AP309A - Novel pyrrolopyridines, pharmaceutical compositions containing them and their preparations. - Google Patents

Novel pyrrolopyridines, pharmaceutical compositions containing them and their preparations. Download PDF

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Publication number
AP309A
AP309A APAP/P/1992/000369A AP9200369A AP309A AP 309 A AP309 A AP 309A AP 9200369 A AP9200369 A AP 9200369A AP 309 A AP309 A AP 309A
Authority
AP
ARIPO
Prior art keywords
compound
formula
alkyl
pharmaceutically acceptable
pyridine
Prior art date
Application number
APAP/P/1992/000369A
Other languages
English (en)
Other versions
AP9200369A0 (en
Inventor
Carin Brivin
Marie Elebring
Stig Carlsson
Robert Carter
Original Assignee
Ab Astra
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ab Astra filed Critical Ab Astra
Publication of AP9200369A0 publication Critical patent/AP9200369A0/xx
Application granted granted Critical
Publication of AP309A publication Critical patent/AP309A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
APAP/P/1992/000369A 1991-03-27 1992-03-23 Novel pyrrolopyridines, pharmaceutical compositions containing them and their preparations. AP309A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9100920A SE9100920D0 (sv) 1991-03-27 1991-03-27 New active compounds

Publications (2)

Publication Number Publication Date
AP9200369A0 AP9200369A0 (en) 1992-04-30
AP309A true AP309A (en) 1994-01-13

Family

ID=20382295

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/1992/000369A AP309A (en) 1991-03-27 1992-03-23 Novel pyrrolopyridines, pharmaceutical compositions containing them and their preparations.

Country Status (30)

Country Link
US (1) US5439917A (es)
EP (2) EP0580616A1 (es)
JP (1) JP3122792B2 (es)
CN (1) CN1067892A (es)
AP (1) AP309A (es)
AT (1) ATE175672T1 (es)
AU (1) AU655634B2 (es)
BG (1) BG98124A (es)
CA (1) CA2106880A1 (es)
DE (1) DE69228142T2 (es)
DK (1) DK0509974T3 (es)
ES (1) ES2129039T3 (es)
FI (1) FI934203A (es)
GR (1) GR3029834T3 (es)
HU (1) HUT65948A (es)
IE (1) IE920915A1 (es)
IL (1) IL101347A0 (es)
IS (1) IS3827A (es)
JO (1) JO1704B1 (es)
MA (1) MA22477A1 (es)
MX (1) MX9201324A (es)
NO (1) NO933425L (es)
NZ (1) NZ241943A (es)
SE (1) SE9100920D0 (es)
SK (1) SK103093A3 (es)
TN (1) TNSN92026A1 (es)
TW (1) TW198032B (es)
WO (1) WO1992017477A1 (es)
YU (1) YU30292A (es)
ZA (1) ZA921823B (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9100920D0 (sv) * 1991-03-27 1991-03-27 Astra Ab New active compounds
US6852739B1 (en) * 1999-02-26 2005-02-08 Nitromed Inc. Methods using proton pump inhibitors and nitric oxide donors
CA2699568C (en) * 1999-12-24 2013-03-12 Aventis Pharma Limited Azaindoles
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
GB0115109D0 (en) 2001-06-21 2001-08-15 Aventis Pharma Ltd Chemical compounds
MY140561A (en) * 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
EP1490364B1 (en) 2002-03-28 2007-09-26 Eisai R&D Management Co., Ltd. 7-azaindoles as inhibitors of c-jun n-terminal kinases for the treatment of neurodegenerative disorders
CA2493618A1 (en) * 2002-08-01 2004-02-12 Nitromed, Inc. Nitrosated proton pump inhibitors, compositions and methods of use
GB0305142D0 (en) * 2003-03-06 2003-04-09 Eisai London Res Lab Ltd Synthesis
PL1606261T3 (pl) 2003-03-10 2010-04-30 Astrazeneca Ab Nowy sposób przygotowania roflumilastu
US6981980B2 (en) 2003-03-19 2006-01-03 Phagia Technology Self-inflating intragastric volume-occupying device
WO2004101565A2 (en) * 2003-05-16 2004-11-25 Eisai Co., Ltd. Jnk inhibitors
GB0405055D0 (en) * 2004-03-05 2004-04-07 Eisai London Res Lab Ltd JNK inhibitors
ES2421916T3 (es) * 2005-03-16 2013-09-06 Nycomed Gmbh Forma farmacéutica de sabor enmascarado que contiene roflumilast
GB0516156D0 (en) * 2005-08-05 2005-09-14 Eisai London Res Lab Ltd JNK inhibitors
CL2007002617A1 (es) 2006-09-11 2008-05-16 Sanofi Aventis Compuestos derivados de pirrolo[2,3-b]pirazin-6-ilo; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar inflamacion de las articulaciones, artritis reumatoide, tumores, linfoma de las celulas del manto.
EP2486910A3 (en) 2006-10-27 2012-08-22 The Curators Of The University Of Missouri Multi-chambered apparatus comprising a dispenser head
EP2252274A4 (en) 2008-02-20 2011-05-11 Univ Missouri COMPOSITION COMPRISING A COMBINATION OF OMEPRAZOLE AND LANSOPRAZOLE, AND A BUFFER AGENT, AND METHODS OF USING THE SAME
KR102348222B1 (ko) * 2020-05-15 2022-01-10 대한민국 아동지킴이 과속방지시설

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0509974A1 (en) * 1991-03-27 1992-10-21 Astra Aktiebolag Pyrrolo[2,3-b]pyridines having therapeutic activity and a process for the preparation thereof

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0509974A1 (en) * 1991-03-27 1992-10-21 Astra Aktiebolag Pyrrolo[2,3-b]pyridines having therapeutic activity and a process for the preparation thereof

Also Published As

Publication number Publication date
ATE175672T1 (de) 1999-01-15
DK0509974T3 (da) 1999-08-30
EP0580616A1 (en) 1994-02-02
NO933425L (no) 1993-10-25
BG98124A (en) 1994-11-15
NZ241943A (en) 1993-12-23
IL101347A0 (en) 1992-11-15
MX9201324A (es) 1992-10-01
CA2106880A1 (en) 1992-09-28
CN1067892A (zh) 1993-01-13
US5439917A (en) 1995-08-08
SE9100920D0 (sv) 1991-03-27
ZA921823B (en) 1992-11-25
HU9302741D0 (en) 1993-12-28
AP9200369A0 (en) 1992-04-30
WO1992017477A1 (en) 1992-10-15
ES2129039T3 (es) 1999-06-01
AU655634B2 (en) 1995-01-05
AU1426092A (en) 1992-11-02
IS3827A (is) 1992-09-28
FI934203A0 (fi) 1993-09-24
IE920915A1 (en) 1992-10-07
SK103093A3 (en) 1994-08-10
DE69228142D1 (de) 1999-02-25
HUT65948A (en) 1994-08-29
JPH06506448A (ja) 1994-07-21
EP0509974A1 (en) 1992-10-21
FI934203A (fi) 1993-09-24
NO933425D0 (no) 1993-09-24
EP0509974B1 (en) 1999-01-13
YU30292A (sh) 1995-01-31
TNSN92026A1 (fr) 1993-06-08
JP3122792B2 (ja) 2001-01-09
GR3029834T3 (en) 1999-06-30
TW198032B (es) 1993-01-11
DE69228142T2 (de) 1999-07-22
JO1704B1 (en) 1992-12-15
MA22477A1 (fr) 1992-10-01

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