ATE425984T1 - Trizyklische antibakterielle makrolidderivate - Google Patents
Trizyklische antibakterielle makrolidderivateInfo
- Publication number
- ATE425984T1 ATE425984T1 AT03731049T AT03731049T ATE425984T1 AT E425984 T1 ATE425984 T1 AT E425984T1 AT 03731049 T AT03731049 T AT 03731049T AT 03731049 T AT03731049 T AT 03731049T AT E425984 T1 ATE425984 T1 AT E425984T1
- Authority
- AT
- Austria
- Prior art keywords
- macrolide derivatives
- antibacterial
- compounds
- tricyclic
- tricyclic antibacterial
- Prior art date
Links
- 230000000844 anti-bacterial effect Effects 0.000 title abstract 2
- 239000003120 macrolide antibiotic agent Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 4
- 238000000034 method Methods 0.000 abstract 3
- 229940002612 prodrug Drugs 0.000 abstract 2
- 239000000651 prodrug Substances 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 208000035143 Bacterial infection Diseases 0.000 abstract 1
- 208000022362 bacterial infectious disease Diseases 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 238000011321 prophylaxis Methods 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13679602A | 2002-04-30 | 2002-04-30 | |
| US20570802A | 2002-07-26 | 2002-07-26 | |
| US42230903A | 2003-04-24 | 2003-04-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE425984T1 true ATE425984T1 (de) | 2009-04-15 |
Family
ID=29407678
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT03731049T ATE425984T1 (de) | 2002-04-30 | 2003-04-25 | Trizyklische antibakterielle makrolidderivate |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP1501846B1 (de) |
| JP (1) | JP2005530758A (de) |
| AT (1) | ATE425984T1 (de) |
| CA (1) | CA2484095A1 (de) |
| DE (1) | DE60326710D1 (de) |
| MX (1) | MXPA04010818A (de) |
| WO (1) | WO2003093289A1 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2469304A1 (en) | 2001-12-05 | 2003-06-19 | Ortho-Mcneil Pharmaceutical, Inc. | 6-o acyl ketolide antibacterials |
| DK200201957A (da) | 2002-12-20 | 2003-01-20 | Alpharma Aps | 10-substituted erythromycin ketolides and methods of making |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA51730C2 (uk) * | 1996-09-04 | 2002-12-16 | Ебботт Лабораторіз | 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців |
-
2003
- 2003-04-25 WO PCT/US2003/012971 patent/WO2003093289A1/en not_active Ceased
- 2003-04-25 CA CA002484095A patent/CA2484095A1/en not_active Abandoned
- 2003-04-25 MX MXPA04010818A patent/MXPA04010818A/es unknown
- 2003-04-25 JP JP2004501428A patent/JP2005530758A/ja active Pending
- 2003-04-25 DE DE60326710T patent/DE60326710D1/de not_active Expired - Fee Related
- 2003-04-25 EP EP03731049A patent/EP1501846B1/de not_active Expired - Lifetime
- 2003-04-25 AT AT03731049T patent/ATE425984T1/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| JP2005530758A (ja) | 2005-10-13 |
| EP1501846B1 (de) | 2009-03-18 |
| WO2003093289A1 (en) | 2003-11-13 |
| EP1501846A1 (de) | 2005-02-02 |
| DE60326710D1 (de) | 2009-04-30 |
| CA2484095A1 (en) | 2003-11-13 |
| MXPA04010818A (es) | 2005-03-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |