IL151206A0 - Process for the simple preparation of (3-chloro-4-fluorophenyl)-7-(3-morpholin-4-yl-propoxy)-6-nitroquinazolin-4-yl]-amine or (3-chloro-4-yl-propoxy)-6-nitroquinazolin-4-yl]-amine or (3-chloro-4-fluorophenyl)-[7(3-morpholin-4-yl-propoxy)-6-aminoquinazolin-4-yl]-amine - Google Patents

Process for the simple preparation of (3-chloro-4-fluorophenyl)-7-(3-morpholin-4-yl-propoxy)-6-nitroquinazolin-4-yl]-amine or (3-chloro-4-yl-propoxy)-6-nitroquinazolin-4-yl]-amine or (3-chloro-4-fluorophenyl)-[7(3-morpholin-4-yl-propoxy)-6-aminoquinazolin-4-yl]-amine

Info

Publication number
IL151206A0
IL151206A0 IL15120601A IL15120601A IL151206A0 IL 151206 A0 IL151206 A0 IL 151206A0 IL 15120601 A IL15120601 A IL 15120601A IL 15120601 A IL15120601 A IL 15120601A IL 151206 A0 IL151206 A0 IL 151206A0
Authority
IL
Israel
Prior art keywords
propoxy
chloro
amine
nitroquinazolin
morpholin
Prior art date
Application number
IL15120601A
Other languages
English (en)
Original Assignee
Godecke Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Godecke Gmbh filed Critical Godecke Gmbh
Publication of IL151206A0 publication Critical patent/IL151206A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
IL15120601A 2000-02-26 2001-01-23 Process for the simple preparation of (3-chloro-4-fluorophenyl)-7-(3-morpholin-4-yl-propoxy)-6-nitroquinazolin-4-yl]-amine or (3-chloro-4-yl-propoxy)-6-nitroquinazolin-4-yl]-amine or (3-chloro-4-fluorophenyl)-[7(3-morpholin-4-yl-propoxy)-6-aminoquinazolin-4-yl]-amine IL151206A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10009267A DE10009267A1 (de) 2000-02-26 2000-02-26 Verfahren zur einfachen Herstellung von (3-Chlor-4-fluor-phenyl)-[7-(3-morpholin-4-yl-propoxy)-6-nitro-quinazolin-4-yl]-amin bzw. (3-Chlor-4-fluor-phenyl)-[7-(3-morpholin-4-yl-propoxy)-6-amino-quinazolin-4-yl]-amin
PCT/EP2001/000695 WO2001062743A2 (de) 2000-02-26 2001-01-23 Verfahren zur einfachen herstellung von (3-chlor-4-fluor-phenyl)-[7-(3-morpholin-4-yl-propoxy)-6-nitro-quinazolin-4-yl]-amin bzw. (3-chlor-4-fluor-phenyl)-[7-(3-morpholin-4-yl-propoxy)-6-amino -quinazolin-4-yl]-amin

Publications (1)

Publication Number Publication Date
IL151206A0 true IL151206A0 (en) 2003-04-10

Family

ID=7632648

Family Applications (1)

Application Number Title Priority Date Filing Date
IL15120601A IL151206A0 (en) 2000-02-26 2001-01-23 Process for the simple preparation of (3-chloro-4-fluorophenyl)-7-(3-morpholin-4-yl-propoxy)-6-nitroquinazolin-4-yl]-amine or (3-chloro-4-yl-propoxy)-6-nitroquinazolin-4-yl]-amine or (3-chloro-4-fluorophenyl)-[7(3-morpholin-4-yl-propoxy)-6-aminoquinazolin-4-yl]-amine

Country Status (31)

