ATE433971T1 - Neue azolderivate - Google Patents

Neue azolderivate

Info

Publication number
ATE433971T1
ATE433971T1 AT03812297T AT03812297T ATE433971T1 AT E433971 T1 ATE433971 T1 AT E433971T1 AT 03812297 T AT03812297 T AT 03812297T AT 03812297 T AT03812297 T AT 03812297T AT E433971 T1 ATE433971 T1 AT E433971T1
Authority
AT
Austria
Prior art keywords
disorders
methine
diseases
nitrogen
present
Prior art date
Application number
AT03812297T
Other languages
English (en)
Inventor
Norikazu Otake
Yuji Haga
Makoto Jitsuoka
Akio Kanatani
Original Assignee
Banyu Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Banyu Pharma Co Ltd filed Critical Banyu Pharma Co Ltd
Application granted granted Critical
Publication of ATE433971T1 publication Critical patent/ATE433971T1/de

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Obesity (AREA)
  • Addiction (AREA)
  • Urology & Nephrology (AREA)
  • Reproductive Health (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pregnancy & Childbirth (AREA)
  • Gynecology & Obstetrics (AREA)
  • Emergency Medicine (AREA)
  • Nutrition Science (AREA)
  • Child & Adolescent Psychology (AREA)
AT03812297T 2002-11-29 2003-11-25 Neue azolderivate ATE433971T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002346997 2002-11-29
PCT/JP2003/015018 WO2004050652A1 (ja) 2002-11-29 2003-11-25 新規アゾール誘導体

Publications (1)

Publication Number Publication Date
ATE433971T1 true ATE433971T1 (de) 2009-07-15

Family

ID=32462868

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03812297T ATE433971T1 (de) 2002-11-29 2003-11-25 Neue azolderivate

Country Status (8)

Country Link
US (2) US7365079B2 (de)
EP (1) EP1566384B1 (de)
JP (2) JPWO2004050652A1 (de)
AT (1) ATE433971T1 (de)
AU (1) AU2003302640B2 (de)
CA (1) CA2507742A1 (de)
DE (1) DE60328035D1 (de)
WO (1) WO2004050652A1 (de)

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US20090018150A1 (en) * 2003-07-24 2009-01-15 Asterand Uk Limited 5-Ht2b Receptor Antagonists
JP2007506731A (ja) * 2003-09-26 2007-03-22 ファイザー・プロダクツ・インク Ｎｐｙｙ５受容体アンタゴニストによる急速眼球運動（ｒｅｍ）睡眠妨害に関連する神経障害の治療
US7838552B2 (en) 2004-06-04 2010-11-23 Forest Laboratories Holdings Limited Compositions comprising nebivolol
US7803838B2 (en) * 2004-06-04 2010-09-28 Forest Laboratories Holdings Limited Compositions comprising nebivolol
RU2007109794A (ru) 2004-08-19 2008-09-27 Вертекс Фармасьютикалз, Инкорпорейтед (Us) Модуляторы мускариновых рецепторов
US7786141B2 (en) 2004-08-19 2010-08-31 Vertex Pharmaceuticals Incorporated Dihydrospiroindene modulators of muscarinic receptors
ATE429426T1 (de) * 2004-09-07 2009-05-15 Banyu Pharma Co Ltd Carbamoylsubstituiertes spiro-derivat
WO2006058303A2 (en) 2004-11-29 2006-06-01 Vertex Pharmaceuticals Incorporated Modulators of muscarinic receptors
US20070035750A1 (en) * 2005-08-10 2007-02-15 Canon Kabushiki Kaisha Configurable device model for n-channel device
WO2007055941A2 (en) * 2005-11-03 2007-05-18 Merck & Co., Inc. Histone deacetylase inhibitors with aryl-pyrazolyl motifs
CA2629018C (en) * 2005-11-10 2013-12-31 Banyu Pharmaceutical Co., Ltd. Aza-substituted spiro derivative
AU2006330866A1 (en) * 2005-12-22 2007-07-05 Vertex Pharmaceuticals Incorporated Modulators of muscarinic receptors
RU2008137583A (ru) * 2006-02-22 2010-03-27 Вертекс Фармасьютикалз Инкорпорейшн (Us) Спиропиперидины в качестве модуляторов мускариновых рецепторов
RU2008137593A (ru) * 2006-02-22 2010-03-27 Вертекс Фармасьютикалз Инкорпорейтед (Us) Модуляторы мускариновых рецепторов
US7858790B2 (en) * 2006-06-29 2010-12-28 Vertex Pharmaceuticals Incorporated Modulators of muscarinic receptors
EP2051712A2 (de) * 2006-08-15 2009-04-29 Vertex Pharmceuticals Incorporated Modulatoren muskarinischer rezeptoren
AU2007284350A1 (en) 2006-08-18 2008-02-21 Vertex Pharmaceuticals Incorporated Modulators of muscarinic receptors
WO2008056687A1 (en) * 2006-11-09 2008-05-15 Daiichi Sankyo Company, Limited Novel spiropiperidine derivative
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JP5597210B2 (ja) * 2009-02-17 2014-10-01 メルク カナダ インコーポレイテッド ステアロイル−補酵素ａデルタ−９デサチュラーゼの阻害剤として有用な新規スピロ化合物
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US20060111380A1 (en) 2006-05-25
CA2507742A1 (en) 2004-06-17
WO2004050652A1 (ja) 2004-06-17
US7589096B2 (en) 2009-09-15
EP1566384A1 (de) 2005-08-24
US7365079B2 (en) 2008-04-29
EP1566384A4 (de) 2007-11-21
JPWO2004050652A1 (ja) 2006-03-30
US20080188507A1 (en) 2008-08-07
JP2010215654A (ja) 2010-09-30
DE60328035D1 (de) 2009-07-30
EP1566384B1 (de) 2009-06-17

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