AR240043A1 - Procedimiento para preparar derivados de 2-fenoxi o feniltriometil-3-fluoralilamina. - Google Patents

Procedimiento para preparar derivados de 2-fenoxi o feniltriometil-3-fluoralilamina.

Info

Publication number
AR240043A1
AR240043A1 AR300950A AR30095085A AR240043A1 AR 240043 A1 AR240043 A1 AR 240043A1 AR 300950 A AR300950 A AR 300950A AR 30095085 A AR30095085 A AR 30095085A AR 240043 A1 AR240043 A1 AR 240043A1
Authority
AR
Argentina
Prior art keywords
phenyltryomethyl
fluoralylamine
phenoxy
derivatives
preparing
Prior art date
Application number
AR300950A
Other languages
English (en)
Spanish (es)
Original Assignee
Merell Dow Pharmaceticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merell Dow Pharmaceticals Inc filed Critical Merell Dow Pharmaceticals Inc
Application granted granted Critical
Publication of AR240043A1 publication Critical patent/AR240043A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40Halogenated unsaturated alcohols
    • C07C33/42Halogenated unsaturated alcohols acyclic
    • C07C33/423Halogenated unsaturated alcohols acyclic containing only double bonds as unsaturation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/54Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AR300950A 1984-07-13 1985-07-11 Procedimiento para preparar derivados de 2-fenoxi o feniltriometil-3-fluoralilamina. AR240043A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US63055684A 1984-07-13 1984-07-13

Publications (1)

Publication Number Publication Date
AR240043A1 true AR240043A1 (es) 1990-01-31

Family

ID=24527644

Family Applications (1)

Application Number Title Priority Date Filing Date
AR300950A AR240043A1 (es) 1984-07-13 1985-07-11 Procedimiento para preparar derivados de 2-fenoxi o feniltriometil-3-fluoralilamina.

Country Status (20)

Country Link
EP (1) EP0168013B1 (fi)
JP (1) JPS61257952A (fi)
KR (1) KR900008113B1 (fi)
AR (1) AR240043A1 (fi)
AT (1) ATE32711T1 (fi)
AU (1) AU575973B2 (fi)
CA (1) CA1256453A (fi)
DE (1) DE3561723D1 (fi)
DK (1) DK166878C (fi)
ES (1) ES8603809A1 (fi)
FI (1) FI84057C (fi)
GB (1) GB2162518B (fi)
HU (1) HU195181B (fi)
IE (1) IE58305B1 (fi)
IL (1) IL75739A (fi)
NO (1) NO161313C (fi)
NZ (1) NZ212675A (fi)
PH (1) PH21647A (fi)
PT (1) PT80805B (fi)
ZA (1) ZA855101B (fi)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE71933T1 (de) * 1985-12-05 1992-02-15 Merrell Dow Pharma Nichtaromatische fluoralkylamin-mao-inhibitoren.
EP0283168A3 (en) * 1987-03-16 1989-06-14 American Home Products Corporation Fluorooxirane carboxylates
US4822812A (en) * 1987-05-21 1989-04-18 Merrell Dow Pharmaceuticals Inc. β-(Fluoromethylene)-5-hydroxytryptophan and derivatives and their use as prodrugs for MAO inhibition
US5252608A (en) * 1988-02-25 1993-10-12 Merrell Dow Pharmaceuticals Inc. Inhibitors of lysyl oxidase
US5059714A (en) * 1988-02-25 1991-10-22 Merrell Dow Pharmaceuticals Inc. Inhibitors of lysyl oxidase
US4965288A (en) * 1988-02-25 1990-10-23 Merrell Dow Pharmaceuticals Inc. Inhibitors of lysyl oxidase
US5120764A (en) * 1988-11-01 1992-06-09 Merrell Dow Pharmaceuticals Inc. Inhibitors of lysyl oxidase
US5488188A (en) * 1994-09-29 1996-01-30 Merrell Dow Pharmaceuticals Inc. Process for the preparation of (E)-1-amino-2-(fluoromethylene)-4-(p-fluorophenyl)butane, novel processes for preparing an intermediate thereof, and novel intermediates thereof
US20070293548A1 (en) * 2006-03-31 2007-12-20 Wang Eric Y Inhibitors of semicarbazide-sensitive amine oxidase (SSAO) and VAP-1 mediated adhesion useful for treatment and prevention of diseases
SG10201707020TA (en) 2012-05-02 2017-10-30 Boehringer Ingelheim Int Substituted 3-haloallylamine inhibitors of ssao and uses thereof
WO2024044813A1 (en) * 2022-08-29 2024-03-07 Pharmaxis Ltd. Novel selective inhibitors of lysyl oxidases

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1027611A (en) * 1962-01-04 1966-04-27 May & Baker Ltd Phenoxy- and phenylthio-alkylamines and acid addition salts thereof
US3205136A (en) * 1962-12-24 1965-09-07 Smith Kline French Lab Antidepressant phenyloxyalkylamines
US3513198A (en) * 1965-10-22 1970-05-19 Hoffmann La Roche Aryloxy- and arylthio-acetylenic amines and the salts thereof
CH480306A (de) * 1966-06-03 1969-10-31 Ciba Geigy Verfahren zur Herstellung von schwefelhaltigen Aminen

Also Published As

Publication number Publication date
NO161313B (no) 1989-04-24
NO852810L (no) 1986-01-14
KR860001048A (ko) 1986-02-22
CA1256453A (en) 1989-06-27
JPH0530823B2 (fi) 1993-05-11
EP0168013A1 (en) 1986-01-15
HU195181B (en) 1988-04-28
DK320585A (da) 1986-01-14
PT80805A (en) 1985-08-01
KR900008113B1 (ko) 1990-10-31
PT80805B (pt) 1987-09-18
FI852748L (fi) 1986-01-14
DE3561723D1 (de) 1988-04-07
EP0168013B1 (en) 1988-03-02
ZA855101B (en) 1986-05-28
FI84057C (fi) 1991-10-10
GB2162518A (en) 1986-02-05
NZ212675A (en) 1988-02-29
GB2162518B (en) 1987-11-18
IL75739A0 (en) 1985-11-29
DK166878B (da) 1993-07-26
ES545111A0 (es) 1986-01-01
JPS61257952A (ja) 1986-11-15
IL75739A (en) 1988-07-31
GB8517454D0 (en) 1985-08-14
FI84057B (fi) 1991-06-28
DK166878C (da) 1993-12-13
DK320585D0 (da) 1985-07-12
AU4466085A (en) 1986-01-16
IE851746L (en) 1986-01-13
NO161313C (no) 1989-08-02
HUT38604A (en) 1986-06-30
AU575973B2 (en) 1988-08-11
IE58305B1 (en) 1993-09-08
ES8603809A1 (es) 1986-01-01
PH21647A (en) 1988-01-13
ATE32711T1 (de) 1988-03-15
FI852748A0 (fi) 1985-07-11

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