ZA921005B - Imidazopyridine PAF/H 1 antagonists. - Google Patents

Imidazopyridine PAF/H 1 antagonists.

Info

Publication number
ZA921005B
ZA921005B ZA921005A ZA921005A ZA921005B ZA 921005 B ZA921005 B ZA 921005B ZA 921005 A ZA921005 A ZA 921005A ZA 921005 A ZA921005 A ZA 921005A ZA 921005 B ZA921005 B ZA 921005B
Authority
ZA
South Africa
Prior art keywords
pct
paf
antagonists
sec
imidazopyridine
Prior art date
Application number
ZA921005A
Other languages
English (en)
Inventor
David Alker
Robert John Bass
Kelvin Cooper
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of ZA921005B publication Critical patent/ZA921005B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cosmetics (AREA)
  • Steroid Compounds (AREA)
  • Prostheses (AREA)
ZA921005A 1991-02-13 1992-02-12 Imidazopyridine PAF/H 1 antagonists. ZA921005B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB919102997A GB9102997D0 (en) 1991-02-13 1991-02-13 Therapeutic agents

Publications (1)

Publication Number Publication Date
ZA921005B true ZA921005B (en) 1993-08-12

Family

ID=10689943

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA921005A ZA921005B (en) 1991-02-13 1992-02-12 Imidazopyridine PAF/H 1 antagonists.

Country Status (29)

Country Link
US (1) US5358953A (cs)
EP (1) EP0572425B1 (cs)
JP (1) JP2506541B2 (cs)
KR (1) KR970005302B1 (cs)
CN (1) CN1040326C (cs)
AT (1) ATE109482T1 (cs)
AU (1) AU650322B2 (cs)
BR (1) BR9205615A (cs)
CA (1) CA2099381C (cs)
CZ (1) CZ280504B6 (cs)
DE (1) DE69200304T2 (cs)
DK (1) DK0572425T3 (cs)
EG (1) EG20085A (cs)
ES (1) ES2059212T3 (cs)
FI (1) FI933531A0 (cs)
GB (1) GB9102997D0 (cs)
HU (2) HUT65947A (cs)
IE (1) IE65125B1 (cs)
IL (1) IL100887A (cs)
MX (1) MX9200589A (cs)
MY (1) MY108437A (cs)
NO (1) NO300592B1 (cs)
NZ (1) NZ241597A (cs)
PL (1) PL169304B1 (cs)
RU (1) RU2114845C1 (cs)
TW (1) TW227000B (cs)
WO (1) WO1992014734A1 (cs)
YU (1) YU48238B (cs)
ZA (1) ZA921005B (cs)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2042421B1 (es) * 1992-05-22 1994-08-01 Uriach & Cia Sa J Procedimiento para la obtencion de la 8-cloro-11-*1-*(5-metil-3-piridil)metil*-4-piperidiliden*-6,11-dihidro-5h-benzo*5,6*ciclohepta*1,2-b*piridina.
WO1996005201A1 (en) * 1994-08-10 1996-02-22 British Biotech Pharmaceuticals Limited Imidazopyridine derivatives as dual histamine (h1) and platelet activating factor (paf) antagonists
ES2087038B1 (es) * 1994-11-07 1997-03-16 Uriach & Cia Sa J Nuevas piperidinas con actividad antagonista del paf.
WO1997006167A1 (en) * 1995-08-05 1997-02-20 British Biotech Pharmaceuticals Limited Imidazopyridine derivatives
US5567711A (en) * 1995-04-19 1996-10-22 Abbott Laboratories Indole-3-carbonyl and indole-3-sulfonyl derivatives as platelet activating factor antagonists
GB9508748D0 (en) * 1995-04-28 1995-06-14 British Biotech Pharm Benzimidazole derivatives
SE9801526D0 (sv) * 1998-04-29 1998-04-29 Astra Ab New compounds
CA2774959C (en) 2000-08-04 2016-05-31 Dmi Biosciences, Inc. Method of using diketopiperazines and composition containing them
CN103191410B (zh) 2003-05-15 2015-03-04 安皮奥制药股份有限公司 T-细胞介导的疾病的治疗
US7687515B2 (en) * 2006-01-17 2010-03-30 N.V. Organon 6-phenyl-1H-imidazo[4,5-c]pyridine-4-carbonitrile derivatives
ES2527588T3 (es) 2008-01-30 2015-01-27 Nippon Zoki Pharmaceutical Co., Ltd. Derivado de piperidina
EP2300011A4 (en) 2008-05-27 2012-06-20 Dmi Life Sciences Inc THERAPEUTIC PROCESSES AND COMPOUNDS
EP2727919B1 (en) * 2011-06-28 2019-05-08 Fujian Mindong Rejuvenation Pharmaceutical Co., Ltd. Benzocycloheptanethiophene derivatives for anti-allergic reactions
EP2766029B1 (en) 2011-10-10 2020-03-25 Ampio Pharmaceuticals, Inc. Treatment of degenerative joint disease
CN103841934A (zh) 2011-10-10 2014-06-04 安皮奥制药股份有限公司 增强免疫耐受的可植入的医疗装置及其制造与植入方法
PH12014500715A1 (en) * 2011-10-28 2014-05-12 Ampio Pharmaceuticals Inc Treatment of rhinitis
SG10201707619RA (en) 2013-03-15 2017-10-30 Ampio Pharmaceuticals Inc Compositions for the mobilization, homing, expansion and differentiation of stem cells and methods of using the same
KR20170045274A (ko) 2014-08-18 2017-04-26 앰피오 파마슈티컬스 인코퍼레이티드 관절 징후의 치료
EP3310375A4 (en) 2015-06-22 2019-02-20 Ampio Pharmaceuticals, Inc. USE OF LOW-MOLECULAR FRACTIONS OF HUMAN SERUMALBUMINE IN THE TREATMENT OF ILLNESSES

