ATE433971T1 - Neue azolderivate - Google Patents

Neue azolderivate

Info

Publication number
ATE433971T1
ATE433971T1 AT03812297T AT03812297T ATE433971T1 AT E433971 T1 ATE433971 T1 AT E433971T1 AT 03812297 T AT03812297 T AT 03812297T AT 03812297 T AT03812297 T AT 03812297T AT E433971 T1 ATE433971 T1 AT E433971T1
Authority
AT
Austria
Prior art keywords
disorders
methine
diseases
nitrogen
present
Prior art date
Application number
AT03812297T
Other languages
English (en)
Inventor
Norikazu Otake
Yuji Haga
Makoto Jitsuoka
Akio Kanatani
Original Assignee
Banyu Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Banyu Pharma Co Ltd filed Critical Banyu Pharma Co Ltd
Application granted granted Critical
Publication of ATE433971T1 publication Critical patent/ATE433971T1/de

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Obesity (AREA)
  • Addiction (AREA)
  • Urology & Nephrology (AREA)
  • Reproductive Health (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pregnancy & Childbirth (AREA)
  • Gynecology & Obstetrics (AREA)
  • Emergency Medicine (AREA)
  • Nutrition Science (AREA)
  • Child & Adolescent Psychology (AREA)
AT03812297T 2002-11-29 2003-11-25 Neue azolderivate ATE433971T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002346997 2002-11-29
PCT/JP2003/015018 WO2004050652A1 (ja) 2002-11-29 2003-11-25 新規アゾール誘導体

Publications (1)

Publication Number Publication Date
ATE433971T1 true ATE433971T1 (de) 2009-07-15

Family

ID=32462868

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03812297T ATE433971T1 (de) 2002-11-29 2003-11-25 Neue azolderivate

Country Status (8)

Country Link
US (2) US7365079B2 (de)
EP (1) EP1566384B1 (de)
JP (2) JPWO2004050652A1 (de)
AT (1) ATE433971T1 (de)
AU (1) AU2003302640B2 (de)
CA (1) CA2507742A1 (de)
DE (1) DE60328035D1 (de)
WO (1) WO2004050652A1 (de)

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JP2006528617A (ja) * 2003-07-24 2006-12-21 ファーマジーン ラボラトリーズ リミテッド ５−ｈｔ２ｂ受容体アンタゴニスト
BRPI0414804A (pt) * 2003-09-26 2006-11-14 Pfizer Prod Inc tratamento de perturbações neurológicas relacionadas com perturbações de sono para movimentos oculares rápidos (rem) com antagonistas dos receptores npy y5
US7803838B2 (en) * 2004-06-04 2010-09-28 Forest Laboratories Holdings Limited Compositions comprising nebivolol
US7838552B2 (en) 2004-06-04 2010-11-23 Forest Laboratories Holdings Limited Compositions comprising nebivolol
RU2007109794A (ru) * 2004-08-19 2008-09-27 Вертекс Фармасьютикалз, Инкорпорейтед (Us) Модуляторы мускариновых рецепторов
US7786141B2 (en) * 2004-08-19 2010-08-31 Vertex Pharmaceuticals Incorporated Dihydrospiroindene modulators of muscarinic receptors
EP1795527B1 (de) * 2004-09-07 2009-04-22 Banyu Pharmaceutical Co., Ltd. Carbamoylsubstituiertes spiro-derivat
AU2005309365B2 (en) * 2004-11-29 2011-10-06 Vertex Pharmaceuticals Incorporated Modulators of muscarinic receptors
US20070035750A1 (en) * 2005-08-10 2007-02-15 Canon Kabushiki Kaisha Configurable device model for n-channel device
US8026260B2 (en) * 2005-11-03 2011-09-27 Merck Sharp & Dohme Corp. Histone deacetylase inhibitors with aryl-pyrazolyl-motifs
JP4371164B2 (ja) 2005-11-10 2009-11-25 萬有製薬株式会社 アザ置換スピロ誘導体
AU2006330866A1 (en) * 2005-12-22 2007-07-05 Vertex Pharmaceuticals Incorporated Modulators of muscarinic receptors
ATE517106T1 (de) * 2006-02-22 2011-08-15 Vertex Pharma Kondensierte spiropiperidine als modulatoren muskarinartiger rezeptoren
EP1988892A2 (de) 2006-02-22 2008-11-12 Vertex Pharmaceuticals Incorporated Modulatoren muskarinischer rezeptoren
CN101500565A (zh) * 2006-06-29 2009-08-05 弗特克斯药品有限公司 毒蕈碱性受体的调节剂
CN101553231A (zh) * 2006-08-15 2009-10-07 弗特克斯药品有限公司 毒蕈碱受体调节剂
JP2010501561A (ja) 2006-08-18 2010-01-21 バーテックス ファーマシューティカルズ インコーポレイテッド ムスカリン受容体の調節剤
WO2008056687A1 (fr) * 2006-11-09 2008-05-15 Daiichi Sankyo Company, Limited Nouveau dérivé de spiropipéridine
CA2700724A1 (en) * 2007-10-03 2009-04-09 Vertex Pharmaceuticals Incorporated Modulators of muscarinic receptors
WO2010094120A1 (en) * 2009-02-17 2010-08-26 Merck Frosst Canada Ltd. Novel spiro compounds useful as inhibitors of stearoyl-coenzyme a delta-9 desaturase
JP5739674B2 (ja) 2010-09-27 2015-06-24 任天堂株式会社 情報処理プログラム、情報処理装置、情報処理システム、および、情報処理方法
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TW201600522A (zh) * 2014-02-20 2016-01-01 赫孚孟拉羅股份公司 螺－唑酮

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EP1566384A4 (de) 2007-11-21
US20060111380A1 (en) 2006-05-25
CA2507742A1 (en) 2004-06-17
US7589096B2 (en) 2009-09-15
JPWO2004050652A1 (ja) 2006-03-30
AU2003302640B2 (en) 2009-09-24
JP2010215654A (ja) 2010-09-30
EP1566384B1 (de) 2009-06-17
US7365079B2 (en) 2008-04-29
DE60328035D1 (de) 2009-07-30
EP1566384A1 (de) 2005-08-24
US20080188507A1 (en) 2008-08-07
WO2004050652A1 (ja) 2004-06-17
AU2003302640A1 (en) 2004-06-23

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