AR221721A1 - PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4, A 5,9B-HEXAHIDRO-1H-PIRIDOL (4,3-B) -INDOL, INTERMEDIARIES USED THEREOF AND PROCEDURE FOR PREPARING SUCH INTERMEDIARIES - Google Patents

PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4, A 5,9B-HEXAHIDRO-1H-PIRIDOL (4,3-B) -INDOL, INTERMEDIARIES USED THEREOF AND PROCEDURE FOR PREPARING SUCH INTERMEDIARIES

Info

Publication number
AR221721A1
AR221721A1 AR276191A AR27619179A AR221721A1 AR 221721 A1 AR221721 A1 AR 221721A1 AR 276191 A AR276191 A AR 276191A AR 27619179 A AR27619179 A AR 27619179A AR 221721 A1 AR221721 A1 AR 221721A1
Authority
AR
Argentina
Prior art keywords
procedure
intermediaries
piridol
hexahidro
indol
Prior art date
Application number
AR276191A
Other languages
Spanish (es)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of AR221721A1 publication Critical patent/AR221721A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AR276191A 1977-05-23 1979-04-16 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4, A 5,9B-HEXAHIDRO-1H-PIRIDOL (4,3-B) -INDOL, INTERMEDIARIES USED THEREOF AND PROCEDURE FOR PREPARING SUCH INTERMEDIARIES AR221721A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US79939277A 1977-05-23 1977-05-23

Publications (1)

Publication Number Publication Date
AR221721A1 true AR221721A1 (en) 1981-03-13

Family

ID=25175793

Family Applications (2)

Application Number Title Priority Date Filing Date
AR271956A AR217688A1 (en) 1977-05-23 1978-04-28 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4A, 5,9B-HEXAHIDRO-1H-PIRIDO (4,3-B) -INDOL
AR276191A AR221721A1 (en) 1977-05-23 1979-04-16 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4, A 5,9B-HEXAHIDRO-1H-PIRIDOL (4,3-B) -INDOL, INTERMEDIARIES USED THEREOF AND PROCEDURE FOR PREPARING SUCH INTERMEDIARIES

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR271956A AR217688A1 (en) 1977-05-23 1978-04-28 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4A, 5,9B-HEXAHIDRO-1H-PIRIDO (4,3-B) -INDOL

Country Status (31)

Country Link
JP (1) JPS53144600A (en)
AR (2) AR217688A1 (en)
AT (1) AT368995B (en)
AU (1) AU499618B1 (en)
BE (1) BE867249A (en)
CA (1) CA1094071A (en)
CH (1) CH634321A5 (en)
CS (1) CS207612B2 (en)
DD (4) DD138321A5 (en)
DE (1) DE2822465C2 (en)
DK (1) DK226678A (en)
EG (1) EG13590A (en)
FI (1) FI63402C (en)
FR (1) FR2392023A1 (en)
GB (1) GB1586655A (en)
GR (1) GR69985B (en)
HU (3) HU188802B (en)
IE (1) IE46975B1 (en)
IL (1) IL54755A (en)
IT (1) IT1096307B (en)
LU (1) LU79684A1 (en)
NL (1) NL7804210A (en)
NO (2) NO150204C (en)
NZ (1) NZ187333A (en)
PH (1) PH13756A (en)
PL (5) PL114541B1 (en)
PT (1) PT68058B (en)
SE (2) SE441448B (en)
SU (4) SU873883A3 (en)
YU (4) YU91478A (en)
ZA (1) ZA782918B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4224329A (en) * 1979-01-23 1980-09-23 Pfizer Inc. 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4451655A (en) * 1982-05-17 1984-05-29 Pfizer Inc. Process for preparing carboline derivatives and compounds used in their preparation
RU2106864C1 (en) * 1995-10-23 1998-03-20 Николай Серафимович Зефиров New approach to treatment of alzheimer's disease
US6974825B1 (en) 1996-12-20 2005-12-13 Astrazeneca Canada Inc. Compounds with analgesic effect
SE9604786D0 (en) 1996-12-20 1996-12-20 Astra Pharma Inc New compounds
SE9904675D0 (en) 1999-12-20 1999-12-20 Astra Pharma Inc Novel compounds
SE0101771D0 (en) 2001-05-18 2001-05-18 Astrazeneca Ab Novel compounds
SE0101773D0 (en) 2001-05-18 2001-05-18 Astrazeneca Ab Novel compounds
SE0101769D0 (en) 2001-05-18 2001-05-18 Astrazeneca Ab Novel compounds
SE0101770D0 (en) 2001-05-18 2001-05-18 Astrazeneca Ab Novel compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR205452A1 (en) * 1973-12-06 1976-05-07 Endo Lab METHOD TO PREPARE NEW TRANS-2, 3, 4, 4A, 5, 9B-HEXAHYDRO-5-PHENYL-1H-PYRID (4,3-B) INDOLES
JPS50126699A (en) * 1974-03-20 1975-10-04
US4001263A (en) * 1974-04-01 1977-01-04 Pfizer Inc. 5-Aryl-1,2,3,4-tetrahydro-γ-carbolines

