AR241421A1 - Procedimiento para la elaboracion de azacicloalcanos-sustitutivos. - Google Patents
Procedimiento para la elaboracion de azacicloalcanos-sustitutivos.Info
- Publication number
- AR241421A1 AR241421A1 AR86303163A AR30316386A AR241421A1 AR 241421 A1 AR241421 A1 AR 241421A1 AR 86303163 A AR86303163 A AR 86303163A AR 30316386 A AR30316386 A AR 30316386A AR 241421 A1 AR241421 A1 AR 241421A1
- Authority
- AR
- Argentina
- Prior art keywords
- elaboration
- azacycloalkanes
- proceeding
- substituents
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
- C07C205/55—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
- C07C205/56—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups bound to carbon atoms of six-membered aromatic rings and carboxyl groups bound to acyclic carbon atoms of the carbon skeleton
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Indole Compounds (AREA)
- Steroid Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyrrole Compounds (AREA)
Abstract
PROCEDIMIENTO PARA LA ELABORACION DE COMPUESTOS DE AZACICLOALCANOS SUSTITUIDOS DE FORMULA I, R1 ES -ALQUILO, -ALQUENILO, -ALQUINILO, - CICLOALQUIL-ALQUILO O BENCILO, R2 ES H O -ALCANOILO Y SUS SALES, A PARTIR DE FORMULA II, DONDE R1 Y R2 TIENEN LOS SIGNIFICADOS INDICADOS O R1 ES HIDROGENO, SE TRANSFORMA CON DIAZOMETANO. SE EMPLEANEN PRODUCTOS FARMACEUTICOS PARA ENFERMEDADES HORMONALES.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH745082 | 1982-12-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR241421A1 true AR241421A1 (es) | 1992-07-31 |
Family
ID=4325317
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR83295196A AR241590A1 (es) | 1982-12-21 | 1983-12-21 | Procedimiento para elaborar 1-fenil-3-azabiciclo(3.1.0)hexan-2,4-dionas y sus sales. |
AR86303163A AR241421A1 (es) | 1982-12-21 | 1986-02-18 | Procedimiento para la elaboracion de azacicloalcanos-sustitutivos. |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR83295196A AR241590A1 (es) | 1982-12-21 | 1983-12-21 | Procedimiento para elaborar 1-fenil-3-azabiciclo(3.1.0)hexan-2,4-dionas y sus sales. |
Country Status (23)
Country | Link |
---|---|
US (1) | US4839379A (es) |
EP (1) | EP0114033B1 (es) |
JP (1) | JPS59118748A (es) |
KR (1) | KR900009007B1 (es) |
AR (2) | AR241590A1 (es) |
AT (1) | ATE37871T1 (es) |
AU (1) | AU565914B2 (es) |
CA (1) | CA1208649A (es) |
DD (1) | DD222306A5 (es) |
DE (1) | DE3378208D1 (es) |
DK (1) | DK165977C (es) |
ES (3) | ES528179A0 (es) |
FI (1) | FI79838C (es) |
GR (1) | GR81359B (es) |
HK (1) | HK24291A (es) |
HU (1) | HU192836B (es) |
IE (1) | IE56421B1 (es) |
IL (1) | IL70478A (es) |
NO (1) | NO163529C (es) |
NZ (1) | NZ206654A (es) |
PH (1) | PH22052A (es) |
PT (1) | PT77857B (es) |
ZA (1) | ZA839437B (es) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0166692B1 (de) * | 1984-06-20 | 1990-07-11 | Ciba-Geigy Ag | Substituierte Azabicycloheptane, ihre Verwendung, pharmazeutische Präparate, welche diese Verbindungen enthalten, und Verfahren zur Herstellung dieser Verbindungen |
CH683151A5 (de) * | 1991-04-24 | 1994-01-31 | Ciba Geigy Ag | Antikonzeption bei weiblichen Primaten ohne Beeinflussung des menstruellen Zyklus. |
WO1993007141A1 (en) * | 1991-10-11 | 1993-04-15 | Smithkline Beecham Corporation | Heterocyclic 3-phenylpyrrolidin-2-ones, their preparation and use for the manufacture of a medicament for inhibiting tumor necrosis factor production |
US5511916A (en) * | 1991-12-06 | 1996-04-30 | Aldon Pattern, Inc. | Shipping container for dunnage |
RU2007102290A (ru) * | 2004-07-22 | 2008-08-27 | Вайет (Us) | Способ лечения нарушений и заболеваний нервной системы |
EP1773320A1 (en) * | 2004-07-22 | 2007-04-18 | Wyeth | Method for treating nervous system disorders and conditions |
BRPI0512182A (pt) * | 2004-07-22 | 2008-02-19 | Wyeth Corp | método para o tratamento de condições e desordens do sistema nervoso |