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL132137C (cs) * 1963-04-24
WO1989008653A1 (en) * 1988-03-15 1989-09-21 G.D. Searle & Co. 1H/3H-[4-(N,N-DICYCLOALKYL/BRANCHED-ALKYLCARBOXAMIDO)-BENZYL]IMIDAZO[4,5-c]PYRIDINES AS PAF ANTAGONISTS
MY106964A (en) * 1988-04-28 1995-08-30 Schering Corp Fused polycyclic compounds, compositions, methods of manufacture, and their use as paf antagonists, antihistamines and/or antiinflammatory agents.
US5250681A (en) * 1988-06-02 1993-10-05 Ajinomoto Co., Inc. Piperidine derivatives and hypotensives containing the same
US5114919A (en) * 1990-02-26 1992-05-19 Merck & Co., Inc. Adjuncts in cancer chemotherapy
DE69104481T2 (de) * 1990-05-09 1995-02-09 Pfizer Imidazo[4,5-c]pyridine als paf antagonisten.

Also Published As

Publication number Publication date
AU650322B2 (en) 1994-06-16
YU48238B (sh) 1997-08-22
ATE109482T1 (de) 1994-08-15
CN1040326C (zh) 1998-10-21
KR970005302B1 (ko) 1997-04-15
IE920449A1 (en) 1992-08-12
DE69200304D1 (de) 1994-09-08
CA2099381C (en) 1996-07-09
NZ241597A (en) 1993-04-28
IE65125B1 (en) 1995-10-04
FI933531A7 (fi) 1993-08-10
NO932889D0 (no) 1993-08-13
NO300592B1 (no) 1997-06-23
EG20085A (en) 1997-05-31
CN1064275A (zh) 1992-09-09
GB9102997D0 (en) 1991-03-27
YU14392A (sh) 1994-11-15
CS42592A3 (en) 1992-09-16
JPH06504992A (ja) 1994-06-09
WO1992014734A1 (en) 1992-09-03
JP2506541B2 (ja) 1996-06-12
DK0572425T3 (da) 1994-09-12
TW227000B (cs) 1994-07-21
FI933531L (fi) 1993-08-10
AU1168392A (en) 1992-09-15
CA2099381A1 (en) 1992-08-14
DE69200304T2 (de) 1994-12-08
HU211202A9 (en) 1995-11-28
HUT65947A (en) 1994-08-29
MY108437A (en) 1996-09-30
MX9200589A (es) 1992-10-01
NO932889L (no) 1993-08-13
EP0572425B1 (en) 1994-08-03
US5358953A (en) 1994-10-25
IL100887A (en) 1996-01-19
RU2114845C1 (ru) 1998-07-10
CZ280504B6 (cs) 1996-02-14
EP0572425A1 (en) 1993-12-08
PL169304B1 (pl) 1996-06-28
BR9205615A (pt) 1994-05-17
FI933531A0 (fi) 1993-08-10
HU9302327D0 (en) 1993-10-28
ES2059212T3 (es) 1994-11-01
IL100887A0 (en) 1992-11-15

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