Also Published As

Publication number Publication date
SU818484A3 (en) 1981-03-30
IL54755A (en) 1981-02-27
YU221882A (en) 1983-01-21
PL206903A1 (en) 1979-10-22
SE7803625L (en) 1978-11-24
DE2822465C2 (en) 1986-08-28
FI63402B (en) 1983-02-28
JPS53144600A (en) 1978-12-15
GB1586655A (en) 1981-03-25
GR69985B (en) 1982-07-22
ATA369678A (en) 1982-04-15
SE441448B (en) 1985-10-07
NO151862C (en) 1985-06-19
IE781013L (en) 1978-11-23
NO831790L (en) 1978-11-24
NO781770L (en) 1978-11-24
FR2392023A1 (en) 1978-12-22
JPS5711912B2 (en) 1982-03-08
CA1094071A (en) 1981-01-20
DD145536A5 (en) 1980-12-17
HU188802B (en) 1986-05-28
PL117107B1 (en) 1981-07-31
PT68058A (en) 1978-06-01
CS207612B2 (en) 1981-08-31
SU841589A3 (en) 1981-06-23
AU499618B1 (en) 1979-04-26
PH13756A (en) 1980-09-17
PT68058B (en) 1979-10-24
HU187782B (en) 1986-02-28
IL54755A0 (en) 1978-07-31
IT7823673A0 (en) 1978-05-22
HU185009B (en) 1984-11-28
LU79684A1 (en) 1979-12-06
AT368995B (en) 1982-11-25
DD145537A5 (en) 1980-12-17
PL114547B1 (en) 1981-02-28
PL116944B1 (en) 1981-07-31
DE2822465A1 (en) 1978-11-30
DK226678A (en) 1978-11-24
NO150204C (en) 1984-09-05
YU221782A (en) 1983-01-21
DD146186A5 (en) 1981-01-28
DD138321A5 (en) 1979-10-24
NO150204B (en) 1984-05-28
CH634321A5 (en) 1983-01-31
NO151862B (en) 1985-03-11
FR2392023B1 (en) 1980-11-07
FI781612A (en) 1978-11-24
YU221682A (en) 1983-01-21
NZ187333A (en) 1984-05-31
SE8305917D0 (en) 1983-10-27
SE8305917L (en) 1983-10-27
IE46975B1 (en) 1983-11-16
EG13590A (en) 1982-03-31
SE448459B (en) 1987-02-23
AR217688A1 (en) 1980-04-15
SU873883A3 (en) 1981-10-15
BE867249A (en) 1978-11-20
FI63402C (en) 1983-06-10
IT1096307B (en) 1985-08-26
YU91478A (en) 1983-01-21
NL7804210A (en) 1978-11-27
ZA782918B (en) 1979-06-27
YU40796B (en) 1986-06-30
PL114541B1 (en) 1981-02-28
SU843749A3 (en) 1981-06-30

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