ZA821196B - Substituted benzimidazolones and salts thereof, methods of preparation and pharmaceutical compositions thereof - Google Patents
Substituted benzimidazolones and salts thereof, methods of preparation and pharmaceutical compositions thereofInfo
- Publication number
- ZA821196B ZA821196B ZA821196A ZA821196A ZA821196B ZA 821196 B ZA821196 B ZA 821196B ZA 821196 A ZA821196 A ZA 821196A ZA 821196 A ZA821196 A ZA 821196A ZA 821196 B ZA821196 B ZA 821196B
- Authority
- ZA
- South Africa
- Prior art keywords
- salts
- preparation
- methods
- pharmaceutical compositions
- substituted benzimidazolones
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/237,966 US4359468A (en) | 1981-02-25 | 1981-02-25 | Antiallergic N-[4-(indolyl)-piperidino-alkyl]-benzimidazolones |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA821196B true ZA821196B (en) | 1983-10-26 |
Family
ID=22895956
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA821196A ZA821196B (en) | 1981-02-25 | 1982-02-24 | Substituted benzimidazolones and salts thereof, methods of preparation and pharmaceutical compositions thereof |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US4359468A (el) |
| EP (1) | EP0058975B1 (el) |
| JP (1) | JPS57156484A (el) |
| KR (1) | KR890000008B1 (el) |
| AR (1) | AR228475A1 (el) |
| AT (1) | ATE10742T1 (el) |
| AU (1) | AU543948B2 (el) |
| CA (1) | CA1191137A (el) |
| CS (1) | CS227343B2 (el) |
| DD (1) | DD202562A5 (el) |
| DE (1) | DE3261497D1 (el) |
| DK (1) | DK151017C (el) |
| ES (2) | ES509871A0 (el) |
| FI (1) | FI71558C (el) |
| GB (1) | GB2093455B (el) |
| GR (1) | GR74778B (el) |
| HU (1) | HU187652B (el) |
| IE (1) | IE52562B1 (el) |
| IL (1) | IL65097A0 (el) |
| NO (1) | NO157296C (el) |
| NZ (1) | NZ199822A (el) |
| PH (1) | PH17889A (el) |
| PL (1) | PL135472B1 (el) |
| PT (1) | PT74481B (el) |
| SU (1) | SU1088665A3 (el) |
| UA (1) | UA7228A1 (el) |
| YU (1) | YU42758B (el) |
| ZA (1) | ZA821196B (el) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4548939A (en) * | 1984-10-01 | 1985-10-22 | Janssen Pharmaceutica N. V. | 1H-Indol-3-yl containing 1,3-dimethyl-1H-purine-2,6-diones |
| IE58370B1 (en) * | 1985-04-10 | 1993-09-08 | Lundbeck & Co As H | Indole derivatives |
| US4742057A (en) * | 1985-12-05 | 1988-05-03 | Fujisawa Pharmaceutical Co., Ltd. | Antiallergic thiazole compounds |
| FR2613222B1 (fr) * | 1987-04-03 | 1991-06-14 | Guigon Nadine | Composition pour les soins locaux de l'epiderme, notamment du cuir chevelu |
| DK733788A (da) * | 1988-01-14 | 1989-07-15 | Fujisawa Pharmaceutical Co | Indolylpiperidinderivater og fremgangsmaade til fremstilling deraf |
| US5238945A (en) * | 1989-04-11 | 1993-08-24 | H. Lundbeck A/S | Method of treating psychoses |
| GB8908085D0 (en) * | 1989-04-11 | 1989-05-24 | Lundbeck & Co As H | New therapeutic use |
| FR2658823B1 (fr) * | 1990-02-27 | 1992-04-30 | Adir | Nouveaux derives d'aminomethylpiperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent . |
| TW203049B (el) * | 1990-04-13 | 1993-04-01 | Yamanouchi Pharma Co Ltd | |
| DE4414113A1 (de) * | 1994-04-22 | 1995-10-26 | Merck Patent Gmbh | 3-Indolylpiperidine |
| US5965582A (en) * | 1994-08-03 | 1999-10-12 | Asta Medica Aktiengesellschaft | N-benzylindole and benzopyrazole derivatives with anti-asthmatic, anti-allergic, anti-inflammatory and immunemodulating effect |
| US5521196A (en) * | 1994-10-05 | 1996-05-28 | Eli Lilly And Company | 5-HT1F agonists for the treatment of migraine |
| US5521197A (en) * | 1994-12-01 | 1996-05-28 | Eli Lilly And Company | 3-<1-alkylenearyl>-4-<1,2,3,6-tetrahydropyridinyl>-and 3-<1-alkylenearyl>-4-piperidinyl-1h-indoles: new 5-HT1F agonists |
| KR19980703048A (ko) * | 1995-03-20 | 1998-09-05 | 피터쥐.스트링거 | 5-치환-3-(1,2,3,6-테트라히드로피리딘-4-일)- 및 3-(피페리딘-4-일)-1ｈ-인돌: 신규한 5-ｈｔ1ｆ 아고니스트 |
