ATE110079T1 - Triazolo(1,5-c>pyrimido(1,4>azine als bronchodilatatoren. - Google Patents

Triazolo(1,5-c>pyrimido(1,4>azine als bronchodilatatoren.

Info

Publication number
ATE110079T1
ATE110079T1 AT89300876T AT89300876T ATE110079T1 AT E110079 T1 ATE110079 T1 AT E110079T1 AT 89300876 T AT89300876 T AT 89300876T AT 89300876 T AT89300876 T AT 89300876T AT E110079 T1 ATE110079 T1 AT E110079T1
Authority
AT
Austria
Prior art keywords
alkyl
pyrimido
triazolo
compounds
bronchodilators
Prior art date
Application number
AT89300876T
Other languages
English (en)
Inventor
James J Wade
Original Assignee
Riker Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Riker Laboratories Inc filed Critical Riker Laboratories Inc
Application granted granted Critical
Publication of ATE110079T1 publication Critical patent/ATE110079T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT89300876T 1988-02-05 1989-01-30 Triazolo(1,5-c>pyrimido(1,4>azine als bronchodilatatoren. ATE110079T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US15244388A 1988-02-05 1988-02-05

Publications (1)

Publication Number Publication Date
ATE110079T1 true ATE110079T1 (de) 1994-09-15

Family

ID=22542946

Family Applications (1)

Application Number Title Priority Date Filing Date
AT89300876T ATE110079T1 (de) 1988-02-05 1989-01-30 Triazolo(1,5-c>pyrimido(1,4>azine als bronchodilatatoren.

Country Status (11)

Country Link
EP (1) EP0327284B1 (de)
JP (1) JP2694990B2 (de)
KR (1) KR890013026A (de)
AT (1) ATE110079T1 (de)
AU (1) AU596764B2 (de)
CA (1) CA1331178C (de)
DE (1) DE68917491T2 (de)
DK (1) DK47489A (de)
IE (1) IE64917B1 (de)
NZ (1) NZ227720A (de)
ZA (1) ZA89639B (de)

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS50116498A (de) * 1974-02-27 1975-09-11
US4572910A (en) * 1983-03-03 1986-02-25 Riker Laboratories, Inc. Triazolo[1,5-c]pyrimidines substituted by nitrogen-containing heterocyclic rings
DK135184A (da) * 1983-03-03 1984-10-10 Riker Laboratories Inc Triazol(4,3-c)- og triazol(1,5-c)pyrimidiner
EP0181282A1 (de) * 1984-10-01 1986-05-14 Ciba-Geigy Ag Triazolochinazolinverbindungen
EP0217748B1 (de) * 1985-09-30 1991-02-06 Ciba-Geigy Ag 2-Substituierte-e-kondensierte[1,5-c]-Pyrimidine, pharmazeutische Zubereitungen und ihre Verwendung
US4639445A (en) * 1985-10-25 1987-01-27 Riker Laboratories Metabolites of triazolo[1,5-c]pyrimidines
HU195822B (en) * 1985-12-30 1988-07-28 Gyogyszerkutato Intezet Process for producing new pyrimido/5,4-b//1,h/oxazine derivatives
AU612331B2 (en) * 1986-09-30 1991-07-11 Ciba-Geigy Ag 2-substituted-e-fused-(1,2,4)triazolo(1,5-c)pyrimidines pharmaceutical compositions
US4734413A (en) * 1987-03-02 1988-03-29 Riker Laboratories, Inc. Substituted 1,2,4-triazolo[1,5-A]triazines as bronchodilators

Also Published As

Publication number Publication date
JP2694990B2 (ja) 1997-12-24
DK47489A (da) 1989-09-21
CA1331178C (en) 1994-08-02
DK47489D0 (da) 1989-02-02
IE64917B1 (en) 1995-09-20
NZ227720A (en) 1992-10-28
AU2959889A (en) 1989-08-10
KR890013026A (ko) 1989-09-20
EP0327284A3 (de) 1991-05-02
DE68917491T2 (de) 1995-02-16
DE68917491D1 (de) 1994-09-22
JPH02149584A (ja) 1990-06-08
ZA89639B (en) 1990-09-26
IE890210L (en) 1989-08-05
EP0327284A2 (de) 1989-08-09
EP0327284B1 (de) 1994-08-17
AU596764B2 (en) 1990-05-10

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