ZA968661B - Oxazolidinone antibacterial agent with tricyclic substituents. - Google Patents
Oxazolidinone antibacterial agent with tricyclic substituents.Info
- Publication number
- ZA968661B ZA968661B ZA9608661A ZA968661A ZA968661B ZA 968661 B ZA968661 B ZA 968661B ZA 9608661 A ZA9608661 A ZA 9608661A ZA 968661 A ZA968661 A ZA 968661A ZA 968661 B ZA968661 B ZA 968661B
- Authority
- ZA
- South Africa
- Prior art keywords
- antibacterial agent
- oxazolidinone antibacterial
- organisms
- tricyclic substituents
- tricyclic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US737195P | 1995-11-17 | 1995-11-17 |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA968661B true ZA968661B (en) | 1998-04-14 |
Family
ID=21725778
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA9608661A ZA968661B (en) | 1995-11-17 | 1996-10-14 | Oxazolidinone antibacterial agent with tricyclic substituents. |
Country Status (12)
Country | Link |
---|---|
US (2) | US5922707A (xx) |
EP (1) | EP0874852B1 (xx) |
JP (1) | JP2000500489A (xx) |
AT (1) | ATE263172T1 (xx) |
AU (1) | AU7665196A (xx) |
DE (1) | DE69632074T2 (xx) |
DK (1) | DK0874852T3 (xx) |
ES (1) | ES2217329T3 (xx) |
PT (1) | PT874852E (xx) |
TW (1) | TW426683B (xx) |
WO (1) | WO1997019089A1 (xx) |
ZA (1) | ZA968661B (xx) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZA968661B (en) * | 1995-11-17 | 1998-04-14 | Upjohn Co | Oxazolidinone antibacterial agent with tricyclic substituents. |
GB9601666D0 (en) * | 1996-01-27 | 1996-03-27 | Zeneca Ltd | Chemical compounds |
GB9702213D0 (en) | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
GB9609919D0 (en) * | 1996-05-11 | 1996-07-17 | Zeneca Ltd | Chemical compounds |
ID23803A (id) * | 1997-08-15 | 2000-05-11 | Pfizer Prod Inc | Turunan-turunan 2-(4-aril atau heteroaril-piperazin-1-ilmetil)-1h-indola |
GB9717804D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
GB9717807D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
GB9725244D0 (en) | 1997-11-29 | 1998-01-28 | Zeneca Ltd | Chemical compounds |
DE19802239A1 (de) * | 1998-01-22 | 1999-07-29 | Bayer Ag | Neue mit Bicyclen substituierte Oxazolidinone |
DE19802235A1 (de) * | 1998-01-22 | 1999-07-29 | Bayer Ag | Mit tricyclischen Indolen substituierte Oxazolidinone |
US7002020B1 (en) | 1998-01-23 | 2006-02-21 | Pharmacia & Upjohn Company | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
EP1049682A1 (en) | 1998-01-23 | 2000-11-08 | Versicor, Inc. | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
US6562844B2 (en) | 1998-01-23 | 2003-05-13 | Pharmacia & Upjohn Company | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
DE19805117A1 (de) * | 1998-02-09 | 1999-08-12 | Bayer Ag | Neue Oxazolidinone mit azolhaltigen Tricyclen |
TR200003595T2 (tr) * | 1998-06-05 | 2001-07-23 | Astrazeneca Ab | Kimyasal bileşikler |
MY122454A (en) * | 1998-06-05 | 2006-04-29 | Upjohn Co | Use of oxazolidinones for the preparation of a medicament for transdermal delivery |
ES2300151T3 (es) | 1998-09-22 | 2008-06-01 | Astellas Pharma Inc. | Derivados de cianofenilo. |
JP2002535680A (ja) | 1999-01-27 | 2002-10-22 | ファルマシア・アンド・アップジョン・カンパニー | 延長因子p活性モジュレーターのアッセイ方法 |
JP2003501351A (ja) * | 1999-05-27 | 2003-01-14 | ファルマシア・アンド・アップジョン・カンパニー | 抗菌剤としての二環系オキサゾリジノン |
GB9928568D0 (en) | 1999-12-03 | 2000-02-02 | Zeneca Ltd | Chemical compounds |
GB0009803D0 (en) * | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
EP1539745B1 (en) | 2002-08-12 | 2006-03-29 | Pharmacia & Upjohn Company LLC | N-aryl-2-oxazolidinones and their derivatives |
