ATE23862T1 - 6-(aminomethyl)-penicillansaeure-1,1-dioxid-este und zwischenprodukte. - Google Patents

6-(aminomethyl)-penicillansaeure-1,1-dioxid-este und zwischenprodukte.

Info

Publication number
ATE23862T1
ATE23862T1 AT84303736T AT84303736T ATE23862T1 AT E23862 T1 ATE23862 T1 AT E23862T1 AT 84303736 T AT84303736 T AT 84303736T AT 84303736 T AT84303736 T AT 84303736T AT E23862 T1 ATE23862 T1 AT E23862T1
Authority
AT
Austria
Prior art keywords
aminomethyl
dioxide
ests
intermediate products
acid
Prior art date
Application number
AT84303736T
Other languages
English (en)
Inventor
Wayne Ernest Barth
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE23862T1 publication Critical patent/ATE23862T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT84303736T 1983-06-06 1984-06-04 6-(aminomethyl)-penicillansaeure-1,1-dioxid-este und zwischenprodukte. ATE23862T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US50145183A 1983-06-06 1983-06-06
US06/577,478 US4536393A (en) 1983-06-06 1984-02-06 6-(Aminomethyl)penicillanic acid 1,1-dioxide esters and intermediates therefor
EP84303736A EP0128719B1 (de) 1983-06-06 1984-06-04 6-(Aminomethyl)-Penicillansäure-1,1-Dioxid-Ester und Zwischenprodukte

Publications (1)

Publication Number Publication Date
ATE23862T1 true ATE23862T1 (de) 1986-12-15

Family

ID=27053819

Family Applications (1)

Application Number Title Priority Date Filing Date
AT84303736T ATE23862T1 (de) 1983-06-06 1984-06-04 6-(aminomethyl)-penicillansaeure-1,1-dioxid-este und zwischenprodukte.

Country Status (19)

Country Link
US (1) US4536393A (de)
EP (1) EP0128719B1 (de)
KR (1) KR870000323B1 (de)
AT (1) ATE23862T1 (de)
AU (1) AU551338B2 (de)
CA (1) CA1206957A (de)
DE (1) DE3461467D1 (de)
DK (1) DK275784A (de)
ES (1) ES533146A0 (de)
FI (1) FI842254A (de)
GR (1) GR82215B (de)
HU (1) HU193930B (de)
IL (1) IL72005A (de)
NO (1) NO842249L (de)
NZ (1) NZ208382A (de)
PH (1) PH19077A (de)
PL (1) PL143943B1 (de)
PT (1) PT78688A (de)
YU (1) YU97384A (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4590073A (en) * 1984-10-22 1986-05-20 Pfizer Inc. 6-substituted penicillanic acid 1,1-dioxide compounds
US4613462A (en) * 1985-07-02 1986-09-23 Pfizer, Inc. 6-substituted penicillanic acid 1,1-dioxide compounds
US4855419A (en) * 1987-06-16 1989-08-08 University Of Cincinnati Application of 4-[1-oxoalkyl]-2,5-oxazolidinediones in selective stereospecific formation of biologically active α-lactams
US5006661A (en) * 1987-06-16 1991-04-09 University Of Cincinnati Selective stereospecific biologically active beta-lactams
GB2206579B (en) * 1987-07-10 1991-05-29 Erba Farmitalia 6a and 6b-(substituted methyl)-penicillanic acid derivatives

