AP3179A - Benzofuranyl derivatives used as glucokinase inhibitors - Google Patents

Benzofuranyl derivatives used as glucokinase inhibitors

Info

Publication number
AP3179A
AP3179A AP2011005882A AP2011005882A AP3179A AP 3179 A AP3179 A AP 3179A AP 2011005882 A AP2011005882 A AP 2011005882A AP 2011005882 A AP2011005882 A AP 2011005882A AP 3179 A AP3179 A AP 3179A
Authority
AP
ARIPO
Prior art keywords
derivatives used
glucokinase inhibitors
benzofuranyl derivatives
benzofuranyl
glucokinase
Prior art date
Application number
AP2011005882A
Other languages
English (en)
Other versions
AP2011005882A0 (en
Inventor
Jeffrey Allen Pfeferkorn
Anthony Lai Ling
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42124287&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP3179(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of AP2011005882A0 publication Critical patent/AP2011005882A0/xx
Application granted granted Critical
Publication of AP3179A publication Critical patent/AP3179A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Oncology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AP2011005882A 2009-03-11 2010-03-04 Benzofuranyl derivatives used as glucokinase inhibitors AP3179A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US15909909P 2009-03-11 2009-03-11
PCT/IB2010/050943 WO2010103437A1 (en) 2009-03-11 2010-03-04 Benzofuranyl derivatives used as glucokinase inhibitors

Publications (2)

Publication Number Publication Date
AP2011005882A0 AP2011005882A0 (en) 2011-10-31
AP3179A true AP3179A (en) 2015-03-31

Family

ID=42124287

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2011005882A AP3179A (en) 2009-03-11 2010-03-04 Benzofuranyl derivatives used as glucokinase inhibitors

Country Status (38)

Country Link
US (2) US8455496B2 (de)
EP (2) EP2406253B1 (de)
JP (1) JP5086480B2 (de)
KR (1) KR101295937B1 (de)
CN (1) CN102388038B (de)
AP (1) AP3179A (de)
AR (1) AR075729A1 (de)
AU (1) AU2010222589B2 (de)
BR (1) BRPI1013246B1 (de)
CA (1) CA2754681C (de)
CL (1) CL2011002185A1 (de)
CO (1) CO6430427A2 (de)
CR (1) CR20110467A (de)
CU (1) CU24036B1 (de)
DK (1) DK2406253T3 (de)
DO (1) DOP2011000279A (de)
EA (1) EA018894B1 (de)
EC (1) ECSP11011306A (de)
ES (1) ES2427279T3 (de)
GE (1) GEP20156239B (de)
HK (1) HK1164281A1 (de)
HR (1) HRP20130661T1 (de)
IL (1) IL214942A (de)
MA (1) MA33119B1 (de)
MY (1) MY151246A (de)
NI (1) NI201100166A (de)
NZ (1) NZ595024A (de)
PE (1) PE20120668A1 (de)
PL (1) PL2406253T3 (de)
PT (1) PT2406253E (de)
RS (1) RS52903B (de)
SI (1) SI2406253T1 (de)
TN (1) TN2011000454A1 (de)
TW (1) TWI383981B (de)
UA (1) UA99882C2 (de)
UY (1) UY32480A (de)
WO (1) WO2010103437A1 (de)
ZA (1) ZA201106632B (de)

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UA99882C2 (uk) 2012-10-10
JP2012520286A (ja) 2012-09-06
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EP2406253B1 (de) 2013-07-03
HK1164281A1 (en) 2012-09-21
SI2406253T1 (sl) 2013-09-30
ZA201106632B (en) 2012-05-30
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BRPI1013246A2 (pt) 2016-04-05
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KR101295937B1 (ko) 2013-08-14
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