ZA972199B - Novel bridged cyclic amino acids as pharmaceutical agents. - Google Patents

Novel bridged cyclic amino acids as pharmaceutical agents.

Info

Publication number
ZA972199B
ZA972199B ZA9702199A ZA972199A ZA972199B ZA 972199 B ZA972199 B ZA 972199B ZA 9702199 A ZA9702199 A ZA 9702199A ZA 972199 A ZA972199 A ZA 972199A ZA 972199 B ZA972199 B ZA 972199B
Authority
ZA
South Africa
Prior art keywords
amino acids
pct
cyclic amino
pharmaceutical agents
bridged cyclic
Prior art date
Application number
ZA9702199A
Other languages
English (en)
Inventor
David Christopher Horwell
Clare O Keen
Giles S Ratcliffe
Justin S Bryans
Andrew I Morrell
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of ZA972199B publication Critical patent/ZA972199B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/28—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and containing rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A61P25/12—Antiepileptics; Anticonvulsants for grand-mal
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/36—Systems containing two condensed rings the rings having more than two atoms in common
    • C07C2602/42—Systems containing two condensed rings the rings having more than two atoms in common the bicyclo ring system containing seven carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/36—Systems containing two condensed rings the rings having more than two atoms in common
    • C07C2602/46—Systems containing two condensed rings the rings having more than two atoms in common the bicyclo ring system containing nine carbon atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
ZA9702199A 1996-03-14 1997-03-13 Novel bridged cyclic amino acids as pharmaceutical agents. ZA972199B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1343396P 1996-03-14 1996-03-14

Publications (1)

Publication Number Publication Date
ZA972199B true ZA972199B (en) 1997-09-17

Family

ID=21759944

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA9702199A ZA972199B (en) 1996-03-14 1997-03-13 Novel bridged cyclic amino acids as pharmaceutical agents.

Country Status (18)

Country Link
US (1) US6020370A (ru)
EP (1) EP0888285B1 (ru)
JP (1) JP2000506862A (ru)
KR (1) KR100487032B1 (ru)
AT (1) ATE210629T1 (ru)
AU (1) AU731279B2 (ru)
BR (1) BR9708180A (ru)
CZ (1) CZ287598A3 (ru)
DE (1) DE69709070T2 (ru)
EA (1) EA001214B1 (ru)
ES (1) ES2169848T3 (ru)
IL (1) IL125364A0 (ru)
NO (1) NO984204D0 (ru)
NZ (1) NZ331142A (ru)
PL (1) PL185990B1 (ru)
SK (1) SK282848B6 (ru)
WO (1) WO1997033859A1 (ru)
ZA (1) ZA972199B (ru)

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US7141606B2 (en) * 2000-06-26 2006-11-28 Warner-Lambert Company Gabapentin analogues for sleep disorders
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GB2374595A (en) * 2001-04-19 2002-10-23 Warner Lambert Co Fused bicyclic or tricyclic amino acids
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Also Published As

Publication number Publication date
WO1997033859A1 (en) 1997-09-18
EP0888285A1 (en) 1999-01-07
NZ331142A (en) 2001-04-27
SK282848B6 (sk) 2002-12-03
ATE210629T1 (de) 2001-12-15
PL328800A1 (en) 1999-02-15
NO984204L (no) 1998-09-11
AU731279B2 (en) 2001-03-29
JP2000506862A (ja) 2000-06-06
BR9708180A (pt) 1999-07-27
KR100487032B1 (ko) 2005-12-21
SK124898A3 (en) 1999-02-11
PL185990B1 (pl) 2003-09-30
CZ287598A3 (cs) 1999-02-17
EP0888285B1 (en) 2001-12-12
IL125364A0 (en) 1999-03-12
DE69709070D1 (de) 2002-01-24
DE69709070T2 (de) 2002-06-20
AU2127197A (en) 1997-10-01
US6020370A (en) 2000-02-01
EA001214B1 (ru) 2000-12-25
KR19990087755A (ko) 1999-12-27
EA199800797A1 (ru) 1999-04-29
NO984204D0 (no) 1998-09-11
ES2169848T3 (es) 2002-07-16

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