AR027377A1 - Proceso para la simple preparacion de (3-cloro-4-fluorofenilo)-[7-(3-morfolina-4-ilo-propoxi)-6-nitroquinazolina-4-ilo]-mina o (3-cloro-4-fluorofenilo)-[7-(3-morfolina-4-il-propoxi)-6-aminoquinazolina-4-ilo]-amina. - Google Patents

Proceso para la simple preparacion de (3-cloro-4-fluorofenilo)-[7-(3-morfolina-4-ilo-propoxi)-6-nitroquinazolina-4-ilo]-mina o (3-cloro-4-fluorofenilo)-[7-(3-morfolina-4-il-propoxi)-6-aminoquinazolina-4-ilo]-amina.

Info

Publication number
AR027377A1
AR027377A1 ARP010100547A ARP010100547A AR027377A1 AR 027377 A1 AR027377 A1 AR 027377A1 AR P010100547 A ARP010100547 A AR P010100547A AR P010100547 A ARP010100547 A AR P010100547A AR 027377 A1 AR027377 A1 AR 027377A1
Authority
AR
Argentina
Prior art keywords
ilo
chloro
morfolina
propoxi
nitroquinazolina
Prior art date
Application number
ARP010100547A
Other languages
English (en)
Original Assignee
Godecke Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Godecke Gmbh filed Critical Godecke Gmbh
Publication of AR027377A1 publication Critical patent/AR027377A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Se refiere a una reaccion global para la preparacion de (3-cloro-4-fluorofenilo)-[7-(3-morfolina-4-ilo-propoxi)-6-nitroquinazolina-4-ilo]-amina (1) o de(3-cloro-4-fluorofenilo)-[7-(3-morfolina-4-ilo-propoxi)6-aminoquinazolina-4-ilo]amina (2).
ARP010100547A 2000-02-26 2001-02-07 Proceso para la simple preparacion de (3-cloro-4-fluorofenilo)-[7-(3-morfolina-4-ilo-propoxi)-6-nitroquinazolina-4-ilo]-mina o (3-cloro-4-fluorofenilo)-[7-(3-morfolina-4-il-propoxi)-6-aminoquinazolina-4-ilo]-amina. AR027377A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10009267A DE10009267A1 (de) 2000-02-26 2000-02-26 Verfahren zur einfachen Herstellung von (3-Chlor-4-fluor-phenyl)-[7-(3-morpholin-4-yl-propoxy)-6-nitro-quinazolin-4-yl]-amin bzw. (3-Chlor-4-fluor-phenyl)-[7-(3-morpholin-4-yl-propoxy)-6-amino-quinazolin-4-yl]-amin

Publications (1)

Publication Number Publication Date
AR027377A1 true AR027377A1 (es) 2003-03-26

Family

ID=7632648

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP010100547A AR027377A1 (es) 2000-02-26 2001-02-07 Proceso para la simple preparacion de (3-cloro-4-fluorofenilo)-[7-(3-morfolina-4-ilo-propoxi)-6-nitroquinazolina-4-ilo]-mina o (3-cloro-4-fluorofenilo)-[7-(3-morfolina-4-il-propoxi)-6-aminoquinazolina-4-ilo]-amina.

Country Status (31)

Country Link
US (1) US20030050313A1 (es)
EP (1) EP1265874B1 (es)
JP (1) JP2003524006A (es)
KR (1) KR20030011773A (es)
CN (1) CN1171877C (es)
AR (1) AR027377A1 (es)
AT (1) ATE296810T1 (es)
AU (1) AU2001228478A1 (es)
BR (1) BR0108695A (es)
CA (1) CA2401171A1 (es)
CO (1) CO5280058A1 (es)
DE (2) DE10009267A1 (es)
EA (1) EA005213B1 (es)
EG (1) EG23221A (es)
ES (1) ES2240483T3 (es)
GT (1) GT200100025A (es)
HK (1) HK1054551B (es)
HU (1) HUP0204510A3 (es)
IL (1) IL151206A0 (es)
MX (1) MXPA02008301A (es)
MY (1) MY133846A (es)
PA (1) PA8512701A1 (es)
PE (1) PE20011073A1 (es)
PL (1) PL357774A1 (es)
PT (1) PT1265874E (es)
SV (1) SV2002000320A (es)
TN (1) TNSN01031A1 (es)
UY (1) UY26594A1 (es)
WO (1) WO2001062743A2 (es)
YU (1) YU62502A (es)
ZA (1) ZA200206107B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20040945A1 (es) * 2003-02-05 2004-12-14 Warner Lambert Co Preparacion de quinazolinas substituidas
WO2006081741A1 (fr) * 2005-02-05 2006-08-10 Piaoyang Sun Dérivés de quinazoline ou leurs sels de qualité pharmaceutique, synthèse et applications médicales desdites substances
JP5250901B2 (ja) * 2007-02-23 2013-07-31 学校法人慶應義塾 アニリノキナゾリン系化合物及びその用途
US7829574B2 (en) * 2008-05-09 2010-11-09 Hutchison Medipharma Enterprises Limited Substituted quinazoline compounds and their use in treating angiogenesis-related diseases
CN105399688A (zh) * 2015-12-02 2016-03-16 西南科技大学 一种吉非替尼的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0892789T4 (da) * 1996-04-12 2010-04-06 Warner Lambert Co Irreversible inhibitorer af tyrosin kinaser

Also Published As

Publication number Publication date
HK1054551B (zh) 2005-06-03
WO2001062743A2 (de) 2001-08-30
ZA200206107B (en) 2003-07-31
CA2401171A1 (en) 2001-08-30
HUP0204510A3 (en) 2003-07-28
YU62502A (sh) 2005-03-15
DE10009267A1 (de) 2001-08-30
PE20011073A1 (es) 2001-12-16
AU2001228478A1 (en) 2001-09-03
HUP0204510A2 (en) 2003-05-28
WO2001062743A3 (de) 2002-03-14
GT200100025A (es) 2003-09-22
PA8512701A1 (es) 2002-02-21
KR20030011773A (ko) 2003-02-11
EA200200885A1 (ru) 2003-02-27
JP2003524006A (ja) 2003-08-12
PL357774A1 (en) 2004-07-26
CN1171877C (zh) 2004-10-20
EA005213B1 (ru) 2004-12-30
HK1054551A1 (en) 2003-12-05
ATE296810T1 (de) 2005-06-15
PT1265874E (pt) 2005-08-31
CO5280058A1 (es) 2003-05-30
ES2240483T3 (es) 2005-10-16
TNSN01031A1 (en) 2005-11-10
MY133846A (en) 2007-11-30
US20030050313A1 (en) 2003-03-13
EP1265874B1 (de) 2005-06-01
EP1265874A2 (de) 2002-12-18
BR0108695A (pt) 2002-12-10
CN1406232A (zh) 2003-03-26
IL151206A0 (en) 2003-04-10
SV2002000320A (es) 2002-06-07
DE50106391D1 (de) 2005-07-07
MXPA02008301A (es) 2004-05-14
EG23221A (en) 2004-08-31
UY26594A1 (es) 2001-09-28

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