ZA99981B - Oral liquid formulations of benzoxazinones HIV reverse transcriptase inhibitors. - Google Patents

Oral liquid formulations of benzoxazinones HIV reverse transcriptase inhibitors.

Info

Publication number
ZA99981B
ZA99981B ZA9900981A ZA99981A ZA99981B ZA 99981 B ZA99981 B ZA 99981B ZA 9900981 A ZA9900981 A ZA 9900981A ZA 99981 A ZA99981 A ZA 99981A ZA 99981 B ZA99981 B ZA 99981B
Authority
ZA
South Africa
Prior art keywords
benzoxazinones
reverse transcriptase
oral liquid
liquid formulations
transcriptase inhibitors
Prior art date
Application number
ZA9900981A
Other languages
English (en)
Inventor
Surendra M Bahal
Michael B Maurin
Original Assignee
Du Pont Pharm Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont Pharm Co filed Critical Du Pont Pharm Co
Publication of ZA99981B publication Critical patent/ZA99981B/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Virology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA9900981A 1998-02-17 1999-02-08 Oral liquid formulations of benzoxazinones HIV reverse transcriptase inhibitors. ZA99981B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7488198P 1998-02-17 1998-02-17

Publications (1)

Publication Number Publication Date
ZA99981B true ZA99981B (en) 2000-08-08

Family

ID=22122226

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA9900981A ZA99981B (en) 1998-02-17 1999-02-08 Oral liquid formulations of benzoxazinones HIV reverse transcriptase inhibitors.

Country Status (19)

Country Link
US (1) US6235733B1 (de)
EP (1) EP1054674B1 (de)
JP (1) JP2002502878A (de)
CN (1) CN1170541C (de)
AR (1) AR018092A1 (de)
AT (1) ATE345802T1 (de)
AU (1) AU745008C (de)
BR (2) BRPI9908132B8 (de)
CA (1) CA2319609C (de)
DE (1) DE69934097T2 (de)
ES (1) ES2277429T3 (de)
HK (1) HK1030749A1 (de)
HR (1) HRP990049A2 (de)
IL (1) IL137763A0 (de)
MY (1) MY139034A (de)
NZ (1) NZ506579A (de)
TW (1) TW528596B (de)
WO (1) WO1999040921A2 (de)
ZA (1) ZA99981B (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3525792A4 (de) * 2016-10-11 2020-04-22 Aucta Pharmaceuticals Pulver für orale suspensionen mit lamotrigin

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0484281B2 (de) * 1990-11-02 2000-11-22 Novartis AG Zyklosporine
US5494936A (en) * 1992-04-27 1996-02-27 Vyrex Corporation Delivery formulation for probucol
US5665720A (en) 1992-08-07 1997-09-09 Merck & Co., Inc. Benzoxazinones as inhibitors of HIV reverse transcriptase
WO1995020389A1 (en) 1994-01-28 1995-08-03 Merck & Co., Inc. Benzoxazinones as inhibitors of hiv reverse transcriptase
WO1997040833A1 (en) 1996-05-02 1997-11-06 Merck & Co., Inc. Hiv protease inhibitors useful for the treatment of aids
CA2268953A1 (en) * 1996-10-02 1998-04-09 Du Pont Pharmaceuticals Company 4,4-disubstituted-1,4-dihydro-2h-3,1-benzoxazin-2-ones useful as hiv reverse transcriptase inhibitors and intermediates and processes for making the same

Also Published As

Publication number Publication date
JP2002502878A (ja) 2002-01-29
ES2277429T3 (es) 2007-07-01
BRPI9908132B1 (pt) 2015-07-14
ATE345802T1 (de) 2006-12-15
WO1999040921A2 (en) 1999-08-19
AU745008B2 (en) 2002-03-07
BRPI9908132B8 (pt) 2016-11-16
CA2319609A1 (en) 1999-08-19
EP1054674B1 (de) 2006-11-22
NZ506579A (en) 2002-11-26
HRP990049A2 (en) 1999-12-31
AU2682799A (en) 1999-08-30
IL137763A0 (en) 2001-10-31
HK1030749A1 (en) 2001-05-18
WO1999040921A3 (en) 1999-11-04
AU745008C (en) 2003-03-27
DE69934097T2 (de) 2007-06-28
DE69934097D1 (de) 2007-01-04
CA2319609C (en) 2007-09-18
BRPI9908132C1 (pt) 2021-05-25
BR9908132A (pt) 2000-12-05
CN1170541C (zh) 2004-10-13
US6235733B1 (en) 2001-05-22
AR018092A1 (es) 2001-10-31
MY139034A (en) 2009-08-28
EP1054674A2 (de) 2000-11-29
TW528596B (en) 2003-04-21
CN1291098A (zh) 2001-04-11

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