| GB9825413D0 (en) | 1998-11-19 | 1999-01-13 | Lilly Co Eli | Pharmaceutical compounds |
| GB9903784D0 (en) * | 1999-02-18 | 1999-04-14 | Lilly Co Eli | Pharmaceutical compounds |
| WO2004047769A2 (en) * | 2002-11-26 | 2004-06-10 | Isis Pharmaceuticals, Inc. | Benzimidazoles and analogs thereof as antibacterials |
| US7759365B2 (en) * | 2005-04-30 | 2010-07-20 | Boehringer Ingelheim International Gmbh | Piperidine-substituted indoles |
| JP2009515833A (ja) * | 2005-10-24 | 2009-04-16 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | ３−ピペリジン−４−イル−インドールｏｒｌ−１受容体モジュレーター |
| US8462477B2 (en) | 2010-09-13 | 2013-06-11 | Analog Devices, Inc. | Junction field effect transistor for voltage protection |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE794333A (fr) * | 1972-01-20 | 1973-07-19 | Wyeth John & Brother Ltd | Composes heterocycliques azotes therapeutiques |
| US3954764A (en) * | 1973-03-30 | 1976-05-04 | Hoffmann-La Roche Inc. | Dibenzo [b,f]thiepins bearing piperazinyl substitution |
| DE2322470A1 (de) * | 1973-05-04 | 1974-11-21 | Boehringer Sohn Ingelheim | Neue indolyl-piperidino-(bzw. 1,2,5,6tetrahydro-pyridyl-)butyrophenone und verfahren zu ihrer herstellung |
| ZA76475B (en) * | 1975-03-10 | 1977-08-31 | Ciba Geigy Ag | Indolyalkylpiperidines |
| US4147786A (en) * | 1976-02-02 | 1979-04-03 | Ciba-Geigy Corporation | 1-Indolylalkyl-3-or 4-trimethyleneurido-piperidines |
| FR2469411A1 (fr) * | 1979-11-15 | 1981-05-22 | Science Union & Cie | Nouveaux derives de la piperidylbenzimidazolinone, leurs procedes de preparation et les compositions pharmaceutiques les renfermant |
| US4254127A (en) * | 1980-04-03 | 1981-03-03 | Janssen Pharmaceutica, N.V. | 1,3-Dihydro-1-[(1-piperidinyl)alkyl]-2H-benzimidazol-2-one derivatives |
-
1981
- 1981-02-25 US US06/237,966 patent/US4359468A/en not_active Expired - Lifetime
-
1982
- 1982-02-19 PH PH26888A patent/PH17889A/en unknown
- 1982-02-20 EP EP82101315A patent/EP0058975B1/de not_active Expired
- 1982-02-20 DE DE8282101315T patent/DE3261497D1/de not_active Expired
- 1982-02-20 AT AT82101315T patent/ATE10742T1/de not_active IP Right Cessation
- 1982-02-22 GR GR67368A patent/GR74778B/el unknown
- 1982-02-22 DD DD82237583A patent/DD202562A5/de not_active IP Right Cessation
- 1982-02-23 PL PL1982235187A patent/PL135472B1/pl unknown
- 1982-02-23 CS CS821228A patent/CS227343B2/cs unknown
- 1982-02-23 FI FI820594A patent/FI71558C/fi not_active IP Right Cessation
- 1982-02-24 GB GB8205386A patent/GB2093455B/en not_active Expired
- 1982-02-24 IE IE401/82A patent/IE52562B1/en not_active IP Right Cessation
- 1982-02-24 IL IL65097A patent/IL65097A0/xx not_active IP Right Cessation
- 1982-02-24 HU HU82566A patent/HU187652B/hu not_active IP Right Cessation
- 1982-02-24 ZA ZA821196A patent/ZA821196B/xx unknown
- 1982-02-24 NZ NZ199822A patent/NZ199822A/en unknown
- 1982-02-24 CA CA000396960A patent/CA1191137A/en not_active Expired
- 1982-02-24 SU SU823396888A patent/SU1088665A3/ru active
- 1982-02-24 YU YU410/82A patent/YU42758B/xx unknown
- 1982-02-24 NO NO820583A patent/NO157296C/no unknown
- 1982-02-24 PT PT74481A patent/PT74481B/pt not_active IP Right Cessation
- 1982-02-24 AR AR288538A patent/AR228475A1/es active
- 1982-02-24 DK DK079882A patent/DK151017C/da not_active IP Right Cessation
- 1982-02-24 UA UA3396888A patent/UA7228A1/uk unknown
- 1982-02-24 ES ES509871A patent/ES509871A0/es active Granted
- 1982-02-24 JP JP57028704A patent/JPS57156484A/ja active Granted
- 1982-02-25 KR KR8200868A patent/KR890000008B1/ko active
- 1982-02-25 AU AU80783/82A patent/AU543948B2/en not_active Ceased
- 1982-12-07 ES ES517988A patent/ES517988A0/es active Granted
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