AP3048A - Agomelatine hydrohalide complex and preparation method thereof - Google Patents

Agomelatine hydrohalide complex and preparation method thereof

Info

Publication number
AP3048A
AP3048A AP2011005845A AP2011005845A AP3048A AP 3048 A AP3048 A AP 3048A AP 2011005845 A AP2011005845 A AP 2011005845A AP 2011005845 A AP2011005845 A AP 2011005845A AP 3048 A AP3048 A AP 3048A
Authority
AP
ARIPO
Prior art keywords
preparation
agomelatine
complex
hydrohalide complex
agomelatine hydrohalide
Prior art date
Application number
AP2011005845A
Other languages
English (en)
Other versions
AP2011005845A0 (en
Inventor
Peng Zhang
Hanbin Shan
Zhedong Yuan
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40878634&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP3048(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Servier Lab filed Critical Servier Lab
Publication of AP2011005845A0 publication Critical patent/AP2011005845A0/xx
Application granted granted Critical
Publication of AP3048A publication Critical patent/AP3048A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C07C233/17—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/18—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C01—INORGANIC CHEMISTRY
    • C01B—NON-METALLIC ELEMENTS; COMPOUNDS THEREOF; METALLOIDS OR COMPOUNDS THEREOF NOT COVERED BY SUBCLASS C01C
    • C01B7/00—Halogens; Halogen acids
    • C01B7/01—Chlorine; Hydrogen chloride
    • C—CHEMISTRY; METALLURGY
    • C01—INORGANIC CHEMISTRY
    • C01B—NON-METALLIC ELEMENTS; COMPOUNDS THEREOF; METALLOIDS OR COMPOUNDS THEREOF NOT COVERED BY SUBCLASS C01C
    • C01B7/00—Halogens; Halogen acids
    • C01B7/09—Bromine; Hydrogen bromide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AP2011005845A 2009-02-27 2010-02-26 Agomelatine hydrohalide complex and preparation method thereof AP3048A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN2009100467821A CN101481321B (zh) 2009-02-27 2009-02-27 阿戈美拉汀卤化氢复合物及其制备方法
PCT/CN2010/070780 WO2010097052A1 (zh) 2009-02-27 2010-02-26 阿戈美拉汀卤化氢复合物及其制备方法

Publications (2)

Publication Number Publication Date
AP2011005845A0 AP2011005845A0 (en) 2011-08-31
AP3048A true AP3048A (en) 2014-11-30

Family

ID=40878634

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2011005845A AP3048A (en) 2009-02-27 2010-02-26 Agomelatine hydrohalide complex and preparation method thereof

Country Status (36)

Country Link
US (1) US8524949B2 (xx)
EP (1) EP2418195B1 (xx)
JP (1) JP5426693B2 (xx)
KR (1) KR101284202B1 (xx)
CN (1) CN101481321B (xx)
AP (1) AP3048A (xx)
AU (1) AU2010217082B2 (xx)
BR (1) BRPI1008767B1 (xx)
CA (1) CA2753449C (xx)
CL (1) CL2011002090A1 (xx)
CO (1) CO6420335A2 (xx)
CR (1) CR20110446A (xx)
CU (1) CU20110163A7 (xx)
CY (1) CY1117100T1 (xx)
DK (1) DK2418195T3 (xx)
EA (1) EA021939B1 (xx)
EC (1) ECSP11011290A (xx)
ES (1) ES2530730T3 (xx)
GE (1) GEP20156221B (xx)
HN (1) HN2011002291A (xx)
HR (1) HRP20150072T1 (xx)
IL (1) IL214682A (xx)
MA (1) MA33063B1 (xx)
MX (1) MX2011008946A (xx)
MY (1) MY154015A (xx)
NI (1) NI201100163A (xx)
NZ (1) NZ594773A (xx)
PE (1) PE20120652A1 (xx)
PL (1) PL2418195T3 (xx)
PT (1) PT2418195E (xx)
RS (1) RS53751B1 (xx)
SG (1) SG173691A1 (xx)
SI (1) SI2418195T1 (xx)
UA (1) UA97619C2 (xx)
WO (1) WO2010097052A1 (xx)
ZA (1) ZA201106048B (xx)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102106806B (zh) * 2009-12-29 2013-04-17 上海中西制药有限公司 一种固体制剂的制备方法及所得固体制剂
CN102190595A (zh) * 2010-03-17 2011-09-21 上海医药工业研究院 阿戈美拉汀溴化氢水合物及其制备方法
CN102190594A (zh) 2010-03-17 2011-09-21 上海医药工业研究院 阿戈美拉汀氯化氢水合物及其制备方法
CN101870662B (zh) * 2010-05-21 2013-03-20 中山大学 结晶型阿戈美拉汀溶剂化物及其制备方法
WO2012046253A2 (en) * 2010-10-08 2012-04-12 Msn Laboratories Limited Process for the preparation of n-[2- (7-methoxy-l-naphthyl) ethyl] acetamide and its novel crystalline forms
EP2517700B1 (en) * 2011-04-28 2013-07-17 Zentiva, k.s. Pharmaceutically acceptable cocrystals of N-[2-(7-methoxy-1-naphthyl]acetamide and methods of their preparation
EP2551257A1 (en) * 2011-07-28 2013-01-30 Laboratorios Del. Dr. Esteve, S.A. Co-crystals of agomelatine with co-crystal-formers
FR2978916B1 (fr) 2011-08-10 2013-07-26 Servier Lab Composition pharmaceutique solide pour administration buccale d'agomelatine
CN102702008B (zh) * 2012-06-03 2014-05-28 上海右手医药科技开发有限公司 阿戈美拉汀硫酸复合物及其制备方法
EP2851363B1 (en) * 2012-05-14 2018-01-03 Shanghai Righthand Pharmtech. Co., Ltd. Agomelatine acid radical composite, and preparation method and application thereof
CN102702041B (zh) * 2012-05-14 2013-08-14 上海右手医药科技开发有限公司 阿戈美拉汀苯磺酸类复合物及其制备方法
CN102718675B (zh) * 2012-06-07 2015-03-25 上海右手医药科技开发有限公司 阿戈美拉汀甲磺酸复合物及其制备方法
ES2590908T3 (es) * 2012-12-17 2016-11-24 Dr. Reddy's Laboratories Ltd. Cocristal de agomelatina con ácido fosfórico
EP2934502A1 (en) 2012-12-21 2015-10-28 Laboratorios Lesvi S.L. Process for prepararing n-(2-(7-methoxy-1-naphthalenyl)ethyl) acetamide and solid forms thereof
FR3001894A1 (fr) 2013-02-08 2014-08-15 Servier Lab Composition pharmaceutique solide pour administration buccale d'agomelatine
ME03741B (me) * 2013-07-29 2021-04-20 Shanghai Inst Pharmaceutical Ind Konpleksi agomelatina i sulfonskih kisjelina, postupak njihove proizvodnje i proizvodnje farmaceutskih pripravaka koji ih sadržavaju
ES2734562T3 (es) * 2013-07-31 2019-12-10 Servier Lab Co-cristales de agomelatina y ácido p-toluensulfónico, su procedimiento de preparación y composiciones farmacéuticas que los contienen

