ZA906810B - Heterogeneous synthesis of azepinones from esters - Google Patents

Heterogeneous synthesis of azepinones from esters

Info

Publication number
ZA906810B
ZA906810B ZA906810A ZA906810A ZA906810B ZA 906810 B ZA906810 B ZA 906810B ZA 906810 A ZA906810 A ZA 906810A ZA 906810 A ZA906810 A ZA 906810A ZA 906810 B ZA906810 B ZA 906810B
Authority
ZA
South Africa
Prior art keywords
cyclized
methoxyphenyl
hydroxy
amino
acid
Prior art date
Application number
ZA906810A
Other languages
English (en)
Inventor
Daniel Eugene Martin
Eugene Martin Daniel
Original Assignee
Marion Merrell Dow Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Marion Merrell Dow Inc filed Critical Marion Merrell Dow Inc
Publication of ZA906810B publication Critical patent/ZA906810B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ZA906810A 1989-08-31 1990-08-27 Heterogeneous synthesis of azepinones from esters ZA906810B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US40065889A 1989-08-31 1989-08-31

Publications (1)

Publication Number Publication Date
ZA906810B true ZA906810B (en) 1991-10-30

Family

ID=23584491

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA906810A ZA906810B (en) 1989-08-31 1990-08-27 Heterogeneous synthesis of azepinones from esters

Country Status (13)

Country Link
EP (1) EP0415384B1 (de)
JP (1) JP3090212B2 (de)
KR (1) KR0163585B1 (de)
AT (1) ATE150459T1 (de)
AU (1) AU628217B2 (de)
CA (1) CA2024124C (de)
DD (1) DD295367A5 (de)
DE (1) DE69030222T2 (de)
ES (1) ES2101682T3 (de)
HU (1) HU206103B (de)
IE (1) IE903151A1 (de)
IL (1) IL95509A (de)
ZA (1) ZA906810B (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1249318B (it) * 1991-05-23 1995-02-22 Zambon Spa Processo per la preparazione di benzotiazepine per ciclizzazione con acidi fosfonici
DE4313413A1 (de) * 1993-04-23 1994-10-27 Basf Ag 3-(Het)aryloxy(thio)-Carbonsäurederivate, Verfahren und Zwischenprodukte zu ihrer Herstellung

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4567175A (en) * 1983-06-03 1986-01-28 Tanabe Seiyaku Co., Ltd. 8-Chloro-1,5-benzothiazepine derivatives
ZA893392B (en) * 1988-05-24 1990-01-31 Hoffmann La Roche Process for the manufacture of optically active naphthothiazepinones
ATE116643T1 (de) * 1989-04-28 1995-01-15 Tanabe Seiyaku Co Verfahren zur herstellung von 1,5- benzothiazepinderivaten.
JPH0798813B2 (ja) * 1989-04-28 1995-10-25 田辺製薬株式会社 １，５―ベンゾチアゼピン誘導体の製法

Also Published As

Publication number Publication date
IL95509A0 (en) 1991-06-30
EP0415384A3 (en) 1992-04-15
KR910004584A (ko) 1991-03-29
DE69030222T2 (de) 1997-10-16
IL95509A (en) 1994-10-07
EP0415384B1 (de) 1997-03-19
HU905508D0 (en) 1991-02-28
IE903151A1 (en) 1991-03-27
KR0163585B1 (ko) 1998-12-01
CA2024124A1 (en) 1991-03-01
CA2024124C (en) 2003-04-15
AU628217B2 (en) 1992-09-10
JP3090212B2 (ja) 2000-09-18
ATE150459T1 (de) 1997-04-15
DE69030222D1 (de) 1997-04-24
JPH0393778A (ja) 1991-04-18
HUT59118A (en) 1992-04-28
HU206103B (en) 1992-08-28
AU6138290A (en) 1991-03-07
DD295367A5 (de) 1991-10-31
ES2101682T3 (es) 1997-07-16
EP0415384A2 (de) 1991-03-06

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