES2398939T3 (es) * 2008-02-22 2013-03-22 Actelion Pharmaceuticals Ltd. Derivados de oxazolidinona
KR100980681B1 (ko) 2008-09-16 2010-09-07 한국과학기술연구원 디플루오로페닐 유도체를 갖는 신규한 옥사졸리디논 유도체또는 이의 약학적으로 허용가능한 염, 이의 제조방법 및 이를 유효성분으로 하는 항생제 조성물
US8722686B2 (en) 2008-09-19 2014-05-13 Pfizer Inc. Hydroxamic acid derivatives useful as antibacterial agents
MY158520A (en) 2008-10-07 2016-10-14 Actelion Pharmaceuticals Ltd Tricyclic oxazolidinone antibiotic compounds
CN102224151A (zh) 2008-11-20 2011-10-19 万能药生物有限公司 新的抗微生物剂
JP5696142B2 (ja) 2009-06-26 2015-04-08 パナセア バイオテック リミテッド 新規アザビシクロヘキサン類
CA2899583A1 (en) 2009-12-16 2011-06-23 Pfizer Inc. N-linked hydroxamic acid derivatives useful as antibacterial agents
AU2012238374B2 (en) * 2011-04-08 2015-04-02 Pfizer Inc. Isoxazole derivatives useful as antibacterial agents
UA112897C2 (uk) 2012-05-09 2016-11-10 Байєр Фарма Акцієнгезелльшафт Біциклічно заміщені урацили та їх застосування для лікування і/або профілактики захворювань
GB2550437B (en) * 2016-05-20 2021-06-23 Bugworks Res Inc Heterocyclic compounds useful as anti-bacterial agents and method for production
CN113264949B (zh) * 2021-05-31 2022-04-05 西南大学 一类螺苯并噁嗪哌啶α,β-不饱和酮类衍生物的设计合成与应用
CN114133360A (zh) * 2021-11-30 2022-03-04 南京工业大学 一种含氟苯并[d]-1,3-氧氮杂卓化合物及其合成方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19802239A1 (de) * 1998-01-22 1999-07-29 Bayer Ag Neue mit Bicyclen substituierte Oxazolidinone
WO2000029409A1 (de) * 1998-11-17 2000-05-25 Bayer Aktiengesellschaft Neue heterocyclyl-substituierte oxazolidon-derivate
WO2005082897A1 (en) * 2004-01-28 2005-09-09 Pharmacia & Upjohn Company Llc Oxazolidinone antibacterial agents

Also Published As

Publication number Publication date
CA2642406A1 (en) 2007-08-23
EP1987025A1 (en) 2008-11-05
WO2007093904A1 (en) 2007-08-23
JP2009526832A (ja) 2009-07-23
DE602007002476D1 (de) 2009-10-29
ES2331930T3 (es) 2010-01-20
EP1987025B1 (en) 2009-09-16
US20090318431A1 (en) 2009-12-24
DK1987025T3 (da) 2009-12-07

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