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050182276A1 (en) * 2004-02-13 2005-08-18 Jean-Claude Souvie Process for the synthesis and crystalline form of agomelatine
CN1907958A (zh) * 2005-08-03 2007-02-07 瑟维尔实验室 阿戈美拉汀的新晶形ⅴ、它的制备方法和包含它的药物组合物
EP1752440A1 (en) * 2004-01-15 2007-02-14 Tosoh Corporation Amine compound having fluorene group as framework, process for producing the amine compound, and use of the amine compound

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2658818B1 (fr) * 1990-02-27 1993-12-31 Adir Cie Nouveaux derives a structure naphtalenique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
FR2778662B1 (fr) * 1998-05-12 2000-06-16 Adir Nouveaux composes cycliques substitues, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2795326B1 (fr) * 1999-06-28 2001-08-31 Adir Composition pharmaceutique solide thermoformable a liberation controlee
KR100994169B1 (ko) 2002-05-24 2010-11-15 바이엘 크롭사이언스 아게 티오알킬아민 유도체의 제조방법
FR2899472B1 (fr) * 2006-04-07 2008-09-12 Servier Lab Utilisation de l'agomelatine pour l'obtention de medicaments destines au traitement du trouble anxiete generalisee

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1752440A1 (en) * 2004-01-15 2007-02-14 Tosoh Corporation Amine compound having fluorene group as framework, process for producing the amine compound, and use of the amine compound
US20050182276A1 (en) * 2004-02-13 2005-08-18 Jean-Claude Souvie Process for the synthesis and crystalline form of agomelatine
CN1907958A (zh) * 2005-08-03 2007-02-07 瑟维尔实验室 阿戈美拉汀的新晶形ⅴ、它的制备方法和包含它的药物组合物

Also Published As

Publication number Publication date
EA021939B1 (ru) 2015-10-30
KR20110117721A (ko) 2011-10-27
CN101481321B (zh) 2012-04-18
PT2418195E (pt) 2014-12-26
RS53751B1 (en) 2015-06-30
HRP20150072T1 (xx) 2015-03-13
SG173691A1 (en) 2011-09-29
WO2010097052A1 (zh) 2010-09-02
ZA201106048B (en) 2012-10-31
GEP20156221B (en) 2015-01-26
MA33063B1 (fr) 2012-02-01
BRPI1008767A2 (pt) 2016-06-28
ECSP11011290A (es) 2011-09-30
HN2011002291A (es) 2014-04-07
US20110313198A1 (en) 2011-12-22
CR20110446A (es) 2011-10-18
EP2418195A1 (en) 2012-02-15
CY1117100T1 (el) 2017-04-05
MY154015A (en) 2015-04-30
SI2418195T1 (sl) 2015-03-31
DK2418195T3 (en) 2015-03-02
NI201100163A (es) 2011-12-12
EP2418195B1 (en) 2014-11-19
JP5426693B2 (ja) 2014-02-26
CO6420335A2 (es) 2012-04-16
MX2011008946A (es) 2011-09-27
CA2753449A1 (en) 2010-09-02
AU2010217082B2 (en) 2012-05-03
CU20110163A7 (es) 2012-02-15
UA97619C2 (ru) 2012-02-27
IL214682A (en) 2015-10-29
IL214682A0 (en) 2011-11-30
BRPI1008767B1 (pt) 2021-06-15
AP2011005845A0 (en) 2011-08-31
ES2530730T3 (es) 2015-03-05
PE20120652A1 (es) 2012-06-14
AU2010217082A1 (en) 2011-09-08
CN101481321A (zh) 2009-07-15
EA201101208A1 (ru) 2012-04-30
EP2418195A4 (en) 2013-01-16
JP2012519155A (ja) 2012-08-23
US8524949B2 (en) 2013-09-03
CA2753449C (en) 2014-01-07
PL2418195T3 (pl) 2015-04-30
CL2011002090A1 (es) 2012-02-03
NZ594773A (en) 2013-03-28
KR101284202B1 (ko) 2013-07-09

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