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3487079A (en) * 1966-01-14 1969-12-30 Bristol Myers Co Certain alpha-amino bicyclic beta-lactam carboxylic acids
US4207323A (en) * 1975-11-21 1980-06-10 Merck & Co., Inc. 6-Substituted methyl penicillins, derivatives and analogues thereof
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
US4237051A (en) * 1979-04-19 1980-12-02 Schering Corporation Stereospecific production of 6- or 7-carbon-substituted-β-lactams
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4309347A (en) * 1979-05-16 1982-01-05 Pfizer Inc. Penicillanoyloxymethyl penicillanate 1,1,1',1'-tetraoxide
DE2927004A1 (de) * 1979-07-04 1981-05-27 Bayer Ag, 5090 Leverkusen Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4260598A (en) * 1979-10-22 1981-04-07 Pfizer Inc. Method for increasing antibacterial effectiveness of a β-lactam antibiotic
US4342768A (en) * 1979-10-22 1982-08-03 Pfizer Inc. Bis-esters of 1,1-alkanediols with 6-beta-hydroxymethylpenicillanic acid 1,1-dioxide and beta-lactam antibiotics
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
JPS6019908B2 (ja) * 1980-04-30 1985-05-18 カネボウ株式会社 １，３−ジオキソレン−２−オン誘導体
CA1212105A (en) * 1980-04-30 1986-09-30 Shoji Ikeda Ampicillin esters and production thereof
EP0069962B1 (de) * 1981-07-15 1985-01-02 Kanebo, Ltd. 1,1-Dioxopenicillansäure-Ester, Verfahren zu seiner Herstellung und seine Verwendung als Beta-lactamase Hemmstoff
JPS5832882A (ja) * 1981-07-18 1983-02-25 Kanebo Ltd ６−〔（ヘキサヒドロ−１ｈ−アゼピン−１−イル）メチレンアミノ〕ペニシラン酸の新規エステルおよびその製造法

Also Published As

Publication number Publication date
ES8506023A1 (es) 1985-06-01
ES533146A0 (es) 1985-06-01
KR850000445A (ko) 1985-02-27
FI842254A0 (fi) 1984-06-05
DE3461467D1 (en) 1987-01-15
DK275784D0 (da) 1984-06-04
IL72005A (en) 1988-02-29
CA1206957A (en) 1986-07-02
HU193930B (en) 1987-12-28
IL72005A0 (en) 1984-10-31
PT78688A (en) 1984-07-01
NO842249L (no) 1984-12-07
PL143943B1 (en) 1988-03-31
HUT34202A (en) 1985-02-28
US4536393A (en) 1985-08-20
EP0128719B1 (de) 1986-11-26
YU97384A (en) 1986-06-30
PL248044A1 (en) 1985-03-26
FI842254A (fi) 1984-12-07
NZ208382A (en) 1987-05-29
AU551338B2 (en) 1986-04-24
EP0128719A1 (de) 1984-12-19
AU2907884A (en) 1984-12-13
PH19077A (en) 1985-12-19
DK275784A (da) 1984-12-07
KR870000323B1 (ko) 1987-02-27
GR82215B (de) 1984-12-13

Similar Documents

Publication Publication Date Title
SE8003603L (sv) Bis-estrar av metandiol med penicilliner och penicillansyra-1,1-dioxid
IT8220820A0 (it) Processo per l'idrogenolosi di esteri di acidi carbossilici.
DE3868886D1 (de) Fettsaeure-zusammensetzungen.
NO874251L (no) Kryssbundete estere av hyaluronsyre.
DE3875286T2 (de) Essentielle fettsaeure enthaltende zusammensetzungen.
NO885601D0 (no) Eventuelt kvataererte fettsyreestre av oxalkylerte alkyl-alkylendiaminer.
DE3583220D1 (de) Verwendung von dipeptidderivaten fuer die herstellung von arzneimitteln zur behandlung von an amyotropher lateralsklerose erkrankten.
DK0652208T3 (da) Phenylalkan(en)syrer
IT7828313A0 (it) Procedimento per la produzione di acidi carbossilici e/o di loro esteri.
MY104306A (en) Diasteriomeric 5r, 6s-6-(1r-hydroxyethyl)-2-(cis-1-oxo- 3-thiolanythio)-2-penem-3-carboxylic acids.
ATE23862T1 (de) 6-(aminomethyl)-penicillansaeure-1,1-dioxid-este und zwischenprodukte.
BE877351A (fr) Produits de traitement d'etats de seborrhee
IE820342L (en) Penicillins
IT1224636B (it) Esteri penem 6 sostituiti come agenti antinfiammatori e antidegenerativi.
NO872439D0 (no) Fremgangsmaate for fremstilling av fettsyrer.
DE3783412D1 (de) Herstellungsverfahren von substituierten benzoesaeureestern.
ATE66459T1 (de) Herstellungsverfahren von trifluormethylverbindungen.
PT88578A (pt) Process for the manufacture of 2,6-methanopyrrolo-3-benzazocines of intermediates useful for their manufacture and of pharmaceutical compositions containing them
BA97159B1 (bs) Postupak za dobivanje 1,1-dioksida penicilanske kiseline i njegovih estara

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee