AP370A - Process for the preparation of substituted steroidal dienes. - Google Patents
Process for the preparation of substituted steroidal dienes. Download PDFInfo
- Publication number
- AP370A AP370A APAP/P/1993/000473A AP9300473A AP370A AP 370 A AP370 A AP 370A AP 9300473 A AP9300473 A AP 9300473A AP 370 A AP370 A AP 370A
- Authority
- AP
- ARIPO
- Prior art keywords
- reagent
- process according
- chloride
- vilsmeier reagent
- source
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
- C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0066—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US81717992A | 1992-01-06 | 1992-01-06 | |
US94134892A | 1992-09-04 | 1992-09-04 |
Publications (2)
Publication Number | Publication Date |
---|---|
AP9300473A0 AP9300473A0 (en) | 1993-01-31 |
AP370A true AP370A (en) | 1994-11-10 |
Family
ID=27124147
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
APAP/P/1993/000473A AP370A (en) | 1992-01-06 | 1993-01-05 | Process for the preparation of substituted steroidal dienes. |
Country Status (23)
Country | Link |
---|---|
EP (1) | EP0643723A4 (no) |
JP (1) | JPH07505138A (no) |
KR (1) | KR940703849A (no) |
CN (1) | CN1077201A (no) |
AP (1) | AP370A (no) |
AU (1) | AU666167B2 (no) |
BG (1) | BG98887A (no) |
BR (1) | BR9305786A (no) |
CA (1) | CA2127272A1 (no) |
CZ (1) | CZ161994A3 (no) |
FI (1) | FI943214A (no) |
HU (1) | HUT68273A (no) |
IL (1) | IL104302A (no) |
MA (1) | MA22761A1 (no) |
MX (1) | MX9300025A (no) |
NO (1) | NO942535D0 (no) |
NZ (1) | NZ246788A (no) |
OA (1) | OA09961A (no) |
RU (1) | RU94038223A (no) |
SI (1) | SI9300006A (no) |
SK (1) | SK80094A3 (no) |
TW (1) | TW300226B (no) |
WO (1) | WO1993014106A1 (no) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5683995A (en) * | 1992-11-18 | 1997-11-04 | Smithkline Beecham Corporation | 17 substituted acyl-3-carboxy 3,5-diene steroidals as α-reductase inhibitors |
US5641765A (en) * | 1992-11-18 | 1997-06-24 | Smithkline Beecham Corporation | 17-αand 17-βsubstituted acyl-3-carboxy-3,5-dienes and use in inhibiting 5-α-reductase |
KR20070034574A (ko) | 2004-06-08 | 2007-03-28 | 템플 유니버시티-오브 더 커먼웰쓰 시스템 오브 하이어 에듀케이션 | 헤테로아릴 술폰 및 술폰아미드 및 이들의 치료상의 용도 |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5017568A (en) * | 1987-04-29 | 1991-05-21 | Smithkline Beecham Corporation | Steriod 5-alpha-reductase inhibitors |
-
1993
- 1993-01-04 IL IL104302A patent/IL104302A/en not_active IP Right Cessation
- 1993-01-05 AP APAP/P/1993/000473A patent/AP370A/en active
- 1993-01-05 MA MA23050A patent/MA22761A1/fr unknown
- 1993-01-06 RU RU94038223/04A patent/RU94038223A/ru unknown
- 1993-01-06 SI SI19939300006A patent/SI9300006A/sl unknown
- 1993-01-06 JP JP5512542A patent/JPH07505138A/ja active Pending
- 1993-01-06 CN CN93101175A patent/CN1077201A/zh active Pending
- 1993-01-06 CA CA002127272A patent/CA2127272A1/en not_active Abandoned
- 1993-01-06 NZ NZ246788A patent/NZ246788A/en unknown
- 1993-01-06 EP EP93902957A patent/EP0643723A4/en not_active Ceased
- 1993-01-06 CZ CZ941619A patent/CZ161994A3/cs unknown
- 1993-01-06 HU HU9402030A patent/HUT68273A/hu unknown
- 1993-01-06 WO PCT/US1993/000079 patent/WO1993014106A1/en not_active Application Discontinuation
- 1993-01-06 SK SK800-94A patent/SK80094A3/sk unknown
- 1993-01-06 BR BR9305786A patent/BR9305786A/pt not_active Application Discontinuation
- 1993-01-06 AU AU34348/93A patent/AU666167B2/en not_active Ceased
