AR226854A1 - Procedimiento para preparar derivados de acido trans-3-(4-oxo-4h-quinazolin-3-il)-2-propenoico - Google Patents
Procedimiento para preparar derivados de acido trans-3-(4-oxo-4h-quinazolin-3-il)-2-propenoicoInfo
- Publication number
- AR226854A1 AR226854A1 AR281693A AR28169380A AR226854A1 AR 226854 A1 AR226854 A1 AR 226854A1 AR 281693 A AR281693 A AR 281693A AR 28169380 A AR28169380 A AR 28169380A AR 226854 A1 AR226854 A1 AR 226854A1
- Authority
- AR
- Argentina
- Prior art keywords
- quinazolin
- oxo
- procedure
- acid derivatives
- propenoic acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
- C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5572879A | 1979-07-09 | 1979-07-09 | |
| US06/142,903 US4281127A (en) | 1979-07-09 | 1980-04-23 | Trans-3-(4-oxo-4H-quinazolin-3-yl)-2-propenoic acid derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR226854A1 true AR226854A1 (es) | 1982-08-31 |
Family
ID=26734565
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR281693A AR226854A1 (es) | 1979-07-09 | 1980-07-08 | Procedimiento para preparar derivados de acido trans-3-(4-oxo-4h-quinazolin-3-il)-2-propenoico |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US4281127A (enExample) |
| EP (1) | EP0023594B1 (enExample) |
| AR (1) | AR226854A1 (enExample) |
| AU (1) | AU521014B2 (enExample) |
| CA (1) | CA1134825A (enExample) |
| DE (1) | DE3067830D1 (enExample) |
| DK (1) | DK150483C (enExample) |
| ES (2) | ES8106302A1 (enExample) |
| FI (1) | FI74279C (enExample) |
| GR (1) | GR65952B (enExample) |
| HK (1) | HK52187A (enExample) |
| HU (1) | HU184797B (enExample) |
| IE (1) | IE49938B1 (enExample) |
| IL (1) | IL60514A (enExample) |
| MC (1) | MC1333A1 (enExample) |
| NO (1) | NO154426C (enExample) |
| NZ (1) | NZ194259A (enExample) |
| PH (1) | PH16413A (enExample) |
| PT (1) | PT71512B (enExample) |
| SG (1) | SG20887G (enExample) |
| YU (1) | YU42348B (enExample) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4599336A (en) * | 1983-08-08 | 1986-07-08 | Hoffmann-La Roche Inc. | Derivatives of (E)-3-(4-oxo-4H-quinazolin-3-yl)-2-propenamide |
| GB9404485D0 (en) * | 1994-03-09 | 1994-04-20 | Cancer Res Campaign Tech | Benzamide analogues |
| US6706721B1 (en) * | 1998-04-29 | 2004-03-16 | Osi Pharmaceuticals, Inc. | N-(3-ethynylphenylamino)-6,7-bis(2-methoxyethoxy)-4-quinazolinamine mesylate anhydrate and monohydrate |
| US7230000B1 (en) | 1999-10-27 | 2007-06-12 | Cytokinetics, Incorporated | Methods and compositions utilizing quinazolinones |
| US6545004B1 (en) | 1999-10-27 | 2003-04-08 | Cytokinetics, Inc. | Methods and compositions utilizing quinazolinones |
| US7087613B2 (en) * | 1999-11-11 | 2006-08-08 | Osi Pharmaceuticals, Inc. | Treating abnormal cell growth with a stable polymorph of N-(3-ethynylphenyl)-6,7-bis(2-methoxyethoxy)-4-quinazolinamine hydrochloride |
| UA74803C2 (uk) | 1999-11-11 | 2006-02-15 | Осі Фармасьютікалз, Інк. | Стійкий поліморф гідрохлориду n-(3-етинілфеніл)-6,7-біс(2-метоксіетокси)-4-хіназолінаміну, спосіб його одержання (варіанти) та фармацевтичне застосування |
| US7009049B2 (en) * | 2002-02-15 | 2006-03-07 | Cytokinetics, Inc. | Syntheses of quinazolinones |
| US7214800B2 (en) * | 2002-05-09 | 2007-05-08 | Cytokinetics, Inc. | Compounds, compositions, and methods |
| US7166595B2 (en) * | 2002-05-09 | 2007-01-23 | Cytokinetics, Inc. | Compounds, methods and compositions |
