ATE404551T1 - 3-hydroxymethylbenzo b thiophen-derivate und verfahren zu deren herstellung - Google Patents

3-hydroxymethylbenzo b thiophen-derivate und verfahren zu deren herstellung

Info

Publication number
ATE404551T1
ATE404551T1 AT02724673T AT02724673T ATE404551T1 AT E404551 T1 ATE404551 T1 AT E404551T1 AT 02724673 T AT02724673 T AT 02724673T AT 02724673 T AT02724673 T AT 02724673T AT E404551 T1 ATE404551 T1 AT E404551T1
Authority
AT
Austria
Prior art keywords
group
carbons
hydroxymethylbenzo
production
trihalomethoxy
Prior art date
Application number
AT02724673T
Other languages
English (en)
Inventor
Hirosi Saitou
Tsuyoshi Mizuno
Naoki Tsuchiya
Original Assignee
Teijin Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teijin Pharma Ltd filed Critical Teijin Pharma Ltd
Application granted granted Critical
Publication of ATE404551T1 publication Critical patent/ATE404551T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/64—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
AT02724673T 2001-05-07 2002-05-02 3-hydroxymethylbenzo b thiophen-derivate und verfahren zu deren herstellung ATE404551T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2001135928 2001-05-07

Publications (1)

Publication Number Publication Date
ATE404551T1 true ATE404551T1 (de) 2008-08-15

Family

ID=18983308

Family Applications (1)

Application Number Title Priority Date Filing Date
AT02724673T ATE404551T1 (de) 2001-05-07 2002-05-02 3-hydroxymethylbenzo b thiophen-derivate und verfahren zu deren herstellung

Country Status (13)

Country Link
US (1) US6774245B2 (de)
EP (1) EP1298130B1 (de)
JP (1) JP3999131B2 (de)
KR (1) KR20030031486A (de)
CN (1) CN1205204C (de)
AT (1) ATE404551T1 (de)
CA (1) CA2414298A1 (de)
DE (1) DE60228182D1 (de)
HK (1) HK1052352B (de)
NO (1) NO20030058L (de)
NZ (1) NZ523407A (de)
PL (1) PL358478A1 (de)
WO (1) WO2002090345A1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ522150A (en) * 2001-02-22 2006-03-31 Teijin Ltd Benzo[b]thiophene derivatives and processes for preparing the same
CL2004001034A1 (es) * 2003-05-14 2005-03-28 Teijin Pharma Ltd Formas cristalinas de acido 4-(1-((,etilbenzotiofen-3-il)me til)benzimidazol-2-iltio)butanoico; procedimiento de preparacion de las formas cristalinas; composicion farmaceutica; y su uso para el tratamiento de enfermedades inflamatorias, alergicas, r
JP4387360B2 (ja) * 2003-08-22 2009-12-16 帝人ファーマ株式会社 キマーゼ阻害剤を有効成分として含有する薬剤
JPWO2006052026A1 (ja) * 2004-11-12 2008-05-29 帝人ファーマ株式会社 ベンズイミダゾール誘導体の酸性塩及びその結晶
BRPI0617924A2 (pt) 2005-10-27 2016-08-23 Teijin Pharma Ltd processo de produção, e, composto
TW200734321A (en) 2005-10-27 2007-09-16 Teijin Pharma Ltd Benzo [b] thiophen derivatives and a process for producing benzo [b] thiophen derivatives
CN102850246B (zh) * 2012-07-10 2015-04-22 江西理工大学 一种苯胺类衍生物引入巯基的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6320060B1 (en) * 1998-03-31 2001-11-20 Shionogi & Co., Ltd. Process for producing 5-hydroxybenzo[b] thiophene-3-carboxylic acid derivatives
CN1198819C (zh) 2000-01-17 2005-04-27 帝人株式会社 苯并咪唑衍生物

Also Published As

Publication number Publication date
EP1298130B1 (de) 2008-08-13
WO2002090345A1 (en) 2002-11-14
AU2002255294C1 (en) 2002-11-18
US20030191325A1 (en) 2003-10-09
KR20030031486A (ko) 2003-04-21
HK1052352A1 (en) 2003-09-11
HK1052352B (zh) 2008-11-07
CN1462271A (zh) 2003-12-17
EP1298130A1 (de) 2003-04-02
EP1298130A4 (de) 2005-03-30
NZ523407A (en) 2005-04-29
NO20030058L (no) 2003-03-05
NO20030058D0 (no) 2003-01-06
JP3999131B2 (ja) 2007-10-31
CN1205204C (zh) 2005-06-08
PL358478A1 (en) 2004-08-09
CA2414298A1 (en) 2002-12-30
US6774245B2 (en) 2004-08-10
DE60228182D1 (de) 2008-09-25
JPWO2002090345A1 (ja) 2004-08-26

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Legal Events

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