- 1993-01-06 KR KR1019940702343A patent/KR940703849A/ko not_active Application Discontinuation
- 1993-01-06 MX MX9300025A patent/MX9300025A/es unknown
- 1993-01-29 TW TW082100552A patent/TW300226B/zh active
-
1994
- 1994-07-04 OA OA60533A patent/OA09961A/en unknown
- 1994-07-05 NO NO942535A patent/NO942535D0/no unknown
- 1994-07-05 FI FI943214A patent/FI943214A/fi unknown
- 1994-07-05 BG BG98887A patent/BG98887A/bg unknown
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5017568A (en) * | 1987-04-29 | 1991-05-21 | Smithkline Beecham Corporation | Steriod 5-alpha-reductase inhibitors |
Also Published As
Publication number | Publication date |
---|---|
HUT68273A (en) | 1995-06-28 |
SI9300006A (en) | 1993-09-30 |
AU3434893A (en) | 1993-08-03 |
WO1993014106A1 (en) | 1993-07-22 |
CZ161994A3 (en) | 1995-03-15 |
SK80094A3 (en) | 1994-12-07 |
OA09961A (en) | 1995-12-11 |
JPH07505138A (ja) | 1995-06-08 |
HU9402030D0 (en) | 1994-09-28 |
TW300226B (no) | 1997-03-11 |
EP0643723A1 (en) | 1995-03-22 |
BR9305786A (pt) | 1997-02-18 |
NZ246788A (en) | 1996-11-26 |
AP9300473A0 (en) | 1993-01-31 |
FI943214A0 (fi) | 1994-07-05 |
AU666167B2 (en) | 1996-02-01 |
RU94038223A (ru) | 1997-04-20 |
IL104302A0 (en) | 1993-05-13 |
NO942535L (no) | 1994-07-05 |
EP0643723A4 (en) | 1995-05-10 |
MX9300025A (es) | 1994-01-31 |
FI943214A (fi) | 1994-07-05 |
NO942535D0 (no) | 1994-07-05 |
CA2127272A1 (en) | 1993-07-22 |
IL104302A (en) | 1998-02-22 |
BG98887A (bg) | 1995-05-31 |
MA22761A1 (fr) | 1993-10-01 |
KR940703849A (ko) | 1994-12-12 |
CN1077201A (zh) | 1993-10-13 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
Abarbri et al. | Efficient synthesis of conjugated (2E)-or (2Z)-en-4-ynoic acids and (2E, 4E)-or (2Z, 4E)-dienoic acids via palladium-catalysed cross coupling | |
US8143463B2 (en) | Process for the preparation of delmopinol and derivatives thereof | |
JP3173602B2 (ja) | エンイン誘導体の新規製造中間体及びその製造法 | |
AP370A (en) | Process for the preparation of substituted steroidal dienes. | |
JPH05507271A (ja) | 10β―H―ステロイドの製法 | |
AP361A (en) | Process for the preparation of substituted steroidal benzo esters and acids. | |
CA1156646A (en) | 5.beta.-HYDROXY-.DELTA..SUP.6-STEROIDS | |
JP3672969B2 (ja) | ハロアルキルフェロセンの合成方法 | |
CN110156738B (zh) | 一种伊鲁烷型倍半萜反应中间体及天然产物的全合成方法 | |
JP2002030046A (ja) | アリールオレフィンのアミノ化によるアリールエチルアミンの製造法 | |
EP1207153A1 (en) | Process for the preparation of indole derivatives or salts thereof | |
US5908944A (en) | Methylation or ethylation agent and process for 1,4-addition of a methyl or ethyl group to an α, β-unsaturated keto compound | |
Mukaiyama et al. | A convenient method for the synthesis of α, β-unsaturated carbonyl compounds | |
SI9300067A (en) | Process for the preparation of substituted steroidal dienes | |
Kotlarek | Metal-hexamethylphosphoramide reduction. IV. Birch-like reduction of 2, 6-and 2, 7-dimethoxynaphthalenes | |
JPH05208981A (ja) | イミダゾチアゾロン誘導体の調製法 | |
Caputo et al. | Chemistry of Ethanediyl S, S-Acetals-4. Promising Way to Cis-Substituted Olefins, Stereoselectively from Carbonyl Compounds | |
US20090221831A1 (en) | Method for Producing N,N-Bis(Pyridin-2Ylmethyl)-1,1-Bis(Pyridin-2-Yl)-1-Aminoalkane Compounds and Metal Complex Salts Containing These Compounds | |
JPH04273886A (ja) | モノハロアルキルフェロセンおよび4−クロロブチルフェロセンの合成方法 | |
GB2028809A (en) | Dextrorotatory octahydro- indoloquinolizines | |
JPH10507176A (ja) | 17−ベータ−置換アンドロスタ−3,5−ジエン−3−カルボン酸の製法 | |
NO134114B (no) | ||
JPS6087264A (ja) | ピリジン類の臭化水素及び臭素の付加体の製造法 |