JP2009502798A (ja) * | 2005-07-21 | 2009-01-29 | ワイス | 神経系障害および状態の処置方法 |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE548074A (es) * | ||||
US2673205A (en) * | 1951-02-13 | 1954-03-23 | Ciba Pharm Prod Inc | 3-disubstituted dioxopiperidines and the manufacture thereof |
US2848455A (en) * | 1955-07-18 | 1958-08-19 | Ciba Pharm Prod Inc | Alpha-(p-amino-phenyl)-alpha-lower alkyl glutarimides |
GB1015618A (en) * | 1962-04-10 | 1966-01-05 | Aspro Nicholas Ltd | Glutarimide therapeutic compositions |
US3166571A (en) * | 1962-06-06 | 1965-01-19 | American Cyanamid Co | 1-phenyl-1, 2-cyclopropane dicarboximides |
US3621012A (en) * | 1969-08-18 | 1971-11-16 | Union Carbide Corp | Oxidation of lactams to cyclic imides |
US4164404A (en) * | 1973-06-25 | 1979-08-14 | American Cyanamid Company | Dithiindicarboximide, dithiolanedicarboximide, thiapyrandicarboximide and pyrandicarboximide derivatives as plant growth regulants |
US4231935A (en) * | 1975-07-31 | 1980-11-04 | American Cyanamid Company | 1-Phenyl-3-azabicyclo[3.1.0]hexanes |
US4131611A (en) * | 1975-07-31 | 1978-12-26 | American Cyanamid Company | Azabicyclohexanes |
IL65843A (en) * | 1977-08-11 | 1986-12-31 | American Cyanamid Co | Pharmaceutical compositions for the treatment of depression containing 3-aza-bicyclo(3.1.0)hexane derivatives and certain novel compounds of this type |
US4289762A (en) * | 1980-06-27 | 1981-09-15 | Merrell Dow Pharmaceuticals Inc. | 10-(1,2-Propadienyl) steroids as irreversible aromatase inhibitors |
US4322416A (en) * | 1980-06-27 | 1982-03-30 | Merrell Dow Pharmaceuticals Inc. | 10-Alkynyl steroids |
DE3121153A1 (de) * | 1981-05-22 | 1982-12-09 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | "verwendung von aromatase-hemmern zur prophylaxe und therapie der prostatahyperplasie" |
US4435419A (en) * | 1981-07-01 | 1984-03-06 | American Cyanamid Company | Method of treating depression using azabicyclohexanes |
EP0166692B1 (de) * | 1984-06-20 | 1990-07-11 | Ciba-Geigy Ag | Substituierte Azabicycloheptane, ihre Verwendung, pharmazeutische Präparate, welche diese Verbindungen enthalten, und Verfahren zur Herstellung dieser Verbindungen |
-
1983
- 1983-12-15 AT AT83810594T patent/ATE37871T1/de not_active IP Right Cessation
- 1983-12-15 DE DE8383810594T patent/DE3378208D1/de not_active Expired
- 1983-12-15 EP EP83810594A patent/EP0114033B1/de not_active Expired
- 1983-12-19 ES ES528179A patent/ES528179A0/es active Granted
- 1983-12-19 FI FI834663A patent/FI79838C/fi not_active IP Right Cessation
- 1983-12-19 IL IL70478A patent/IL70478A/xx unknown
- 1983-12-19 DD DD83258172A patent/DD222306A5/de not_active IP Right Cessation
- 1983-12-19 CA CA000443588A patent/CA1208649A/en not_active Expired
- 1983-12-20 NZ NZ206654A patent/NZ206654A/en unknown
- 1983-12-20 PH PH30009A patent/PH22052A/en unknown
- 1983-12-20 AU AU22704/83A patent/AU565914B2/en not_active Ceased
- 1983-12-20 KR KR1019830006031A patent/KR900009007B1/ko not_active IP Right Cessation
- 1983-12-20 ZA ZA839437A patent/ZA839437B/xx unknown
- 1983-12-20 PT PT77857A patent/PT77857B/pt not_active IP Right Cessation
- 1983-12-20 JP JP58238994A patent/JPS59118748A/ja active Pending
- 1983-12-20 DK DK586283A patent/DK165977C/da active
- 1983-12-20 NO NO834710A patent/NO163529C/no unknown
- 1983-12-20 HU HU834356A patent/HU192836B/hu not_active IP Right Cessation
- 1983-12-20 GR GR73300A patent/GR81359B/el unknown
- 1983-12-20 IE IE3006/83A patent/IE56421B1/en not_active IP Right Cessation
- 1983-12-21 AR AR83295196A patent/AR241590A1/es active
-
1985
- 1985-05-23 ES ES543431A patent/ES8607941A1/es not_active Expired
- 1985-05-23 ES ES543430A patent/ES8603832A1/es not_active Expired
-
1986
- 1986-02-18 AR AR86303163A patent/AR241421A1/es active
-
1987
- 1987-07-28 US US07/080,240 patent/US4839379A/en not_active Expired - Lifetime
-
1991
- 1991-03-26 HK HK242/91A patent/HK24291A/xx unknown
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