AR019678A1 - Compuestos organicos - Google Patents

Compuestos organicos

Info

Publication number
AR019678A1
AR019678A1 ARP990102880A ARP990102880A AR019678A1 AR 019678 A1 AR019678 A1 AR 019678A1 AR P990102880 A ARP990102880 A AR P990102880A AR P990102880 A ARP990102880 A AR P990102880A AR 019678 A1 AR019678 A1 AR 019678A1
Authority
AR
Argentina
Prior art keywords
alkyl
optionally substituted
unsubstituted
halogen
hydrogen
Prior art date
Application number
ARP990102880A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of AR019678A1 publication Critical patent/AR019678A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/76—1,3-Oxazoles; Hydrogenated 1,3-oxazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/84—Naphthothiazoles

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Compuestos benzazol de la formula (1, donde: R1 y R2 son iguales o diferentes, y significan hidrogeno, hidroxilo, amino, halogeno, alquilo C1-6,haloalquilo C1-6, alquenilo C2-6, haloalquenilo C2-6, cicloalquilo C3-6, halocicloalquilo C3-6, alcoxi C1-6, haloalcoxi C1-6, fenilo insustituido, o fenilo queestá opcionalmente sustituido por halogeno o alquilo C1-6; nitro, ciano, isotiocianato, carboxi, alcoxi C1-6-carbonilo, haloalcoxi C1-6-carbonilo, alquiloC1-6-carbamido, que está opcionalmente sustituido por fenilo, o por fenoxi insustituido o sustituido por halogeno; PhNH(CO)NH, alquilo C1-6-sulfonilo,haloalquilo C1-6-sulfonilo, benzoílo insustituido u opcionalmente sustituido por halogeno; feniltionilo insustituido u opcionalmente sustituidopor halogeno, ofenilsulfonilo; R3 y R4, independientemente uno del otro, hidrogeno, R1, R2, o son juntos un puente de CH=CH-CH=CH; X es NR5, O o S; R5 es hidrogeno o alquiloC1-6; Y es N, CR6, o C=O; R6 es hidrogeno, hidroxilo, alquilo C1-6, alquiloC1-6-carbonilo, alcoxi C1-6, ciano, 2-di(alquilo C1-6)aminoetenilo, (alquilo C1-6)NHC(=S)NHCH2, fenilo, tiazolilo, fenilamino, en donde el grupo fenilo está insustituido u opcionalmente sustituido por alcoxi C1-6; alquilo C1-6-carbamido,alcoxi C1-6-carbamido, guanidilo, amino, hidroxialquilo C2-6-amino, o fenilsulfonilamino, en donde el grupo fenilo está insustituido u opcionalmente sustituidopor alquilo C1-6; Z es N o CR7; y R7 es hidrogeno o alquilo C1-6, se pueden utilizar como composicionesrepelentes de insectos, de ácaros, y de garrapatas, yse pueden producir de una manera conocida; proceso para la preparacion de composiciones repelentes de insectos, uso de dichos compuestos y proceso para alejarinsectos, ácaros o garrapatas de lugares o materiales en donde se quiera.
ARP990102880A 1998-06-18 1999-06-16 Compuestos organicos AR019678A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH132098 1998-06-18

Publications (1)

Publication Number Publication Date
AR019678A1 true AR019678A1 (es) 2002-03-13

Family

ID=4207690

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP990102880A AR019678A1 (es) 1998-06-18 1999-06-16 Compuestos organicos

Country Status (18)

Country Link
US (1) US6410578B1 (es)
EP (1) EP1087952B1 (es)
JP (1) JP2002518381A (es)
KR (1) KR100597913B1 (es)
CN (1) CN1302293A (es)
AR (1) AR019678A1 (es)
AT (1) ATE268327T1 (es)
AU (1) AU753691B2 (es)
BR (1) BR9911353A (es)
CA (1) CA2330977A1 (es)
DE (1) DE69917777T2 (es)
DK (1) DK1087952T3 (es)
ES (1) ES2221748T3 (es)
NZ (1) NZ507440A (es)
PT (1) PT1087952E (es)
RU (1) RU2227458C2 (es)
WO (1) WO1999065886A1 (es)
ZA (1) ZA200006206B (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000034248A1 (en) 1998-12-04 2000-06-15 Neurosearch A/S New benzimidazolone-, benzoxazolone-, or benzothiazolone derivatives as ion channel modulating agents
CO5261573A1 (es) 1999-11-19 2003-03-31 Novartis Ag Derivados de benzoxa y bezotiazol, compuesto y composicion farmaceutica que los contiene y proceso para la preparacion de la mencionada composicion
US6448281B1 (en) 2000-07-06 2002-09-10 Boehringer Ingelheim (Canada) Ltd. Viral polymerase inhibitors
EP1581217A4 (en) * 2002-11-01 2007-07-11 Merck & Co Inc CARBONYLAMINO-BENZIMIDAZOLE DERIVATIVES AS MODULATORS OF THE ANDROGEN RECEPTOR
US20050261347A1 (en) * 2003-10-24 2005-11-24 Wyeth Dihydrobenzofuranyl alkanamine derivatives and methods for using same
US7435837B2 (en) * 2003-10-24 2008-10-14 Wyeth Dihydrobenzofuranyl alkanamine derivatives and methods for using same
ES2431314T3 (es) 2004-02-20 2013-11-26 Boehringer Ingelheim International Gmbh Inhibidores de polimerasa vírica
BRPI0517466A (pt) * 2004-10-22 2008-10-07 Bayer Cropscience Ag derivados de 3-(dihaloalquenil) fenila inseticidas
JP2008538581A (ja) * 2005-04-22 2008-10-30 ワイス ｛［（２ｒ）−７−（２，６−ジクロロフェニル）−５−フルオロ−２，３−ジヒドロ−１−ベンゾフラン−２−イル］メチル｝アミン塩酸塩の結晶形態
TW200720255A (en) 2005-07-13 2007-06-01 Taiho Pharmaceutical Co Ltd Benzoimidazole compound capable of inhibiting prostaglandin d synthetase
FR2967672B1 (fr) 2010-11-22 2012-12-28 Sanofi Aventis Derives de nitrobenzothiazoles, leur preparation et leurs applications therapeutiques
JP6143713B2 (ja) * 2014-06-16 2017-06-07 住友化学株式会社 ネズミ目動物忌避剤

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3624204A (en) * 1969-04-24 1971-11-30 Mikhail Konstantinovich Stepan Protective agent against mosquitoes, sand-flies, black-flies, gnats, horse-flies, fleas and ticks
BE758241A (fr) 1969-11-03 1971-04-30 Agfa Gevaert Nv Bereiding van 2-alkyl-thiazolen en 2-alkyl-selenazolen met een geanelleerde aromatische ring
CH565164A5 (en) * 1971-12-07 1975-08-15 Ciba Geigy Ag Isocyanato-benzoxazoles-benzothiazoles and benimidazoles - as anthelmintics and antimicrobials
US4003750A (en) 1973-05-03 1977-01-18 Eastman Kodak Company Silver halide emulsion containing photographic sensitizing dyes
FR2244506B1 (es) 1973-06-26 1977-02-25 Inst Nat Sante Rech Med
US3876791A (en) * 1973-11-30 1975-04-08 Uniroyal Inc Control of acarids using certain benzothiazoles or benzothiazolines
CH585214A5 (en) * 1974-09-12 1977-02-28 Ciba Geigy Ag Prepn. of anthelmintic (6)-isothiocyano-benzo-thiazoles - from (6)-amino-benzothiazoles
GB1507457A (en) 1974-11-12 1978-04-12 Agfa Gevaert Fixer compositions used in planographic printing
SE7713314L (sv) * 1976-12-17 1978-06-18 Rohm & Haas Artropodrepellenter
EP0007616B1 (de) * 1978-07-27 1982-05-12 Ciba-Geigy Ag Isothiocyanobenzthiazolderivat, Verfahren zu seiner Herstellung und seine Anwendung in anthelmintischen Mitteln
US4356180A (en) * 1979-02-02 1982-10-26 The United States Of America As Represented By The Secretary Of Agriculture Insect repellants
US4455308A (en) 1979-07-10 1984-06-19 Rohm And Haas Company Arthropod repellents
US4389401A (en) * 1979-07-10 1983-06-21 Rohm And Haas Company Arthropod repellents
DE3528032A1 (de) 1985-08-05 1987-02-05 Hoechst Ag Verfahren zur herstellung 2-substituierter benzthiazole
DE4018070A1 (de) 1990-06-06 1991-12-12 Bayer Ag Morpholinoharnstoff-derivate
JPH05291828A (ja) 1992-04-10 1993-11-05 Toshiba Corp 逓倍回路
JPH05294828A (ja) * 1992-04-17 1993-11-09 Kanebo Ltd 皮膚外用剤組成物
JPH09175926A (ja) * 1995-12-25 1997-07-08 Kanebo Ltd 皮膚外用剤組成物
US5601963A (en) * 1996-06-28 1997-02-11 Polaroid Corporation Silver halide emulsions
GB9619284D0 (en) * 1996-09-16 1996-10-30 Celltech Therapeutics Ltd Chemical compounds

Also Published As

Publication number Publication date
EP1087952B1 (en) 2004-06-02
KR100597913B1 (ko) 2006-07-10
WO1999065886A1 (en) 1999-12-23
PT1087952E (pt) 2004-08-31
ATE268327T1 (de) 2004-06-15
AU753691B2 (en) 2002-10-24
AU4611799A (en) 2000-01-05
BR9911353A (pt) 2001-03-13
ZA200006206B (en) 2001-06-25
DE69917777T2 (de) 2005-08-04
DE69917777D1 (de) 2004-07-08
RU2227458C2 (ru) 2004-04-27
EP1087952A1 (en) 2001-04-04
ES2221748T3 (es) 2005-01-01
CA2330977A1 (en) 1999-12-23
NZ507440A (en) 2003-04-29
DK1087952T3 (da) 2004-10-04
KR20010052966A (ko) 2001-06-25
CN1302293A (zh) 2001-07-04
JP2002518381A (ja) 2002-06-25
US6410578B1 (en) 2002-06-25

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