DK275784D0 - 6-(aminomethyl)penicillansyre-1,1-dioxid-estere, som er hydrolyserbare under fysiologiske betingelser, og aminobeskyttede 6-(aminomethyl)penicillansyre-forbindelser til anvendelse som mellemprodukter herfor - Google Patents
6-(aminomethyl)penicillansyre-1,1-dioxid-estere, som er hydrolyserbare under fysiologiske betingelser, og aminobeskyttede 6-(aminomethyl)penicillansyre-forbindelser til anvendelse som mellemprodukter herforInfo
- Publication number
- DK275784D0 DK275784D0 DK275784A DK275784A DK275784D0 DK 275784 D0 DK275784 D0 DK 275784D0 DK 275784 A DK275784 A DK 275784A DK 275784 A DK275784 A DK 275784A DK 275784 D0 DK275784 D0 DK 275784D0
- Authority
- DK
- Denmark
- Prior art keywords
- aminomethyl
- penicillanic acid
- physiological conditions
- under physiological
- lysable
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US50145183A | 1983-06-06 | 1983-06-06 | |
US06/577,478 US4536393A (en) | 1983-06-06 | 1984-02-06 | 6-(Aminomethyl)penicillanic acid 1,1-dioxide esters and intermediates therefor |
Publications (2)
Publication Number | Publication Date |
---|---|
DK275784D0 true DK275784D0 (da) | 1984-06-04 |
DK275784A DK275784A (da) | 1984-12-07 |
Family
ID=27053819
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK275784A DK275784A (da) | 1983-06-06 | 1984-06-04 | 6-(aminomethyl)penicillansyre-1,1-dioxid-estere, som er hydrolyserbare under fysiologiske betingelser, og aminobeskyttede 6-(aminomethyl)penicillansyre-forbindelser til anvendelse som mellemprodukter herfor |
Country Status (19)
Country | Link |
---|---|
US (1) | US4536393A (da) |
EP (1) | EP0128719B1 (da) |
KR (1) | KR870000323B1 (da) |
AT (1) | ATE23862T1 (da) |
AU (1) | AU551338B2 (da) |
CA (1) | CA1206957A (da) |
DE (1) | DE3461467D1 (da) |
DK (1) | DK275784A (da) |
ES (1) | ES533146A0 (da) |
FI (1) | FI842254A (da) |
GR (1) | GR82215B (da) |
HU (1) | HU193930B (da) |
IL (1) | IL72005A (da) |
NO (1) | NO842249L (da) |
NZ (1) | NZ208382A (da) |
PH (1) | PH19077A (da) |
PL (1) | PL143943B1 (da) |
PT (1) | PT78688A (da) |
YU (1) | YU97384A (da) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4590073A (en) * | 1984-10-22 | 1986-05-20 | Pfizer Inc. | 6-substituted penicillanic acid 1,1-dioxide compounds |
US4613462A (en) * | 1985-07-02 | 1986-09-23 | Pfizer, Inc. | 6-substituted penicillanic acid 1,1-dioxide compounds |
US4855419A (en) * | 1987-06-16 | 1989-08-08 | University Of Cincinnati | Application of 4-[1-oxoalkyl]-2,5-oxazolidinediones in selective stereospecific formation of biologically active α-lactams |
US5006661A (en) * | 1987-06-16 | 1991-04-09 | University Of Cincinnati | Selective stereospecific biologically active beta-lactams |
GB2206579B (en) * | 1987-07-10 | 1991-05-29 | Erba Farmitalia | 6a and 6b-(substituted methyl)-penicillanic acid derivatives |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3487079A (en) * | 1966-01-14 | 1969-12-30 | Bristol Myers Co | Certain alpha-amino bicyclic beta-lactam carboxylic acids |
US4207323A (en) * | 1975-11-21 | 1980-06-10 | Merck & Co., Inc. | 6-Substituted methyl penicillins, derivatives and analogues thereof |
US4234579A (en) * | 1977-06-07 | 1980-11-18 | Pfizer Inc. | Penicillanic acid 1,1-dioxides as β-lactamase inhibitors |
IE49881B1 (en) * | 1979-02-13 | 1986-01-08 | Leo Pharm Prod Ltd | B-lactam intermediates |
US4237051A (en) * | 1979-04-19 | 1980-12-02 | Schering Corporation | Stereospecific production of 6- or 7-carbon-substituted-β-lactams |
