ZA906810B - Heterogeneous synthesis of azepinones from esters - Google Patents

Heterogeneous synthesis of azepinones from esters

Info

Publication number
ZA906810B
ZA906810B ZA906810A ZA906810A ZA906810B ZA 906810 B ZA906810 B ZA 906810B ZA 906810 A ZA906810 A ZA 906810A ZA 906810 A ZA906810 A ZA 906810A ZA 906810 B ZA906810 B ZA 906810B
Authority
ZA
South Africa
Prior art keywords
cyclized
methoxyphenyl
hydroxy
amino
acid
Prior art date
Application number
ZA906810A
Other languages
English (en)
Inventor
Daniel Eugene Martin
Eugene Martin Daniel
Original Assignee
Marion Merrell Dow Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Marion Merrell Dow Inc filed Critical Marion Merrell Dow Inc
Publication of ZA906810B publication Critical patent/ZA906810B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ZA906810A 1989-08-31 1990-08-27 Heterogeneous synthesis of azepinones from esters ZA906810B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US40065889A 1989-08-31 1989-08-31

Publications (1)

Publication Number Publication Date
ZA906810B true ZA906810B (en) 1991-10-30

Family

ID=23584491

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA906810A ZA906810B (en) 1989-08-31 1990-08-27 Heterogeneous synthesis of azepinones from esters

Country Status (13)

Country Link
EP (1) EP0415384B1 (ko)
JP (1) JP3090212B2 (ko)
KR (1) KR0163585B1 (ko)
AT (1) ATE150459T1 (ko)
AU (1) AU628217B2 (ko)
CA (1) CA2024124C (ko)
DD (1) DD295367A5 (ko)
DE (1) DE69030222T2 (ko)
ES (1) ES2101682T3 (ko)
HU (1) HU206103B (ko)
IE (1) IE903151A1 (ko)
IL (1) IL95509A (ko)
ZA (1) ZA906810B (ko)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1249318B (it) * 1991-05-23 1995-02-22 Zambon Spa Processo per la preparazione di benzotiazepine per ciclizzazione con acidi fosfonici
DE4313413A1 (de) * 1993-04-23 1994-10-27 Basf Ag 3-(Het)aryloxy(thio)-Carbonsäurederivate, Verfahren und Zwischenprodukte zu ihrer Herstellung

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4567175A (en) * 1983-06-03 1986-01-28 Tanabe Seiyaku Co., Ltd. 8-Chloro-1,5-benzothiazepine derivatives
ZA893392B (en) * 1988-05-24 1990-01-31 Hoffmann La Roche Process for the manufacture of optically active naphthothiazepinones
ATE116643T1 (de) * 1989-04-28 1995-01-15 Tanabe Seiyaku Co Verfahren zur herstellung von 1,5- benzothiazepinderivaten.
JPH0798813B2 (ja) * 1989-04-28 1995-10-25 田辺製薬株式会社 １，５―ベンゾチアゼピン誘導体の製法

Also Published As

Publication number Publication date
IL95509A0 (en) 1991-06-30
EP0415384A3 (en) 1992-04-15
KR910004584A (ko) 1991-03-29
DE69030222T2 (de) 1997-10-16
IL95509A (en) 1994-10-07
EP0415384B1 (en) 1997-03-19
HU905508D0 (en) 1991-02-28
IE903151A1 (en) 1991-03-27
KR0163585B1 (ko) 1998-12-01
CA2024124A1 (en) 1991-03-01
CA2024124C (en) 2003-04-15
AU628217B2 (en) 1992-09-10
JP3090212B2 (ja) 2000-09-18
ATE150459T1 (de) 1997-04-15
DE69030222D1 (de) 1997-04-24
JPH0393778A (ja) 1991-04-18
HUT59118A (en) 1992-04-28
HU206103B (en) 1992-08-28
AU6138290A (en) 1991-03-07
DD295367A5 (de) 1991-10-31
ES2101682T3 (es) 1997-07-16
EP0415384A2 (en) 1991-03-06

Similar Documents

Publication Publication Date Title
HU896131D0 (en) Process for the preparation of 2-[2-[4-/(4-chlorophenyl)phenylmethyl/-1-pyperazinyl]ethoxy]-ethoxi]-acetic acid and its salts
PT81942B (pt) Processo para a preparacao de uma racao alimentar para animais contendo caseina iodada
IL75812A (en) Process for the preparation of halogenated quinolone-carboxylic acids,and 7-chloro-1-cyclopropyl 1,4-dihydro-4-oxo-3-quinoline-carboxylic acid nitrile intermediates therefor
AU628217B2 (en) Heterogeneous synthesis of azepinones from esters
NZ221524A (en) Enzymatic built aqueous liquid detergent with protein stabiliser
ZA858372B (en) Aqueous systems containing amino sulfonic acid derivatives of carboxylic acids
PH20699A (en) Salts of 2-keto-2h-1,2-benzisothiazole 1,1-dioxide as microbicides
PT90584A (pt) Processo de preparacao de agentes diureticos de glutaramidas enantiomericas
FR2693473B1 (fr) Procédé de préparation enzymatique d'hydrolysats de matières protéiques.
GR3032027T3 (en) Process for the preparation of 1,5-benzothiazepines by ring closure of amino esters.
DE3874900D1 (de) Wirkstoff mit die nierenfunktion verbesserndem und diuretischem effekt und verwendung eines darin enthaltenen benzothiazepin-derivates.
CA2030866A1 (en) Process for the preparation of an intermediate of diltiazem
PT92735A (pt) Processo para a preparacao de uma composicao oral antiplaca antibacteriana contendo um novo copolimero de acidos estireno-fosfonicos
ATE48616T1 (de) Analoge von hypokalzemischen polypeptiden, welche den kalziumgehalt des koerpers schonen, deren herstellung, deren verwendung als arznei und diese enthaltende zusammensetzungen.
IT8620997A0 (it) Processo per la preparazione dipirido benzotiazine ad attivita'antibatterica e loro sali con acidi solfonici.
PT95100A (pt) Processo para a preparacao de n-hidroxi-di-benz/b,e/oxepin-alquilaminas e de analogos heterociclicos relacionados com amidas de acidos alcanoicos e de composicoes farmaceuticas que os contem
ES2059020T3 (es) Procedimiento para preparar derivados de 1,5-benzotiazepina.
FI93010B (fi) Menetelmä 1,5-bentsotiatsepiinijohdannaisten valmistamiseksi
FR2577220B1 (fr) Procede d'acetoacetylation de composes aromatiques
FR2589151B1 (fr) Procede de preparation d'esters du diethyleneglycol
BR8601844A (pt) Processo para preparacao de cristais de acrilamida a partir de uma solucao aquosa de acrilamida
PT90618A (pt) Processo para a preparacao de uma tinta anti-vegetativa marinha
IT8619806A0 (it) Processo per la preparazione della n-[2-[[(5-[(dimetilammino)metil]-2furanil)metil] tio] etil-2-nitro-1metiltio-1-etanammina
PT79931A (en) Process for the preparation of 3-amino-2,3,4,5-tetra hydro-1,5-benzothiazepine derivatives and pharmaceutical compossitions therewith
CS380788A1 (en) Method of optically pure erythro-/+/-3-/2-aminophenylthio/-2-hydroxy-3-/4-methoxyphenyl/propanoic acid's production by means of racemate cleavage with application of hydrochloride l-lysine-auxiliary base-system as optically cleavaging agent