ZA908267B - 5-(2-((2-amino-2-oxoethyl)(methyl)amino)ethyl)-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5(5h)-benzothiazepin-4-one derivatives,their preparation and their application in therapy - Google Patents
5-(2-((2-amino-2-oxoethyl)(methyl)amino)ethyl)-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5(5h)-benzothiazepin-4-one derivatives,their preparation and their application in therapyInfo
- Publication number
- ZA908267B ZA908267B ZA908267A ZA908267A ZA908267B ZA 908267 B ZA908267 B ZA 908267B ZA 908267 A ZA908267 A ZA 908267A ZA 908267 A ZA908267 A ZA 908267A ZA 908267 B ZA908267 B ZA 908267B
- Authority
- ZA
- South Africa
- Prior art keywords
- amino
- benzothiazepin
- oxoethyl
- methoxyphenyl
- dihydro
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D281/02—Seven-membered rings
- C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D281/02—Seven-membered rings
- C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8913540A FR2653122B1 (fr) | 1989-10-17 | 1989-10-17 | Derives de 5-[2-[[2-amino-2-oxoethyl]methylamino]ethyl]-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5(5h)-benzothiazepine-4-one, leur preparation et leur application en therapeutique. |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA908267B true ZA908267B (en) | 1991-08-28 |
Family
ID=9386468
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA908267A ZA908267B (en) | 1989-10-17 | 1990-10-16 | 5-(2-((2-amino-2-oxoethyl)(methyl)amino)ethyl)-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5(5h)-benzothiazepin-4-one derivatives,their preparation and their application in therapy |
Country Status (14)
Country | Link |
---|---|
EP (1) | EP0424214A1 (xx) |
JP (1) | JPH03133970A (xx) |
KR (1) | KR910007901A (xx) |
AU (1) | AU6479690A (xx) |
CA (1) | CA2027738A1 (xx) |
FI (1) | FI905089A0 (xx) |
FR (1) | FR2653122B1 (xx) |
HU (1) | HUT57754A (xx) |
IE (1) | IE903720A1 (xx) |
IL (1) | IL95931A0 (xx) |
NO (1) | NO904470L (xx) |
NZ (1) | NZ235717A (xx) |
PT (1) | PT95606A (xx) |
ZA (1) | ZA908267B (xx) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69411387T2 (de) * | 1994-09-16 | 1999-02-25 | Orion Corp. FERMION, Espoo | Verfahren zur Herstellung von pharmazeutisch aktiven Benzothiazepinderivaten. |
WO2005035505A2 (en) * | 2003-09-30 | 2005-04-21 | Artesian Therapeutics, Inc. | Compounds with phosphodiesterase inhibiting and calcium channel blocking activities |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH538492A (de) * | 1970-10-07 | 1973-06-30 | Hoffmann La Roche | Verfahren zur Herstellung von Benzodiazepin-Derivaten |
FR2624117B1 (fr) * | 1987-12-08 | 1991-02-22 | Synthelabo | Derives de hydroxy-3 (methoxy-4 phenyl)-2 (methylamino-2 ethyl)-5 dihydro-2,3 5h-benzothiazepine-1,5 one-4, leur preparation et leur application en therapeutique |
FR2630109B1 (fr) * | 1988-04-19 | 1991-11-29 | Synthelabo | Derives de ((n-(amino-2 oxo-2 ethyl)methylamino)-2 ethyl)-5 hydroxy-3 (methoxy-4 phenyl)-2 dihydro-2,3 5h-benzothiazepine-1,5 one-4, leur preparation et leur application en therapeutique |
-
1989
- 1989-10-17 FR FR8913540A patent/FR2653122B1/fr not_active Expired - Fee Related
-
1990
- 1990-10-10 EP EP90402820A patent/EP0424214A1/fr not_active Withdrawn
- 1990-10-16 NZ NZ235717A patent/NZ235717A/xx unknown
- 1990-10-16 IE IE372090A patent/IE903720A1/en unknown
- 1990-10-16 JP JP2278828A patent/JPH03133970A/ja active Pending
- 1990-10-16 KR KR1019900016471A patent/KR910007901A/ko not_active Application Discontinuation
- 1990-10-16 ZA ZA908267A patent/ZA908267B/xx unknown
- 1990-10-16 PT PT95606A patent/PT95606A/pt not_active Application Discontinuation
- 1990-10-16 IL IL95931A patent/IL95931A0/xx unknown
- 1990-10-16 CA CA002027738A patent/CA2027738A1/en not_active Abandoned
- 1990-10-16 NO NO90904470A patent/NO904470L/no unknown
- 1990-10-16 HU HU906466A patent/HUT57754A/hu unknown
- 1990-10-16 AU AU64796/90A patent/AU6479690A/en not_active Abandoned
- 1990-10-16 FI FI905089A patent/FI905089A0/fi not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
IL95931A0 (en) | 1991-07-18 |
NO904470L (no) | 1991-04-18 |
NO904470D0 (no) | 1990-10-16 |
FR2653122A1 (fr) | 1991-04-19 |
JPH03133970A (ja) | 1991-06-07 |
HUT57754A (en) | 1991-12-30 |
EP0424214A1 (fr) | 1991-04-24 |
AU6479690A (en) | 1991-07-11 |
CA2027738A1 (en) | 1991-04-18 |
HU906466D0 (en) | 1991-04-29 |
FR2653122B1 (fr) | 1994-04-15 |
FI905089A0 (fi) | 1990-10-16 |
PT95606A (pt) | 1991-09-13 |
IE903720A1 (en) | 1991-04-24 |
NZ235717A (en) | 1991-12-23 |
KR910007901A (ko) | 1991-05-30 |
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