ES539822A0 - Procedimiento para la preparacion de pirazolopiridinas. - Google Patents
Procedimiento para la preparacion de pirazolopiridinas.Info
- Publication number
- ES539822A0 ES539822A0 ES539822A ES539822A ES539822A0 ES 539822 A0 ES539822 A0 ES 539822A0 ES 539822 A ES539822 A ES 539822A ES 539822 A ES539822 A ES 539822A ES 539822 A0 ES539822 A0 ES 539822A0
- Authority
- ES
- Spain
- Prior art keywords
- pirazolopiridinas
- procedure
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB848401868A GB8401868D0 (en) | 1984-01-25 | 1984-01-25 | Compounds |
GB848430012A GB8430012D0 (en) | 1984-11-28 | 1984-11-28 | Compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
ES539822A0 true ES539822A0 (es) | 1986-05-16 |
ES8607298A1 ES8607298A1 (es) | 1986-05-16 |
Family
ID=26287220
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES539822A Expired ES8607298A1 (es) | 1984-01-25 | 1985-01-24 | Procedimiento para la preparacion de pirazolopiridinas. |
Country Status (5)
Country | Link |
---|---|
US (1) | US4576952A (es) |
EP (1) | EP0151962A3 (es) |
AU (1) | AU3800785A (es) |
ES (1) | ES8607298A1 (es) |
GR (1) | GR850190B (es) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8404584D0 (en) * | 1984-02-22 | 1984-03-28 | Beecham Group Plc | Compounds |
EP0193329A3 (en) * | 1985-02-22 | 1987-08-19 | Beecham Group Plc | Pyrazolopyridines, their preparation and pharmaceutical compositions containing them |
AT382377B (de) * | 1985-04-27 | 1987-02-25 | Beecham Group Plc | Verfahren zur herstellung von neuen 7-substituierten aminopyrazolo(4,3-b)pyridinen |
EP0239191A3 (en) * | 1986-01-30 | 1988-07-20 | Beecham Group Plc | Pyrazolo[4,3-b]pyridine derivatives, process for their preparation and pharmaceutical compositions containing them |
PE20020506A1 (es) * | 2000-08-22 | 2002-07-09 | Glaxo Group Ltd | Derivados de pirazol fusionados como inhibidores de la proteina cinasa |
US7163940B2 (en) * | 2000-12-15 | 2007-01-16 | Smithkline Beecham Corporation | Pyrazolopyridinyl pyrimidine therapeutic compounds |
AU2002239344A1 (en) | 2000-12-15 | 2002-06-24 | Glaxo Group Limited | Pyrazolopyridines |
EP1366048B1 (en) * | 2001-03-08 | 2004-08-25 | SmithKline Beecham Corporation | Pyrazolopyridine derivatives |
WO2002078700A1 (en) * | 2001-03-30 | 2002-10-10 | Smithkline Beecham Corporation | Pyralopyridines, process for their preparation and use as therapteutic compounds |
US20050107400A1 (en) * | 2001-03-30 | 2005-05-19 | Boyd Leslie F. | Use of pyrazolopyridines as therapeutic compounds |
DE60212949T2 (de) * | 2001-04-10 | 2007-01-04 | Smithkline Beecham Corp. | Antivirale pyrazolopyridin verbindungen |
ES2242028T3 (es) * | 2001-04-27 | 2005-11-01 | Smithkline Beecham Corporation | Derivados de pirazolo(1,5-a)piridina. |
CA2451008A1 (en) * | 2001-06-21 | 2003-01-03 | Smithkline Beecham Corporation | Imidazo[1,2-a!pyridine derivatives for the prophylaxis and treatment of herpes viral infections |
JP2005507878A (ja) * | 2001-09-07 | 2005-03-24 | スミスクライン ビーチャム コーポレーション | ヘルペス感染症を治療するためのピラゾロ−ピリジン類 |
EP1432712B1 (en) * | 2001-10-05 | 2006-05-17 | SmithKline Beecham Corporation | Imidazo-pyridine derivatives for use in the treatment of herpes viral infection |
EP1453830B1 (en) * | 2001-12-11 | 2007-09-12 | SmithKline Beecham Corporation | Pyrazolo-pyridine derivatives as antiherpes agents |
JP2006504728A (ja) * | 2002-10-03 | 2006-02-09 | スミスクライン ビーチャム コーポレーション | ピラソロピリジン誘導体系治療用化合物 |
US7459562B2 (en) | 2004-04-23 | 2008-12-02 | Bristol-Myers Squibb Company | Monocyclic heterocycles as kinase inhibitors |
TW200538453A (en) | 2004-04-26 | 2005-12-01 | Bristol Myers Squibb Co | Bicyclic heterocycles as kinase inhibitors |
US7439246B2 (en) | 2004-06-28 | 2008-10-21 | Bristol-Myers Squibb Company | Fused heterocyclic kinase inhibitors |
US7432373B2 (en) | 2004-06-28 | 2008-10-07 | Bristol-Meyers Squibb Company | Processes and intermediates useful for preparing fused heterocyclic kinase inhibitors |
US20050288290A1 (en) | 2004-06-28 | 2005-12-29 | Borzilleri Robert M | Fused heterocyclic kinase inhibitors |
WO2007035428A1 (en) | 2005-09-15 | 2007-03-29 | Bristol-Myers Squibb Company | Met kinase inhibitors |
US7547782B2 (en) | 2005-09-30 | 2009-06-16 | Bristol-Myers Squibb Company | Met kinase inhibitors |
US9073918B2 (en) | 2010-05-20 | 2015-07-07 | Takeda Pharmaceutical Company Limited | Pyrazolo[4,3-b]pyridine-7-amine inhibitors of ALK5 |
EP3181133B1 (en) | 2010-12-20 | 2019-07-24 | Pfizer Inc | Novel fused pyridine compounds as casein kinase inhibitors |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4115394A (en) * | 1974-05-06 | 1978-09-19 | E. R. Squibb & Sons, Inc. | Amino derivatives of 6-phenylpyrazolo[3,4-b]pyridines |
DE3464368D1 (de) * | 1983-03-09 | 1987-07-30 | Beecham Group Plc | Anti-inflammatory pyrazolo pyridines |
-
1985
- 1985-01-19 EP EP85100558A patent/EP0151962A3/en not_active Withdrawn
- 1985-01-23 AU AU38007/85A patent/AU3800785A/en not_active Abandoned
- 1985-01-23 GR GR850190A patent/GR850190B/el unknown
- 1985-01-23 US US06/693,731 patent/US4576952A/en not_active Expired - Fee Related
- 1985-01-24 ES ES539822A patent/ES8607298A1/es not_active Expired
Also Published As
Publication number | Publication date |
---|---|
US4576952A (en) | 1986-03-18 |
EP0151962A2 (en) | 1985-08-21 |
AU3800785A (en) | 1985-08-01 |
GR850190B (es) | 1985-05-23 |
ES8607298A1 (es) | 1986-05-16 |
EP0151962A3 (en) | 1985-10-02 |
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