US4244951A (en) * | 1979-05-16 | 1981-01-13 | Pfizer Inc. | Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide |
US4309347A (en) * | 1979-05-16 | 1982-01-05 | Pfizer Inc. | Penicillanoyloxymethyl penicillanate 1,1,1',1'-tetraoxide |
DE2927004A1 (de) * | 1979-07-04 | 1981-05-27 | Bayer Ag, 5090 Leverkusen | Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel |
US4342768A (en) * | 1979-10-22 | 1982-08-03 | Pfizer Inc. | Bis-esters of 1,1-alkanediols with 6-beta-hydroxymethylpenicillanic acid 1,1-dioxide and beta-lactam antibiotics |
US4260598A (en) * | 1979-10-22 | 1981-04-07 | Pfizer Inc. | Method for increasing antibacterial effectiveness of a β-lactam antibiotic |
US4287181A (en) * | 1979-10-22 | 1981-09-01 | Pfizer Inc. | Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors |
JPS6019908B2 (ja) * | 1980-04-30 | 1985-05-18 | カネボウ株式会社 | 1,3−ジオキソレン−2−オン誘導体 |
CA1212105A (en) * | 1980-04-30 | 1986-09-30 | Shoji Ikeda | Ampicillin esters and production thereof |
DE3261759D1 (en) * | 1981-07-15 | 1985-02-14 | Kanebo Ltd | Novel ester of 1,1-dioxopenicillanic acid, process for production thereof, and use thereof as beta-lactamase inhibitor |
JPS5832882A (ja) * | 1981-07-18 | 1983-02-25 | Kanebo Ltd | 6−〔(ヘキサヒドロ−1h−アゼピン−1−イル)メチレンアミノ〕ペニシラン酸の新規エステルおよびその製造法 |
-
1984
- 1984-02-06 US US06/577,478 patent/US4536393A/en not_active Expired - Lifetime
- 1984-06-01 PH PH30754A patent/PH19077A/en unknown
- 1984-06-04 EP EP84303736A patent/EP0128719B1/en not_active Expired
- 1984-06-04 PT PT78688A patent/PT78688A/pt unknown
- 1984-06-04 DK DK275784A patent/DK275784A/da not_active Application Discontinuation
- 1984-06-04 GR GR74910A patent/GR82215B/el unknown
- 1984-06-04 IL IL72005A patent/IL72005A/xx unknown
- 1984-06-04 DE DE8484303736T patent/DE3461467D1/de not_active Expired
- 1984-06-04 AT AT84303736T patent/ATE23862T1/de not_active IP Right Cessation
- 1984-06-04 PL PL1984248044A patent/PL143943B1/pl unknown
- 1984-06-04 CA CA000455813A patent/CA1206957A/en not_active Expired
- 1984-06-05 AU AU29078/84A patent/AU551338B2/en not_active Ceased
- 1984-06-05 NZ NZ208382A patent/NZ208382A/en unknown
- 1984-06-05 ES ES533146A patent/ES533146A0/es active Granted
- 1984-06-05 YU YU00973/84A patent/YU97384A/xx unknown
- 1984-06-05 FI FI842254A patent/FI842254A/fi not_active Application Discontinuation
- 1984-06-05 HU HU842177A patent/HU193930B/hu unknown
- 1984-06-05 NO NO842249A patent/NO842249L/no unknown
- 1984-06-05 KR KR1019840003121A patent/KR870000323B1/ko not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
GR82215B (da) | 1984-12-13 |
NZ208382A (en) | 1987-05-29 |
FI842254A (fi) | 1984-12-07 |
IL72005A0 (en) | 1984-10-31 |
EP0128719A1 (en) | 1984-12-19 |
YU97384A (en) | 1986-06-30 |
PT78688A (en) | 1984-07-01 |
KR870000323B1 (ko) | 1987-02-27 |
ATE23862T1 (de) | 1986-12-15 |
ES8506023A1 (es) | 1985-06-01 |
ES533146A0 (es) | 1985-06-01 |
PH19077A (en) | 1985-12-19 |
PL143943B1 (en) | 1988-03-31 |
HUT34202A (en) | 1985-02-28 |
US4536393A (en) | 1985-08-20 |
HU193930B (en) | 1987-12-28 |
DE3461467D1 (en) | 1987-01-15 |
AU551338B2 (en) | 1986-04-24 |
FI842254A0 (fi) | 1984-06-05 |
PL248044A1 (en) | 1985-03-26 |
NO842249L (no) | 1984-12-07 |
EP0128719B1 (en) | 1986-11-26 |
DK275784A (da) | 1984-12-07 |
AU2907884A (en) | 1984-12-13 |
CA1206957A (en) | 1986-07-02 |
IL72005A (en) | 1988-02-29 |
KR850000445A (ko) | 1985-02-27 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
AHB | Application shelved due to non-payment |