ZA201007614B - Indolesulfonyl protecting groups for protection of guanidino and amino groups - Google Patents

Indolesulfonyl protecting groups for protection of guanidino and amino groups

Info

Publication number
ZA201007614B
ZA201007614B ZA2010/07614A ZA201007614A ZA201007614B ZA 201007614 B ZA201007614 B ZA 201007614B ZA 2010/07614 A ZA2010/07614 A ZA 2010/07614A ZA 201007614 A ZA201007614 A ZA 201007614A ZA 201007614 B ZA201007614 B ZA 201007614B
Authority
ZA
South Africa
Prior art keywords
indolesulfonyl
guanidino
protection
groups
amino groups
Prior art date
Application number
ZA2010/07614A
Other languages
English (en)
Inventor
Domingo Mercedes Alvarez
Llobet Albert Isidro
Fernando Albericio
Matthieu Giraud
Original Assignee
Lonza Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza Ag filed Critical Lonza Ag
Publication of ZA201007614B publication Critical patent/ZA201007614B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA2010/07614A 2008-05-05 2010-10-25 Indolesulfonyl protecting groups for protection of guanidino and amino groups ZA201007614B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP08008418 2008-05-05
US9570908P 2008-09-10 2008-09-10
PCT/EP2009/003210 WO2009135645A1 (en) 2008-05-05 2009-05-05 Indolesulfonyl protecting groups for protection of guanidino and amino groups

Publications (1)

Publication Number Publication Date
ZA201007614B true ZA201007614B (en) 2011-07-27

Family

ID=39772857

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA2010/07614A ZA201007614B (en) 2008-05-05 2010-10-25 Indolesulfonyl protecting groups for protection of guanidino and amino groups

Country Status (16)

Country Link
US (1) US8431720B2 (enExample)
EP (2) EP2420489B1 (enExample)
JP (2) JP5567004B2 (enExample)
KR (2) KR101521400B1 (enExample)
CN (1) CN102026971B (enExample)
AU (1) AU2009243730B2 (enExample)
BR (1) BRPI0912355A2 (enExample)
CA (1) CA2721644C (enExample)
CO (1) CO6390068A2 (enExample)
DK (1) DK2420489T3 (enExample)
EA (1) EA022476B1 (enExample)
ES (1) ES2477590T3 (enExample)
IL (1) IL208930A (enExample)
MX (1) MX2010012113A (enExample)
WO (1) WO2009135645A1 (enExample)
ZA (1) ZA201007614B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103626996B (zh) * 2013-11-29 2016-04-27 沈阳药科大学 胍基化的含二硫键聚氨基胺类聚合物及其制备和应用
EP3305780A1 (en) 2016-10-05 2018-04-11 Lonza Ltd Method for the preparation of h-arg(mis)-oh
WO2018064829A1 (en) * 2016-10-09 2018-04-12 Polypeptide Laboratories Holding (Ppl) Ab Method for the preparation of h-arg (mis) -oh
EP3315490A1 (en) 2016-10-31 2018-05-02 Polypeptide Laboratories Holding (PPL) AB Method for the preparation of h-arg(mis)-oh

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10004572A1 (de) * 2000-02-02 2001-08-09 Boehringer Ingelheim Pharma Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
EP1501826B1 (en) 2002-02-01 2006-09-27 F. Hoffman-la Roche AG Substituted indoles as alpha-1 agonists
CN100453537C (zh) * 2004-05-08 2009-01-21 上海依福瑞实业有限公司 一种双保护氨基酸的制备方法
US8585885B2 (en) * 2007-08-28 2013-11-19 Rohm And Haas Electronic Materials Llc Electrochemically deposited indium composites

Also Published As

Publication number Publication date
KR101521400B1 (ko) 2015-05-18
JP5985534B2 (ja) 2016-09-06
AU2009243730B2 (en) 2013-07-18
ES2477590T3 (es) 2014-07-17
EP2280942A1 (en) 2011-02-09
JP5567004B2 (ja) 2014-08-06
US20110060125A1 (en) 2011-03-10
EA022476B1 (ru) 2016-01-29
EP2420489B1 (en) 2014-04-23
MX2010012113A (es) 2010-12-01
AU2009243730A1 (en) 2009-11-12
CN102026971B (zh) 2014-10-29
CA2721644A1 (en) 2009-11-12
JP2011519884A (ja) 2011-07-14
IL208930A (en) 2014-07-31
KR20140061548A (ko) 2014-05-21
IL208930A0 (en) 2011-01-31
HK1154860A1 (en) 2012-05-04
CO6390068A2 (es) 2012-02-29
JP2014193872A (ja) 2014-10-09
CN102026971A (zh) 2011-04-20
CA2721644C (en) 2013-10-15
EP2420489A1 (en) 2012-02-22
KR20110014167A (ko) 2011-02-10
EA201001738A1 (ru) 2011-06-30
WO2009135645A1 (en) 2009-11-12
DK2420489T3 (da) 2014-07-21
US8431720B2 (en) 2013-04-30
KR101493554B1 (ko) 2015-02-16
BRPI0912355A2 (pt) 2015-07-28

Similar Documents

Publication Publication Date Title
GB2462789B (en) Procedures and compositions for reservoir protection
GB0800150D0 (en) Rotational ahterectomy system with enhanced distal protection capability and method of use
IL209477A (en) Pyrrolidine derivatives as 2-metap inhibitors and their pharmacological preparations
IL201406A0 (en) Ischemia / reperfusion protection compositions and methods of using
IL210804A0 (en) Deacetylase inhibitors and uses thereof
SG10201504623VA (en) Peptides and compositions for prevention of cell adhesion and methods of using same
GB0814173D0 (en) Cable protectors and methods of cable protection
SG10201504379VA (en) Peptides and compositions for prevention of cell adhesion and methods of using same
EP2091914A4 (en) TRANSDERMAL ADMINISTRATION SYSTEMS FOR PEPTIDES AND RELATED CONNECTIONS
LT2297057T (lt) Laikina stiklo apsauga
EP2563121A4 (en) METHODS AND COMPOSITIONS FOR PROTECTION AGAINST NEUROTOXIC AGENTS
IL189088A0 (en) Protective divide and method for protection
IL217535A0 (en) Compositions and methods of use for post-radiation protection
GB2458367B (en) Protective suit and methods of manufacture thereof
ZA201007614B (en) Indolesulfonyl protecting groups for protection of guanidino and amino groups
IL194363A0 (en) Bulletproof protector and bulletproof clother
EP2307558A4 (en) COMPOSITIONS AND PROCEDURES FOR THE PROTECTION OF NUCLEOPHILER GROUPS
EP2046377A4 (en) PROCEDURE FOR PROTECTION AGAINST STAPHYLOKOKEN INFECTIONS
GB0819084D0 (en) ESD protection
GB0720717D0 (en) Protection of plastics
EP2265142A4 (en) NAIL PROTECTION APPARATUS
TWI372762B (en) Amino derivatives of b-homoandrostanes and b-heteroandrostanes
PL2512498T3 (pl) Ochrona peptydowa przed toksycznością wywołaną światłem ultrafioletowym
GB0823189D0 (en) Protection of computer systems
GB201005579D0 (en) Fire protected structures and components for fire protection