AR247550A1 - Un procedimiento para la preparacion de nuevas carboxamidas aromaticas - Google Patents
Un procedimiento para la preparacion de nuevas carboxamidas aromaticasInfo
- Publication number
- AR247550A1 AR247550A1 AR90317470A AR31747090A AR247550A1 AR 247550 A1 AR247550 A1 AR 247550A1 AR 90317470 A AR90317470 A AR 90317470A AR 31747090 A AR31747090 A AR 31747090A AR 247550 A1 AR247550 A1 AR 247550A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparation
- medicines
- carboxylic acid
- acid amides
- aromatic carboxylic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/088—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
- C07C233/65—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
- C07C233/66—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
- C07C233/67—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
- C07C233/75—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
- C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
- C07C235/44—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
- C07C235/56—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/12—One of the condensed rings being a six-membered aromatic ring the other ring being at least seven-membered
Abstract
PREPARACION DE COMPUESTOS DE FORMULA I, DONDE R1 ES HALOGENO U OR5; R3 Y R4 Y JUNTOS REPRESENTAN ALQUILENO, R5 ES HIDROGENO, ACILO, ALCOXICARBONILO O ALQUILO SUSTITUIDO O NO POR AMINO, DIALQUILAMINO, MORFOLINO, N- METILPIRERAZINO O IMIDAZOLINO Y M ES -CONH- O -NHCO- EN DONDE DICHO PROCEDIMIENTO COMPRENDE HACER REACCIONAR UN COMPUESTO DE FORMULA II, CON UN COMPUESTO DE FORMULA III DONDE AES CARBOXILO O UN DERIVADO REACTIVO RESPECTIVO Y B ES AMINO O A ES UN GRUPO Y B ES CARBOXILO O UN DERIVADO REACTIVO RESPECTIVO Y R'' ES R1 EN DONDE UN GRUPO AMINO ESTA PROTEGIDO, DESPUES DE LO CUAL SE DISOCIA UN GRUPO PROTECTOR ANIMICO QUE PUEDA ESTAR PRESENTE.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH281889 | 1989-07-28 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR247550A1 true AR247550A1 (es) | 1995-01-31 |
Family
ID=4242276
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR90317470A AR247550A1 (es) | 1989-07-28 | 1990-07-26 | Un procedimiento para la preparacion de nuevas carboxamidas aromaticas |
Country Status (27)
Country | Link |
---|---|
US (1) | US5128470A (es) |
EP (1) | EP0410358B1 (es) |
JP (1) | JPH075533B2 (es) |
KR (1) | KR910002775A (es) |
AR (1) | AR247550A1 (es) |
AT (1) | ATE95167T1 (es) |
AU (1) | AU637623B2 (es) |
CA (1) | CA2020887A1 (es) |
CZ (1) | CZ277709B6 (es) |
DE (1) | DE59002899D1 (es) |
DK (1) | DK0410358T3 (es) |
ES (1) | ES2059919T3 (es) |
FI (1) | FI903740A0 (es) |
HU (1) | HU204773B (es) |
IE (1) | IE902734A1 (es) |
IL (1) | IL95144A (es) |
IS (1) | IS3611A7 (es) |
MC (1) | MC2135A1 (es) |
MX (1) | MX21691A (es) |
MY (1) | MY106704A (es) |
NO (1) | NO903351L (es) |
NZ (1) | NZ234595A (es) |
PH (1) | PH27297A (es) |
PT (1) | PT94839A (es) |
RU (1) | RU1811525C (es) |
YU (1) | YU141690A (es) |
ZA (1) | ZA905738B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0617020A1 (en) * | 1992-04-02 | 1994-09-28 | Shudo, Koichi, Prof. Dr. | Carboxylic acid derivatives having retinoic acid-like activity |
US5631369A (en) * | 1994-08-31 | 1997-05-20 | Eli Lilly And Company | Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceutical agents |
FR2759368B1 (fr) | 1997-02-10 | 2001-06-01 | Galderma Rech Dermatologique | Composes biaromatiques, compositions les contenant et utilisations |
US6664293B2 (en) * | 1999-02-26 | 2003-12-16 | Fujiwawa Pharmaceutical Co., Ltd. | Amide compounds for the potentiation of cholinergic activity |
CA2361819A1 (en) * | 1999-03-17 | 2000-09-21 | Astrazeneca Ab | Amide derivatives |
US6316475B1 (en) * | 2000-11-17 | 2001-11-13 | Abbott Laboratories | Aminoalkoxybiphenylcarboxamides as histamine-3 receptor ligands and their therapeutic applications |
RU2006106920A (ru) | 2003-08-06 | 2007-09-20 | Синомикс Инк. (Us) | Гетеро-олигомерные вкусовые рецепторы t1r, клеточные линии, которые экспрессируют указанные рецепторы и вкусовые соединения |
CA2584307A1 (en) * | 2004-10-15 | 2006-06-15 | Bayer Pharmaceuticals Corporation | Indane amides with antiproliferative activity |
US20100158829A1 (en) * | 2008-12-24 | 2010-06-24 | Conopco, Inc., D/B/A Unilever | Method and Composition for Color Modulation |