BR0316483A (pt) | 2002-11-21 | 2005-10-11 | Upjohn Co | Derivados de n-(4-(piperazin-1-il)-fenil-2-oxazolidinona-5-carboxami da e compostos relacionados como agentes antibacterianos |
EP1594865A2 (en) * | 2003-02-07 | 2005-11-16 | Warner-Lambert Company LLC | Antibacterial agents |
US7795267B2 (en) * | 2003-08-29 | 2010-09-14 | Takeda Pharmaceutical Company Limited | Bicyclic piperazine compound having TGR23 antagonistic activity |
AR057828A1 (es) * | 2005-09-29 | 2007-12-19 | Astrazeneca Ab | Compuestos derivados de azetidina, su preparacion y composicion farmaceuutica |
WO2007087250A2 (en) | 2006-01-23 | 2007-08-02 | Amira Pharmaceuticals, Inc. | Tricyclic inhibitors of 5-lipoxygenase |
CN110734454B (zh) * | 2016-12-12 | 2021-08-17 | 石药集团中奇制药技术(石家庄)有限公司 | 一类含有三环杂芳基的化合物 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3883522A (en) * | 1974-02-11 | 1975-05-13 | Riker Laboratories Inc | Substituted pyrido(1,2,3-de)-1,4-benzoxazines |
US4080499A (en) * | 1976-12-20 | 1978-03-21 | 1 | Substituted 7,8-dihydro-6H-(1,2,5)thiadiazolo(3',4'-5,6)pyrazino(2,3-b)(1,4)oxazines |
US5039690A (en) * | 1987-10-09 | 1991-08-13 | Du Pont Merck Pharmaceutical Company | Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents |
DE68929303T2 (de) * | 1988-09-15 | 2002-05-02 | Pharmacia & Upjohn Co., Kalamazoo | 3-(Stickstoff substituierte)phenyl-5-beta-amidomethyloxazoliden-2-one |
US5225565A (en) * | 1988-09-15 | 1993-07-06 | The Upjohn Company | Antibacterial 3-(fused-ring substituted)phenyl-5β-amidomethyloxazolidin-2-ones |
ES2177539T3 (es) * | 1992-02-13 | 2002-12-16 | Upjohn Co | Benzoxacinas 4-oxo- y 4h-imidazo(5,1-c)(1,4) utilez como agentes de union de receptores de benzodiacepina. |
SK283420B6 (sk) * | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
US5668286A (en) * | 1994-03-15 | 1997-09-16 | Pharmacia & Upjohn Company | Oxazolidinone derivatives and pharmaceutical compositions containing them |
ES2193201T3 (es) * | 1994-11-15 | 2003-11-01 | Upjohn Co | Agentes antibacterianos tipo oxazolidonas sustituidas con oxazina y tiazina biciclica. |
ZA968661B (en) * | 1995-11-17 | 1998-04-14 | Upjohn Co | Oxazolidinone antibacterial agent with tricyclic substituents. |
-
1996
- 1996-10-14 ZA ZA9608661A patent/ZA968661B/xx unknown
- 1996-11-05 DE DE69632074T patent/DE69632074T2/de not_active Expired - Fee Related
- 1996-11-05 EP EP96939496A patent/EP0874852B1/en not_active Expired - Lifetime
- 1996-11-05 DK DK96939496T patent/DK0874852T3/da active
- 1996-11-05 AU AU76651/96A patent/AU7665196A/en not_active Abandoned
- 1996-11-05 ES ES96939496T patent/ES2217329T3/es not_active Expired - Lifetime
- 1996-11-05 PT PT96939496T patent/PT874852E/pt unknown
- 1996-11-05 WO PCT/US1996/017120 patent/WO1997019089A1/en active IP Right Grant
- 1996-11-05 AT AT96939496T patent/ATE263172T1/de not_active IP Right Cessation
- 1996-11-05 JP JP9519726A patent/JP2000500489A/ja not_active Withdrawn
- 1996-11-15 TW TW085114048A patent/TW426683B/zh not_active IP Right Cessation
-
1997
- 1997-05-02 US US08/850,424 patent/US5922707A/en not_active Expired - Fee Related
-
1999
- 1999-02-15 US US09/250,382 patent/US5955460A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
DE69632074T2 (de) | 2005-01-20 |
TW426683B (en) | 2001-03-21 |
US5922707A (en) | 1999-07-13 |
DE69632074D1 (de) | 2004-05-06 |
US5955460A (en) | 1999-09-21 |
WO1997019089A1 (en) | 1997-05-29 |
PT874852E (pt) | 2004-08-31 |
AU7665196A (en) | 1997-06-11 |
EP0874852B1 (en) | 2004-03-31 |
ES2217329T3 (es) | 2004-11-01 |
DK0874852T3 (da) | 2004-06-07 |
ATE263172T1 (de) | 2004-04-15 |
EP0874852A1 (en) | 1998-11-04 |
JP2000500489A (ja) | 2000-01-18 |
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