Country Link
US (1) US20030050313A1 (xx)
EP (1) EP1265874B1 (xx)
JP (1) JP2003524006A (xx)
KR (1) KR20030011773A (xx)
CN (1) CN1171877C (xx)
AR (1) AR027377A1 (xx)
AT (1) ATE296810T1 (xx)
AU (1) AU2001228478A1 (xx)
BR (1) BR0108695A (xx)
CA (1) CA2401171A1 (xx)
CO (1) CO5280058A1 (xx)
DE (2) DE10009267A1 (xx)
EA (1) EA005213B1 (xx)
EG (1) EG23221A (xx)
ES (1) ES2240483T3 (xx)
GT (1) GT200100025A (xx)
HK (1) HK1054551B (xx)
HU (1) HUP0204510A3 (xx)
IL (1) IL151206A0 (xx)
MX (1) MXPA02008301A (xx)
MY (1) MY133846A (xx)
PA (1) PA8512701A1 (xx)
PE (1) PE20011073A1 (xx)
PL (1) PL357774A1 (xx)
PT (1) PT1265874E (xx)
SV (1) SV2002000320A (xx)
TN (1) TNSN01031A1 (xx)
UY (1) UY26594A1 (xx)
WO (1) WO2001062743A2 (xx)
YU (1) YU62502A (xx)
ZA (1) ZA200206107B (xx)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20040945A1 (es) * 2003-02-05 2004-12-14 Warner Lambert Co Preparacion de quinazolinas substituidas
WO2006081741A1 (fr) * 2005-02-05 2006-08-10 Piaoyang Sun Dérivés de quinazoline ou leurs sels de qualité pharmaceutique, synthèse et applications médicales desdites substances
JP5250901B2 (ja) * 2007-02-23 2013-07-31 学校法人慶應義塾 アニリノキナゾリン系化合物及びその用途
US7829574B2 (en) 2008-05-09 2010-11-09 Hutchison Medipharma Enterprises Limited Substituted quinazoline compounds and their use in treating angiogenesis-related diseases
CN105399688A (zh) * 2015-12-02 2016-03-16 西南科技大学 一种吉非替尼的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL190489B1 (pl) * 1996-04-12 2005-12-30 Warner Lambert Co Nieodwracalne inhibitory kinaz tyrozyny, kompozycja farmaceutyczna je zawierająca i ich zastosowanie

Also Published As

Publication number Publication date
HUP0204510A3 (en) 2003-07-28
AR027377A1 (es) 2003-03-26
JP2003524006A (ja) 2003-08-12
CO5280058A1 (es) 2003-05-30
UY26594A1 (es) 2001-09-28
YU62502A (sh) 2005-03-15
MY133846A (en) 2007-11-30
PL357774A1 (en) 2004-07-26
PE20011073A1 (es) 2001-12-16
DE50106391D1 (de) 2005-07-07
GT200100025A (es) 2003-09-22
PA8512701A1 (es) 2002-02-21
WO2001062743A3 (de) 2002-03-14
CN1171877C (zh) 2004-10-20
CN1406232A (zh) 2003-03-26
DE10009267A1 (de) 2001-08-30
KR20030011773A (ko) 2003-02-11
US20030050313A1 (en) 2003-03-13
EA200200885A1 (ru) 2003-02-27
HUP0204510A2 (en) 2003-05-28
HK1054551B (zh) 2005-06-03
MXPA02008301A (es) 2004-05-14
ZA200206107B (en) 2003-07-31
EG23221A (en) 2004-08-31
EP1265874B1 (de) 2005-06-01
AU2001228478A1 (en) 2001-09-03
CA2401171A1 (en) 2001-08-30
EP1265874A2 (de) 2002-12-18
PT1265874E (pt) 2005-08-31
EA005213B1 (ru) 2004-12-30
TNSN01031A1 (en) 2005-11-10
SV2002000320A (es) 2002-06-07
WO2001062743A2 (de) 2001-08-30
ATE296810T1 (de) 2005-06-15
BR0108695A (pt) 2002-12-10
ES2240483T3 (es) 2005-10-16
HK1054551A1 (en) 2003-12-05

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