US8653299B2 (en) | 2011-03-17 | 2014-02-18 | Allergan, Inc. | Dihydronaphthalene and naphthalene derivatives as N-formyl peptide receptor like-1 (FPRL-1) receptor modulators |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3202100A1 (de) * | 1982-01-23 | 1983-08-04 | Basf Ag, 6700 Ludwigshafen | Substituierte benzoesaeure-4-hydroxyanilide, ihre herstellung und diese enthaltende pharmazeutische zubereitungen |
JPS58140054A (ja) * | 1982-02-10 | 1983-08-19 | Sumitomo Chem Co Ltd | インダニルベンツアミド誘導体、その製造法およびこれらを有効成分として含有する農園芸用殺菌剤 |
EP0170105B1 (en) * | 1984-07-07 | 1990-10-17 | Koichi Prof. Dr. Shudo | Benzoic acid derivatives |
LU86258A1 (fr) * | 1986-01-21 | 1987-09-03 | Rech Dermatologiques C I R D S | Composes benzamido aromatique,leur procede de preparation et leur utilisation en medecine humaine ou veterinaire et en cosmetique |
GB8617653D0 (en) * | 1986-07-18 | 1986-08-28 | Ici Plc | Amide derivatives |
US4808631A (en) * | 1986-11-07 | 1989-02-28 | Hoffmann-La Roche Inc. | Aromatic acid derivatives |
US4992576A (en) * | 1987-01-12 | 1991-02-12 | Eli Lilly And Company | Intermediates for leukotriene antagonists |
CA1320490C (en) | 1987-01-12 | 1993-07-20 | Darrel M. Gapinski | Anti-inflammatory agents |
JPS6471843A (en) * | 1987-09-11 | 1989-03-16 | Meiji Seika Kaisha | Novel substituted benzoic acid anilide derivative and plant disease injury controlling agent containing said derivative as active ingredient |
-
1990
- 1990-07-11 CA CA002020887A patent/CA2020887A1/en not_active Abandoned
- 1990-07-12 US US07/551,831 patent/US5128470A/en not_active Expired - Fee Related
- 1990-07-19 YU YU141690A patent/YU141690A/sh unknown
- 1990-07-20 ZA ZA905738A patent/ZA905738B/xx unknown
- 1990-07-20 NZ NZ234595A patent/NZ234595A/xx unknown
- 1990-07-20 IL IL9514490A patent/IL95144A/en not_active IP Right Cessation
- 1990-07-23 AT AT90114101T patent/ATE95167T1/de not_active IP Right Cessation
- 1990-07-23 EP EP90114101A patent/EP0410358B1/de not_active Expired - Lifetime
- 1990-07-23 ES ES90114101T patent/ES2059919T3/es not_active Expired - Lifetime
- 1990-07-23 MX MX2169190A patent/MX21691A/es unknown
- 1990-07-23 DK DK90114101.0T patent/DK0410358T3/da active
- 1990-07-23 HU HU904577A patent/HU204773B/hu not_active IP Right Cessation
- 1990-07-23 DE DE90114101T patent/DE59002899D1/de not_active Expired - Fee Related
- 1990-07-24 MC MC902141A patent/MC2135A1/xx unknown
- 1990-07-25 JP JP2195092A patent/JPH075533B2/ja not_active Expired - Lifetime
- 1990-07-26 FI FI903740A patent/FI903740A0/fi not_active IP Right Cessation
- 1990-07-26 AU AU59892/90A patent/AU637623B2/en not_active Ceased
- 1990-07-26 MY MYPI90001257A patent/MY106704A/en unknown
- 1990-07-26 AR AR90317470A patent/AR247550A1/es active
- 1990-07-27 IS IS3611A patent/IS3611A7/is unknown
- 1990-07-27 PT PT94839A patent/PT94839A/pt not_active Application Discontinuation
- 1990-07-27 CZ CS903740A patent/CZ277709B6/cs unknown
- 1990-07-27 RU SU904830538A patent/RU1811525C/ru active
- 1990-07-27 IE IE273490A patent/IE902734A1/en unknown
- 1990-07-27 PH PH40913A patent/PH27297A/en unknown
- 1990-07-27 KR KR1019900011436A patent/KR910002775A/ko not_active Application Discontinuation
- 1990-07-27 NO NO90903351A patent/NO903351L/no unknown
Also Published As
Publication number | Publication date |
---|---|
HUT54106A (en) | 1991-01-28 |
NZ234595A (en) | 1992-10-28 |
JPH0374353A (ja) | 1991-03-28 |
PT94839A (pt) | 1991-03-20 |
AU637623B2 (en) | 1993-06-03 |
MY106704A (en) | 1995-07-31 |
NO903351L (no) | 1991-01-29 |
CS374090A3 (en) | 1992-01-15 |
EP0410358B1 (de) | 1993-09-29 |
DK0410358T3 (da) | 1993-12-13 |
EP0410358A1 (de) | 1991-01-30 |
AU5989290A (en) | 1991-01-31 |
ES2059919T3 (es) | 1994-11-16 |
NO903351D0 (no) | 1990-07-27 |
ATE95167T1 (de) | 1993-10-15 |
JPH075533B2 (ja) | 1995-01-25 |
IS3611A7 (is) | 1991-01-29 |
CZ277709B6 (en) | 1993-03-17 |
FI903740A0 (fi) | 1990-07-26 |
KR910002775A (ko) | 1991-02-26 |
HU904577D0 (en) | 1990-12-28 |
RU1811525C (ru) | 1993-04-23 |
IL95144A0 (en) | 1991-06-10 |
US5128470A (en) | 1992-07-07 |
IL95144A (en) | 1994-10-07 |
HU204773B (en) | 1992-02-28 |
MC2135A1 (fr) | 1992-01-14 |
DE59002899D1 (de) | 1993-11-04 |
ZA905738B (en) | 1991-03-27 |
CA2020887A1 (en) | 1991-01-29 |
MX21691A (es) | 1993-10-01 |
PH27297A (en) | 1993-05-04 |
YU141690A (sh) | 1993-05-28 |
IE902734A1 (en) | 1991-02-27 |
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