ZA201302390B - Arylosulfonamides for the treatment of cns diseases - Google Patents

Arylosulfonamides for the treatment of cns diseases

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Publication number
ZA201302390B
ZA201302390B ZA2013/02390A ZA201302390A ZA201302390B ZA 201302390 B ZA201302390 B ZA 201302390B ZA 2013/02390 A ZA2013/02390 A ZA 2013/02390A ZA 201302390 A ZA201302390 A ZA 201302390A ZA 201302390 B ZA201302390 B ZA 201302390B
Authority
ZA
South Africa
Prior art keywords
arylosulfonamides
treatment
cns diseases
cns
diseases
Prior art date
Application number
ZA2013/02390A
Other languages
English (en)
Inventor
Marcin Kolaczkowski
Piotr Kowalski
Jolanta Jaskowska
Monika Marcinkowska
Katarzyna Mitka
Adam Bucki
Anna Wesolowska
Maciej Pawlowski
Original Assignee
Adamed Sp Zoo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adamed Sp Zoo filed Critical Adamed Sp Zoo
Publication of ZA201302390B publication Critical patent/ZA201302390B/en

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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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ZA2013/02390A 2010-09-17 2013-04-03 Arylosulfonamides for the treatment of cns diseases ZA201302390B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PL39243610A PL392436A1 (pl) 2010-09-17 2010-09-17 Pochodne arylosulfonamidów do leczenia chorób odśrodkowego układu nerwowego
PCT/EP2011/066054 WO2012035123A1 (en) 2010-09-17 2011-09-16 Arylosulfonamides for the treatment of cns diseases

Publications (1)

Publication Number Publication Date
ZA201302390B true ZA201302390B (en) 2013-12-23

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ZA2013/02390A ZA201302390B (en) 2010-09-17 2013-04-03 Arylosulfonamides for the treatment of cns diseases
ZA2013/05970A ZA201305970B (en) 2010-09-17 2013-08-07 Arylosulfonami for the treatment of cns diseases

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ZA2013/05970A ZA201305970B (en) 2010-09-17 2013-08-07 Arylosulfonami for the treatment of cns diseases

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US (2) US8822517B2 (https=)
EP (1) EP2616440A1 (https=)
JP (1) JP5899218B2 (https=)
KR (1) KR20130143569A (https=)
CN (2) CN104529999A (https=)
AU (1) AU2011303807B2 (https=)
BR (1) BR112013006313A2 (https=)
CA (1) CA2808246A1 (https=)
EA (1) EA022776B1 (https=)
MX (1) MX2013002956A (https=)
NZ (1) NZ607031A (https=)
PL (1) PL392436A1 (https=)
UA (1) UA109793C2 (https=)
WO (1) WO2012035123A1 (https=)
ZA (2) ZA201302390B (https=)

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WO2015158313A1 (en) 2014-04-19 2015-10-22 Sunshine Lake Pharma Co., Ltd. Sulfonamide derivatives and pharmaceutical applications thereof
CN106749219A (zh) * 2015-11-20 2017-05-31 江苏恩华药业股份有限公司 一种内酰胺类衍生物及其应用
CN107602446B (zh) * 2016-07-12 2020-04-07 中国科学院上海药物研究所 1,4-双取代-1,2,3,6-四氢吡啶类化合物、其制备方法、药物组合物及其应用
PT4082616T (pt) * 2019-12-24 2025-12-02 Sumitomo Pharma Co Ltd Derivado de amida ácida alifática
CN116157124A (zh) * 2020-05-29 2023-05-23 大邱庆北尖端医疗产业振兴财团 磺胺衍生物和含其作为活性成分的用于预防或治疗精神疾病的药物组合物
KR102447231B1 (ko) * 2020-05-29 2022-09-27 재단법인 대구경북첨단의료산업진흥재단 설폰아미드 유도체 및 이를 유효성분으로 함유하는 정신질환의 예방 또는 치료용 약학적 조성물

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JP2556722B2 (ja) 1988-02-18 1996-11-20 興和株式会社 新規なスルホンアミド化合物
DE19500689A1 (de) * 1995-01-12 1996-07-18 Merck Patent Gmbh Indolpiperidin-Derivate
TWI242011B (en) * 1997-03-31 2005-10-21 Eisai Co Ltd 1,4-substituted cyclic amine derivatives
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EA201390398A1 (ru) 2013-07-30
EP2616440A1 (en) 2013-07-24
CN104529999A (zh) 2015-04-22
NZ607031A (en) 2014-06-27
EA022776B1 (ru) 2016-02-29
US20130172365A1 (en) 2013-07-04
KR20130143569A (ko) 2013-12-31
JP2013540738A (ja) 2013-11-07
JP5899218B2 (ja) 2016-04-06
US8822517B2 (en) 2014-09-02
ZA201305970B (en) 2014-04-30
AU2011303807A1 (en) 2013-02-28
AU2011303807B2 (en) 2014-07-17
US9120767B2 (en) 2015-09-01
PL392436A1 (pl) 2012-03-26
WO2012035123A1 (en) 2012-03-22
CA2808246A1 (en) 2012-03-22
BR112013006313A2 (pt) 2016-06-07
US20140336200A1 (en) 2014-11-13
UA109793C2 (uk) 2015-10-12
CN103108864A (zh) 2013-05-15
MX2013002956A (es) 2013-05-09

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