AR109930A1 - Proceso para la preparación de ácidos (1r,3r)- y (1s,3s)-2,2-dihalo-3-ciclopropanocarboxílicos (con fenilo sustituido) - Google Patents
Proceso para la preparación de ácidos (1r,3r)- y (1s,3s)-2,2-dihalo-3-ciclopropanocarboxílicos (con fenilo sustituido)Info
- Publication number
- AR109930A1 AR109930A1 ARP170102842A ARP170102842A AR109930A1 AR 109930 A1 AR109930 A1 AR 109930A1 AR P170102842 A ARP170102842 A AR P170102842A AR P170102842 A ARP170102842 A AR P170102842A AR 109930 A1 AR109930 A1 AR 109930A1
- Authority
- AR
- Argentina
- Prior art keywords
- cyclopropanocarboxílicos
- phenyll
- dihalo
- acids
- replaced
- Prior art date
Links
- 239000002253 acid Substances 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 2
- 150000007513 acids Chemical class 0.000 title 1
- GVGFEJPTKINGLP-UHFFFAOYSA-N 2,2-dichlorocyclopropane-1-carboxylic acid Chemical compound OC(=O)C1CC1(Cl)Cl GVGFEJPTKINGLP-UHFFFAOYSA-N 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- -1 amine salt Chemical class 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 238000002955 isolation Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/42—Separation; Purification; Stabilisation; Use of additives
- C07C51/487—Separation; Purification; Stabilisation; Use of additives by treatment giving rise to chemical modification
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/42—Separation; Purification; Stabilisation; Use of additives
- C07C51/50—Use of additives, e.g. for stabilisation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C61/00—Compounds having carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings
- C07C61/16—Unsaturated compounds
- C07C61/40—Unsaturated compounds containing halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
El enantiómero (1R,3R) o (1S,3S) del ácido 2,2-dicloro-3-ciclopropano-carboxílico (con fenilo sustituido) se prepara en un proceso que implica la resolución química de una mezcla racémica de un ácido trans-2,2-dicloro-3-ciclopropanocarboxílico (con fenilo sustituido) con una amina enantiomérica, el aislamiento de una sal de amina diaestereomérica y el tratamiento final de la sal con un ácido.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662406972P | 2016-10-12 | 2016-10-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR109930A1 true AR109930A1 (es) | 2019-02-06 |
Family
ID=60153549
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP170102842A AR109930A1 (es) | 2016-10-12 | 2017-10-11 | Proceso para la preparación de ácidos (1r,3r)- y (1s,3s)-2,2-dihalo-3-ciclopropanocarboxílicos (con fenilo sustituido) |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US10239817B2 (es) |
| EP (1) | EP3526189B1 (es) |
| JP (1) | JP7059265B2 (es) |
| KR (1) | KR102479201B1 (es) |
| CN (1) | CN109863131B (es) |
| AR (1) | AR109930A1 (es) |
| CA (1) | CA3037554C (es) |
| CO (1) | CO2019003644A2 (es) |
| ES (1) | ES2834110T3 (es) |
| IL (1) | IL265990B (es) |
| MX (1) | MX2019004253A (es) |
| TW (1) | TWI758313B (es) |
| WO (1) | WO2018071320A1 (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3578542A1 (en) | 2015-04-17 | 2019-12-11 | Dow AgroSciences LLC | Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto |
| US10258045B2 (en) | 2016-10-12 | 2019-04-16 | Dow Agrosciences Llc | Molecules having pesticidal utility and intermediates, compositions and processes related thereto |
| TWI758313B (zh) | 2016-10-12 | 2022-03-21 | 美商陶氏農業科學公司 | 一種用於製備(1r,3r)-及(1s,3s)-2,2-二鹵基-3-(經取代之苯基)環丙烷甲酸的方法 |
| US20230220427A1 (en) | 2020-04-24 | 2023-07-13 | Corteva Agriscience Llc | Processes related to formation of arylcyclopropyl carboxylic acids |
| CN117098750A (zh) | 2021-03-23 | 2023-11-21 | 科迪华农业科技有限责任公司 | 具有杀有害生物效用的分子以及与其相关的中间体和方法 |