| US7038048B2 (en) * | 2002-05-23 | 2006-05-02 | Cytokinetics, Inc. | 3H-pyridopyrimidin-4-one compounds, compositions, and methods of their use |
| US7041676B2 (en) * | 2002-06-14 | 2006-05-09 | Cytokinetics, Inc. | Compounds, compositions, and methods |
| JP2006501201A (ja) * | 2002-07-23 | 2006-01-12 | サイトキネティクス・インコーポレーテッド | 化合物、組成物および方法 |
| EP1539180A4 (en) * | 2002-08-21 | 2006-08-30 | Cytokinetics Inc | COMPOUNDS, COMPOSITIONS AND METHODS |
| EP1558083A4 (en) * | 2002-09-30 | 2008-04-16 | Cytokinetics Inc | COMPOUNDS, COMPOSITIONS AND METHODS |
| EP1682534A2 (en) * | 2003-11-03 | 2006-07-26 | Cytokinetics, Inc. | Pyrimidin-4-one compounds, compositions, and methods |
| EP1680420A4 (en) * | 2003-11-07 | 2008-09-24 | Cytokinetics Inc | COMPOUNDS, COMPOSITIONS AND METHODS |
| EP1692112A4 (en) * | 2003-12-08 | 2008-09-24 | Cytokinetics Inc | COMPOUNDS, COMPOSITIONS, AND METHODS |
| UY29198A1 (es) * | 2004-11-09 | 2006-05-31 | Cancer Rec Tech Ltd | Derivados sustituidos de quinazolinona y derivados sustituidos de quinazolina-2, 4-diona, composiciones conteniéndolos, procedimientos de preparación y aplicaciones |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2786055A (en) * | 1955-02-10 | 1957-03-19 | Mallinckrodt Chemical Works | Carboxyalkyl-iodoquinazolones |
| US3517005A (en) * | 1967-10-26 | 1970-06-23 | Pfizer & Co C | Certain 2- and 4-substituted quinazolines |
| US3696102A (en) * | 1970-03-09 | 1972-10-03 | Pfizer & Co C | Process for the synthesis of substituted quinazolin-4-ones |
-
1980
- 1980-04-23 US US06/142,903 patent/US4281127A/en not_active Expired - Lifetime
- 1980-07-07 MC MC801458A patent/MC1333A1/fr unknown
- 1980-07-07 NZ NZ194259A patent/NZ194259A/en unknown
- 1980-07-07 CA CA000355555A patent/CA1134825A/en not_active Expired
- 1980-07-07 IL IL60514A patent/IL60514A/xx unknown
- 1980-07-07 HU HU801690A patent/HU184797B/hu not_active IP Right Cessation
- 1980-07-07 GR GR62402A patent/GR65952B/el unknown
- 1980-07-08 PT PT71512A patent/PT71512B/pt unknown
- 1980-07-08 DK DK294780A patent/DK150483C/da active
- 1980-07-08 DE DE8080103896T patent/DE3067830D1/de not_active Expired
- 1980-07-08 ES ES493203A patent/ES8106302A1/es not_active Expired
- 1980-07-08 NO NO802056A patent/NO154426C/no unknown
- 1980-07-08 AR AR281693A patent/AR226854A1/es active
- 1980-07-08 EP EP80103896A patent/EP0023594B1/de not_active Expired
- 1980-07-08 IE IE1412/80A patent/IE49938B1/en not_active IP Right Cessation
- 1980-07-09 FI FI802195A patent/FI74279C/fi not_active IP Right Cessation
- 1980-07-09 PH PH24261A patent/PH16413A/en unknown
- 1980-07-09 AU AU60244/80A patent/AU521014B2/en not_active Ceased
- 1980-07-09 YU YU1766/80A patent/YU42348B/xx unknown
-
1981
- 1981-02-02 ES ES499035A patent/ES8207155A1/es not_active Expired
-
1987
- 1987-02-26 SG SG208/87A patent/SG20887G/en unknown
- 1987-07-09 HK HK521/87A patent/HK52187A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DK294780A (da) | 1981-01-10 |
| IE49938B1 (en) | 1986-01-08 |
| ES499035A0 (es) | 1982-09-16 |
| MC1333A1 (fr) | 1981-04-21 |
| YU42348B (en) | 1988-08-31 |
| IL60514A0 (en) | 1980-09-16 |
| US4281127A (en) | 1981-07-28 |
| FI74279B (fi) | 1987-09-30 |
| SG20887G (en) | 1988-09-16 |
| ES493203A0 (es) | 1981-05-16 |
| NZ194259A (en) | 1984-09-28 |
| EP0023594A1 (de) | 1981-02-11 |
