AR029981A1 - Utilizacion de dihidropiridinas condensadas para la preparacion de agentes destinados al tratamiento de dolores cronicos - Google Patents
Utilizacion de dihidropiridinas condensadas para la preparacion de agentes destinados al tratamiento de dolores cronicosInfo
- Publication number
- AR029981A1 AR029981A1 ARP010103543A ARP010103543A AR029981A1 AR 029981 A1 AR029981 A1 AR 029981A1 AR P010103543 A ARP010103543 A AR P010103543A AR P010103543 A ARP010103543 A AR P010103543A AR 029981 A1 AR029981 A1 AR 029981A1
- Authority
- AR
- Argentina
- Prior art keywords
- condensed
- preparation
- treatment
- chronic pain
- dihydropiridines
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Suspension/Interruption
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4747—Quinolines; Isoquinolines spiro-condensed
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/12—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
- C07D217/14—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
- C07D217/16—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals substituted by oxygen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
El presente se refiere a la utilizacion de dihidropiridinas condensadas y sus sales con ácidos fisiologicamente compatibles para la preparacion de agentes destinados al tratamiento de dolores cronicos, de la formula general (1), en la que A es benzo o tieno; y Z, R1, R2, R3, R4, R5 y R6 son como se han definido en la memoria descriptiva, así como nuevos compuestos de la formula (1).
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10035997A DE10035997A1 (de) | 2000-07-25 | 2000-07-25 | Verwendung von anellierten Dihydropyridinen zur Herstellung von Mitteln für die Behandlung von chronischen Schmerzen |
Publications (1)
Publication Number | Publication Date |
---|---|
AR029981A1 true AR029981A1 (es) | 2003-07-23 |
Family
ID=7650021
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP010103543A Suspension/Interruption AR029981A1 (es) | 2000-07-25 | 2001-07-25 | Utilizacion de dihidropiridinas condensadas para la preparacion de agentes destinados al tratamiento de dolores cronicos |
Country Status (5)
Country | Link |
---|---|
AR (1) | AR029981A1 (es) |
AU (1) | AU2001289719A1 (es) |
DE (1) | DE10035997A1 (es) |
UY (1) | UY26852A1 (es) |
WO (1) | WO2002007714A2 (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2003014089A1 (en) * | 2001-07-31 | 2003-02-20 | Virginia Commonwealth University | Aminotetrahydroisoquinoline derivatives as analgesics |
RU2711646C1 (ru) * | 2019-04-08 | 2020-01-17 | Федеральное государственное бюджетное учреждение науки Институт молекулярной генетики Российской академии наук | Синтез меченного тритием 6,7-диметокси-4,4-диметил-1-[4-(4-трифторметилфенокси)фенил]-3Н-изохинолина |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1386076A (en) * | 1971-06-03 | 1975-03-05 | Wyeth John & Brother Ltd | Isoquinoline derivatives |
CA1330560C (en) * | 1986-05-21 | 1994-07-05 | Maurits E. A. Vandewalle | Di- and tetrahydroisoquinoline derivatives |
GB8921304D0 (en) * | 1989-09-20 | 1989-11-08 | Wyeth John & Brother Ltd | New method of treatment and heterocyclic compounds used therein |
EP0491441A1 (en) * | 1990-12-17 | 1992-06-24 | Shell Internationale Researchmaatschappij B.V. | Fungicidal isoquinoline derivatives |
WO2000044725A1 (de) * | 1999-01-28 | 2000-08-03 | Boehringer Ingelheim Pharma Kg | Anellierte dihydropyridine und verwendung von anellierten dihydropyridinen für die herstellung von mitteln für die behandlung von epilepsie |
-
2000
- 2000-07-25 DE DE10035997A patent/DE10035997A1/de not_active Withdrawn
-
2001
- 2001-07-21 AU AU2001289719A patent/AU2001289719A1/en not_active Abandoned
- 2001-07-21 WO PCT/EP2001/008453 patent/WO2002007714A2/en active Application Filing
- 2001-07-25 UY UY26852A patent/UY26852A1/es not_active Application Discontinuation
- 2001-07-25 AR ARP010103543A patent/AR029981A1/es not_active Suspension/Interruption
Also Published As
Publication number | Publication date |
---|---|
DE10035997A1 (de) | 2002-02-07 |
WO2002007714A2 (en) | 2002-01-31 |
AU2001289719A1 (en) | 2002-02-05 |
WO2002007714A3 (en) | 2002-09-06 |
UY26852A1 (es) | 2002-02-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |