AR017079A1 - Una composicion farmaceutica, un procedimiento para la preparacion de la misma, un metodo de tratamiento y su uso. - Google Patents
Una composicion farmaceutica, un procedimiento para la preparacion de la misma, un metodo de tratamiento y su uso.Info
- Publication number
- AR017079A1 AR017079A1 ARP980104487A ARP980104487A AR017079A1 AR 017079 A1 AR017079 A1 AR 017079A1 AR P980104487 A ARP980104487 A AR P980104487A AR P980104487 A ARP980104487 A AR P980104487A AR 017079 A1 AR017079 A1 AR 017079A1
- Authority
- AR
- Argentina
- Prior art keywords
- pharmaceutical composition
- preparation
- procedure
- same
- treatment method
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1682—Processes
- A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Organic Chemistry (AREA)
- Neurosurgery (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Composicion farmacéutica, un proceso para la preparacion de la misma, un método de tratamiento y su uso, donde dicha composicion farmacéutica comprendemicropartículas poliméricas que incluyen una droga, preferentemente olanzapina, y un ácido graso, cuya composicion puede ser adaptada para proveer unavelocidad de liberacion de droga que es aproximadamente lineal en el tiempo, y que tiene un efecto de liberacion repentina o explosiva insignificante.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9718986.4A GB9718986D0 (en) | 1997-09-09 | 1997-09-09 | Controlled release microsphere delivery system |
Publications (1)
Publication Number | Publication Date |
---|---|
AR017079A1 true AR017079A1 (es) | 2001-08-22 |
Family
ID=10818687
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP980104487A AR017079A1 (es) | 1997-09-09 | 1998-09-09 | Una composicion farmaceutica, un procedimiento para la preparacion de la misma, un metodo de tratamiento y su uso. |
Country Status (10)
Country | Link |
---|---|
EP (1) | EP1011680A2 (es) |
JP (1) | JP2001515862A (es) |
AR (1) | AR017079A1 (es) |
AU (1) | AU745511B2 (es) |
CA (1) | CA2302762A1 (es) |
GB (1) | GB9718986D0 (es) |
NO (1) | NO20001219L (es) |
NZ (1) | NZ502710A (es) |
WO (1) | WO1999012549A2 (es) |
ZA (1) | ZA987762B (es) |
Families Citing this family (34)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6194006B1 (en) | 1998-12-30 | 2001-02-27 | Alkermes Controlled Therapeutics Inc. Ii | Preparation of microparticles having a selected release profile |
US6705757B2 (en) | 1999-11-12 | 2004-03-16 | Alkermes Controlled Therapeutics, Inc. Ii | Method and apparatus for preparing microparticles using in-line solvent extraction |
US6331317B1 (en) | 1999-11-12 | 2001-12-18 | Alkermes Controlled Therapeutics Ii Inc. | Apparatus and method for preparing microparticles |
US6495166B1 (en) | 1999-11-12 | 2002-12-17 | Alkermes Controlled Therapeutics Inc. | Apparatus and method for preparing microparticles using in-line solvent extraction |
ES2169980B1 (es) * | 1999-12-17 | 2003-11-01 | Lipotec Sa | Microcapsulas para la liberacion prolongada de farmacos. |
US6264987B1 (en) | 2000-05-19 | 2001-07-24 | Alkermes Controlled Therapeutics Inc. Ii | Method for preparing microparticles having a selected polymer molecular weight |
US6495164B1 (en) | 2000-05-25 | 2002-12-17 | Alkermes Controlled Therapeutics, Inc. I | Preparation of injectable suspensions having improved injectability |
US6824822B2 (en) | 2001-08-31 | 2004-11-30 | Alkermes Controlled Therapeutics Inc. Ii | Residual solvent extraction method and microparticles produced thereby |
US6471995B1 (en) | 2000-09-27 | 2002-10-29 | Alkermes Controlled Therapeutics, Inc. Ii | Apparatus and method for preparing microparticles using liquid-liquid extraction |
US20020114843A1 (en) | 2000-12-27 | 2002-08-22 | Ramstack J. Michael | Preparation of microparticles having improved flowability |
ES2605402T3 (es) | 2002-06-25 | 2017-03-14 | Takeda Pharmaceutical Company Limited | Procedimiento para producir una composición de liberación sostenida |
JP2006506397A (ja) * | 2002-10-31 | 2006-02-23 | ファイザー・プロダクツ・インク | 固体及び半固体高分子イオン・コンジュゲート |
PL1675573T4 (pl) | 2003-10-23 | 2016-04-29 | Otsuka Pharma Co Ltd | Sterylny preparat do wstrzykiwań arypiprazolu o kontrolowanym uwalnianiu i sposób |
MXPA06011924A (es) | 2004-04-15 | 2007-06-11 | Alkermes Inc | Dispositivo de liberacion continua base polimeros. |
CN101123951A (zh) | 2004-08-31 | 2008-02-13 | 辉瑞产品公司 | 包括低溶解性药物和聚合物的药物剂型 |
US11246913B2 (en) | 2005-02-03 | 2022-02-15 | Intarcia Therapeutics, Inc. | Suspension formulation comprising an insulinotropic peptide |
US7682356B2 (en) | 2006-08-09 | 2010-03-23 | Intarcia Therapeutics, Inc. | Osmotic delivery systems and piston assemblies for use therein |
MX2009003735A (es) * | 2006-10-05 | 2009-04-22 | Panacea Biotec Ltd | Composicion en deposito inyectable y su procedimiento de preparacion. |
GEP20125597B (en) | 2006-12-18 | 2012-08-10 | Takeda Pharmaceutical | Sustained-release composition and production method thereof |
CN105688191A (zh) | 2007-04-23 | 2016-06-22 | 精达制药公司 | 促胰岛素释放肽的混悬制剂及其应用 |
ES2661037T3 (es) | 2007-07-31 | 2018-03-27 | Otsuka Pharmaceutical Co., Ltd. | Procedimientos para producir una suspensión de aripiprazol y una formulación liofilizada |
EP2240155B1 (en) | 2008-02-13 | 2012-06-06 | Intarcia Therapeutics, Inc | Devices, formulations, and methods for delivery of multiple beneficial agents |
US8298561B2 (en) | 2009-09-28 | 2012-10-30 | Intarcia Therapeutics, Inc. | Rapid establishment and/or termination of substantial steady-state drug delivery |
ES2572948T3 (es) * | 2010-11-25 | 2016-06-03 | Shan Dong Luye Pharmaceutical Co., Ltd. | Composiciones de rotigotina o sales farmacéuticamente aceptables de rotigotina |
US20120208755A1 (en) | 2011-02-16 | 2012-08-16 | Intarcia Therapeutics, Inc. | Compositions, Devices and Methods of Use Thereof for the Treatment of Cancers |
JO3410B1 (ar) | 2011-06-07 | 2019-10-20 | Otsuka Pharma Co Ltd | تركيبة أريبيبرازول مجفف بالتبريد |
US9889085B1 (en) | 2014-09-30 | 2018-02-13 | Intarcia Therapeutics, Inc. | Therapeutic methods for the treatment of diabetes and related conditions for patients with high baseline HbA1c |
CA2987766A1 (en) | 2015-06-03 | 2016-12-08 | Intarcia Therapeutics, Inc. | Implant placement and removal systems |
MX2018014016A (es) | 2016-05-16 | 2019-08-01 | Intarcia Therapeutics Inc | Polipéptidos selectivos del receptor de glucagón y métodos para utilizarlos. |
USD860451S1 (en) | 2016-06-02 | 2019-09-17 | Intarcia Therapeutics, Inc. | Implant removal tool |
USD840030S1 (en) | 2016-06-02 | 2019-02-05 | Intarcia Therapeutics, Inc. | Implant placement guide |
WO2018129058A1 (en) | 2017-01-03 | 2018-07-12 | Intarcia Therapeutics, Inc. | Methods comprising continuous administration of a glp-1 receptor agonist and co-adminstration of a drug |
WO2018172850A1 (en) | 2017-03-20 | 2018-09-27 | Teva Pharmaceuticals International Gmbh | Sustained release olanzapine formulaitons |
KR102045721B1 (ko) * | 2019-03-27 | 2019-11-18 | 주식회사 씨트리 | 아픽사반 함유 미립구 제조용 분산상의 조성물 및 이로부터 제조되는 생체적합성 고분자 기반 아픽사반 함유 미립구 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4384975A (en) * | 1980-06-13 | 1983-05-24 | Sandoz, Inc. | Process for preparation of microspheres |
US4389330A (en) * | 1980-10-06 | 1983-06-21 | Stolle Research And Development Corporation | Microencapsulation process |
GB9009229D0 (en) * | 1990-04-25 | 1990-06-20 | Lilly Industries Ltd | Pharmaceutical compounds |
CA2148823C (en) * | 1992-11-17 | 1999-03-09 | Welfide Corporation | Sustained release microsphere preparation containing antipsychotic drug and production process thereof |
IL117612A0 (en) * | 1995-03-24 | 1996-07-23 | Lilly Co Eli | Granule formulation for olanzapine |
-
1997
- 1997-09-09 GB GBGB9718986.4A patent/GB9718986D0/en not_active Ceased
-
1998
- 1998-08-26 ZA ZA9807762A patent/ZA987762B/xx unknown
- 1998-09-07 CA CA002302762A patent/CA2302762A1/en not_active Abandoned
- 1998-09-07 WO PCT/GB1998/002692 patent/WO1999012549A2/en not_active Application Discontinuation
- 1998-09-07 EP EP98941610A patent/EP1011680A2/en not_active Withdrawn
- 1998-09-07 JP JP2000510446A patent/JP2001515862A/ja active Pending
- 1998-09-07 NZ NZ502710A patent/NZ502710A/en unknown
- 1998-09-07 AU AU89925/98A patent/AU745511B2/en not_active Ceased
- 1998-09-09 AR ARP980104487A patent/AR017079A1/es unknown
-
2000
- 2000-03-09 NO NO20001219A patent/NO20001219L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AU8992598A (en) | 1999-03-29 |
CA2302762A1 (en) | 1999-03-18 |
WO1999012549A3 (en) | 1999-05-06 |
JP2001515862A (ja) | 2001-09-25 |
WO1999012549A2 (en) | 1999-03-18 |
NO20001219D0 (no) | 2000-03-09 |
GB9718986D0 (en) | 1997-11-12 |
EP1011680A2 (en) | 2000-06-28 |
NZ502710A (en) | 2001-09-28 |
NO20001219L (no) | 2000-03-09 |
ZA987762B (en) | 2000-02-28 |
AU745511B2 (en) | 2002-03-21 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AR017079A1 (es) | Una composicion farmaceutica, un procedimiento para la preparacion de la misma, un metodo de tratamiento y su uso. | |
BR9611410A (pt) | Método e composição farmacêutica para regular a concentração de lipídios | |
MX9203116A (es) | Articulo compuesto que comprende microestructuras orientadas y metodo para su fabricacion. | |
ES2177022T3 (es) | Un itraconazol que exhibe una solubilidad mejorada, un metodo para preparar el mismo y una composicion farmaceutica para administracion oral que comprende el mismo. | |
MX9201782A (es) | Particulas de sustancias biologicamente activas, sustancialmente insolubles en agua, proceso para su produccion y composicion farmaceutica que las contiene. | |
DE59601880D1 (de) | Verfahren zur herstellung hydrophiler oder teilweise hydrophiler, anorganischer aerogele | |
CO5150154A1 (es) | Composicion de sustrato y metodo para usarlo para el secuestro de irritantes de la piel | |
AR004483A1 (es) | Compuestos para uso en terapia que comprenden un residuo de 1,3-propano diol como agente enlazante entre el residuo de ácido graso y un residuo bioactivo, usos de dichos compuestos y medicamentos , alimentos y formulaciones para el cuidado o tratamiento de la piel que comprenden a dichos compuestos | |
DE3769379D1 (de) | Entzuendungshemmende wirkstoffe, pharmazeutische zusammensetzungen und verfahren zur bekaempfung von entzuendungen. | |
ES2130638T3 (es) | Sistema para la liberacion de sustancia activa, filmogeno, vaporizable, para utilizar en las plantas. | |
BR9510302A (pt) | Forma de dosagem farmacêutical de liberação controlada método para tratamento sintomático da tosse método para preparar uma forma de dosagem farmacêutica de liberação controlada composição para uso no tratamento sintomático da tosse e aplicação de uma forma dosagem de moguisteina de liberação controlada | |
DK647789D0 (da) | Kosmetisk eller farmaceutisk komposition indeholdende mikrosfaerer af polymere eller af fedtstofferforsynet med mindst et aktivt produkt | |
SV2004001556A (es) | Preparaciones acidas de insulina con establidad mejorada | |
EE9700145A (et) | Tsükloalkaanpüridiinid, nende valmistamismeetod, kasutamine ravimite tootmiseks ja nimetatud ühendeid sisaldavad ravimid | |
ES2187201T3 (es) | Empleo de esteroles y de esterolesteres a nanoescala. | |
EE04540B1 (et) | Meetod bioloogiliselt sobivate biodegradeeruvate mikroosakeste valmistamiseks ja mikroosakeste kasutamine | |
ATE236627T1 (de) | Pharmazeutische zubereitung enhaltend eicosapentaensäure und/oder stearidonsäure | |
ES2113095T3 (es) | Preparacion solida de liberacion rapida, su produccion y su uso. | |
ES2137372T3 (es) | Solucion antifungica para las uñas. | |
ES2141208T3 (es) | Utilizacion de una cantidad eficaz de sustancias activas para el tratamiento de pieles mixtas. | |
RS49602B (sr) | Farmaceutske mikrosfere valproinske kiseline za oralnu upotrebu | |
ES2174533T3 (es) | Uso de una mezcla de un diol y un acido alfa-hidroxi para el tratamiento de enfermedades de la piel hiperqueratoticas. | |
ES2103369T3 (es) | Derivados de lanolina como sustancias que aceleran la penetracion y su aplicacion en sustancias farmaceuticas u otras formulaciones que contienen sustancias biologicamente activas. | |
FI972949A0 (fi) | Lääkemuoto kollagenaasin vapauttamiseksi haavoihin ja sen valmistusmenetelmiä | |
MX9304185A (es) | Producto y composicion farmaceutica que lo contiene para el tratamiento de la mastitis y la mestritis bovina. |