| JP2024518272A (ja) | 2021-05-07 | 2024-05-01 | コルテバ アグリサイエンス エルエルシー | ハロシクロプロパン化プロセス |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU205594B (en) * | 1989-01-16 | 1992-05-28 | Chinoin Gyogyszer Es Vegyeszet | Process for producing optical isomeres of cyclopropane-carboxylic acids5 |
| JP3209041B2 (ja) * | 1994-06-15 | 2001-09-17 | 東レ株式会社 | 光学分割剤およびそれを用いた光学活性テトラヒドロフランカルボン酸類の製造法 |
| JP3484510B2 (ja) * | 1995-11-24 | 2004-01-06 | 東レ株式会社 | 光学活性カルボン酸の製造法 |
| FR2765577A1 (fr) | 1997-07-02 | 1999-01-08 | Hoechst Schering Agrevo Sa | Nouveaux amides aromatiques, leur procede de preparation et leur application comme pesticides |
| EP1489066B1 (en) * | 2002-03-06 | 2010-08-04 | Ajinomoto Co., Inc. | Process for production of optically active carboxylic acid |
| MXPA05002874A (es) * | 2002-09-20 | 2005-05-27 | Wyeth Corp | Procedimiento para la sintesis de intermediarios utiles para la sintesis de inhibidores de tubulina. |
| JP4356060B2 (ja) * | 2002-12-05 | 2009-11-04 | 東レ・ファインケミカル株式会社 | 光学活性１−保護インドリン−２−カルボン酸誘導体の製造方法および光学活性インドリン−２−カルボン酸誘導体の製造方法 |
| CN1262535C (zh) * | 2004-04-12 | 2006-07-05 | 浙江大学 | S－(+)－2,2－二甲基环丙烷甲酰胺的合成方法 |
| US7754717B2 (en) | 2005-08-15 | 2010-07-13 | Amgen Inc. | Bis-aryl amide compounds and methods of use |
| CA2662031A1 (en) | 2006-09-06 | 2008-03-13 | F. Hoffmann-La Roche Ag | Heteroaryl derivatives as protein kinase inhibitors |
| US9029107B2 (en) * | 2010-08-31 | 2015-05-12 | Api Corporation | Hydrolase protein |
| US20140142337A1 (en) * | 2011-06-21 | 2014-05-22 | Mitsubishi Gas Chemical Company, Inc. | 1-amino-2-vinylcyclopropane carboxylic acid amide and salt thereof, and method for producing same |
| EP2628721A1 (en) * | 2012-02-20 | 2013-08-21 | LEK Pharmaceuticals d.d. | Synthesis of 2-(3,4-difluorophenyl)cyclopropanecarboxylic acid |
| JP6342422B2 (ja) | 2012-12-19 | 2018-06-13 | ダウ アグロサイエンシィズ エルエルシー | 農薬組成物およびそれらに関する方法 |
| EP3578542A1 (en) | 2015-04-17 | 2019-12-11 | Dow AgroSciences LLC | Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto |
| TWI758313B (zh) | 2016-10-12 | 2022-03-21 | 美商陶氏農業科學公司 | 一種用於製備(1r,3r)-及(1s,3s)-2,2-二鹵基-3-(經取代之苯基)環丙烷甲酸的方法 |
| US10258045B2 (en) | 2016-10-12 | 2019-04-16 | Dow Agrosciences Llc | Molecules having pesticidal utility and intermediates, compositions and processes related thereto |
-
2017
- 2017-08-23 TW TW106128545A patent/TWI758313B/zh active
- 2017-10-09 WO PCT/US2017/055699 patent/WO2018071320A1/en active Application Filing
- 2017-10-09 CA CA3037554A patent/CA3037554C/en active Active
- 2017-10-09 US US15/727,651 patent/US10239817B2/en active Active
- 2017-10-09 JP JP2019519378A patent/JP7059265B2/ja active Active
- 2017-10-09 CN CN201780062351.7A patent/CN109863131B/zh active Active
- 2017-10-09 EP EP17787817.0A patent/EP3526189B1/en active Active
- 2017-10-09 MX MX2019004253A patent/MX2019004253A/es unknown
- 2017-10-09 ES ES17787817T patent/ES2834110T3/es active Active
- 2017-10-09 KR KR1020197010121A patent/KR102479201B1/ko active IP Right Grant
- 2017-10-11 AR ARP170102842A patent/AR109930A1/es active IP Right Grant
-
2019
- 2019-04-11 IL IL265990A patent/IL265990B/en active IP Right Grant
- 2019-04-12 CO CONC2019/0003644A patent/CO2019003644A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN109863131A (zh) | 2019-06-07 |
| CA3037554C (en) | 2024-05-21 |
| MX2019004253A (es) | 2019-07-01 |
| WO2018071320A1 (en) | 2018-04-19 |
| JP2019530709A (ja) | 2019-10-24 |
| NZ751476A (en) | 2021-09-24 |
| CN109863131B (zh) | 2022-04-05 |
| EP3526189A1 (en) | 2019-08-21 |
| JP7059265B2 (ja) | 2022-04-25 |
| KR20190059291A (ko) | 2019-05-30 |
| US20180099919A1 (en) | 2018-04-12 |
| IL265990B (en) | 2021-04-29 |
| TWI758313B (zh) | 2022-03-21 |
| KR102479201B1 (ko) | 2022-12-20 |
| TW201813951A (zh) | 2018-04-16 |
| ES2834110T3 (es) | 2021-06-16 |
| IL265990A (en) | 2019-06-30 |
| CA3037554A1 (en) | 2018-04-19 |
| EP3526189B1 (en) | 2020-09-09 |
| CO2019003644A2 (es) | 2019-04-30 |
| US10239817B2 (en) | 2019-03-26 |
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