| AU6024480A (en) | 1981-03-12 |
| AU521014B2 (en) | 1982-03-11 |
| DE3067830D1 (en) | 1984-06-20 |
| IL60514A (en) | 1985-03-31 |
| ES8106302A1 (es) | 1981-05-16 |
| GR65952B (enExample) | 1981-01-09 |
| PT71512B (en) | 1981-12-11 |
| YU176680A (en) | 1984-12-31 |
| PH16413A (en) | 1983-09-29 |
| CA1134825A (en) | 1982-11-02 |
| EP0023594B1 (de) | 1984-05-16 |
| DK150483B (da) | 1987-03-09 |
| FI74279C (fi) | 1988-01-11 |
| HU184797B (en) | 1984-10-29 |
| NO154426C (no) | 1986-09-17 |
| PT71512A (en) | 1980-08-01 |
| NO802056L (no) | 1981-01-12 |
| IE801412L (en) | 1981-01-09 |
| FI802195A7 (fi) | 1981-01-10 |
| HK52187A (en) | 1987-07-17 |
| DK150483C (da) | 1987-11-09 |
| NO154426B (no) | 1986-06-09 |
| ES8207155A1 (es) | 1982-09-16 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES494352A0 (es) | Procedimiento para preparar derivados de acidos quinolina- carboxilicos | |
| MX6094E (es) | Procedimiento para preparar derivados del acido 6 beta-hidroxialquil penicilanico | |
| AR226854A1 (es) | Procedimiento para preparar derivados de acido trans-3-(4-oxo-4h-quinazolin-3-il)-2-propenoico | |
| AR213000A1 (es) | Procedimiento para preparacion de acido di-n-propil-acetico | |
| ES505207A0 (es) | Procedimiento para preparar derivados de acido quinolina- carboxilico | |
| AR227525A1 (es) | Procedimiento para obtener derivados de acidos ciclohexancarboxilicos | |
| ES488651A0 (es) | Procedimiento para preparar derivados de acido acetico | |
| AR222304A1 (es) | Procedimiento para preparar acido 4-isohexil-1-metilciclohexano-carboxilico | |
| AR229152A1 (es) | Procedimiento para obtener derivados de acidos de 1-tioalcanoilprolina | |
| ES490729A0 (es) | Procedimiento para la preparacion de nuevas imidas de acido ciclobutandicarboxilico | |
| ES492693A0 (es) | Procedimiento para preparar derivados de acido acilaminoben-zoico | |
| ES489924A0 (es) | Un procedimiento para preparar derivados de acido imidazol- dicarboxilico | |
| AR225292A1 (es) | Procedimiento para preparar derivados de acido 6-halogeno-alfametil carbazol-2-acetico | |
| MX5224E (es) | Procedimiento para preparar anilidas de acido ciclopropanocarboxilico | |
| ES503834A0 (es) | Procedimiento para preparar derivados de acido 2-cloro-4- trifluoromtil-5-tiazolcarbotioico | |
| ES491601A0 (es) | Procedimiento para la preparacion de derivados de acido n-acil-amino | |
| AR218294A1 (es) | Procedimiento para la preparacion de derivados de acido oleanoico | |
| MX5206E (es) | Procedimiento para la preparacion de fenoxi-alfa-vinil-bencil-esteres de acido ciclopropancarboxilico | |
| MX5929E (es) | Procedimiento para preparar derivados de acido 2-(3-aril-5-isoxazolil)-benzoico | |
| AR223902A1 (es) | Procedimiento para preparar cloruro de acido gamma-cloroacetoacetico | |
| ES497506A0 (es) | Procedimiento para la obtencion de hidrazida de acido al- quildifenileter-sulfonico | |
| AR225776A1 (es) | Un procedimiento para la preparacion de acido 9-oxo-11 alfa-hidroxi-15-metanosulfonamido-16-genoxi-cis-5 w-omega-tetranor prostenoico | |
| ES489119A0 (es) | Un procedimiento para la preparacion de acido 6-cloro-alfa- metil-carbazol-2-acetico | |
| ES489318A0 (es) | Procedimiento para la obtencion de compuestos de acido 17-c-esteroide- -propionico | |
| ES497849A0 (es) | Procedimiento para la obtencion de compuestos de acido aci- lamino-3-cefem-4-carboxilico |