DK2420489T3 - Indolsulfonylbeskyttelsesgrupper til beskyttelse af guanidino- og aminogrupper - Google Patents

Indolsulfonylbeskyttelsesgrupper til beskyttelse af guanidino- og aminogrupper

Info

Publication number
DK2420489T3
DK2420489T3 DK11007876.3T DK11007876T DK2420489T3 DK 2420489 T3 DK2420489 T3 DK 2420489T3 DK 11007876 T DK11007876 T DK 11007876T DK 2420489 T3 DK2420489 T3 DK 2420489T3
Authority
DK
Denmark
Prior art keywords
protection
indolsulphonyl
aminographs
guanidino
groups
Prior art date
Application number
DK11007876.3T
Other languages
Danish (da)
English (en)
Inventor
Matthieu Giraud
Fernando Albericio
Domingo Mercedes Alvarez
Llobet Albert Isidro
Original Assignee
Lonza Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza Ag filed Critical Lonza Ag
Application granted granted Critical
Publication of DK2420489T3 publication Critical patent/DK2420489T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK11007876.3T 2008-05-05 2009-05-05 Indolsulfonylbeskyttelsesgrupper til beskyttelse af guanidino- og aminogrupper DK2420489T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP08008418 2008-05-05
US9570908P 2008-09-10 2008-09-10
EP09741864A EP2280942A1 (en) 2008-05-05 2009-05-05 Indolesulfonyl protecting groups for protection of guanidino and amino groups

Publications (1)

Publication Number Publication Date
DK2420489T3 true DK2420489T3 (da) 2014-07-21

Family

ID=39772857

Family Applications (1)

Application Number Title Priority Date Filing Date
DK11007876.3T DK2420489T3 (da) 2008-05-05 2009-05-05 Indolsulfonylbeskyttelsesgrupper til beskyttelse af guanidino- og aminogrupper

Country Status (16)

Country Link
US (1) US8431720B2 (enExample)
EP (2) EP2420489B1 (enExample)
JP (2) JP5567004B2 (enExample)
KR (2) KR101521400B1 (enExample)
CN (1) CN102026971B (enExample)
AU (1) AU2009243730B2 (enExample)
BR (1) BRPI0912355A2 (enExample)
CA (1) CA2721644C (enExample)
CO (1) CO6390068A2 (enExample)
DK (1) DK2420489T3 (enExample)
EA (1) EA022476B1 (enExample)
ES (1) ES2477590T3 (enExample)
IL (1) IL208930A (enExample)
MX (1) MX2010012113A (enExample)
WO (1) WO2009135645A1 (enExample)
ZA (1) ZA201007614B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103626996B (zh) * 2013-11-29 2016-04-27 沈阳药科大学 胍基化的含二硫键聚氨基胺类聚合物及其制备和应用
EP3305780A1 (en) 2016-10-05 2018-04-11 Lonza Ltd Method for the preparation of h-arg(mis)-oh
WO2018064829A1 (en) * 2016-10-09 2018-04-12 Polypeptide Laboratories Holding (Ppl) Ab Method for the preparation of h-arg (mis) -oh
EP3315490A1 (en) 2016-10-31 2018-05-02 Polypeptide Laboratories Holding (PPL) AB Method for the preparation of h-arg(mis)-oh

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10004572A1 (de) * 2000-02-02 2001-08-09 Boehringer Ingelheim Pharma Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
EP1501826B1 (en) 2002-02-01 2006-09-27 F. Hoffman-la Roche AG Substituted indoles as alpha-1 agonists
CN100453537C (zh) * 2004-05-08 2009-01-21 上海依福瑞实业有限公司 一种双保护氨基酸的制备方法
US8585885B2 (en) * 2007-08-28 2013-11-19 Rohm And Haas Electronic Materials Llc Electrochemically deposited indium composites

Also Published As

Publication number Publication date
KR101521400B1 (ko) 2015-05-18
JP5985534B2 (ja) 2016-09-06
AU2009243730B2 (en) 2013-07-18
ES2477590T3 (es) 2014-07-17
EP2280942A1 (en) 2011-02-09
JP5567004B2 (ja) 2014-08-06
US20110060125A1 (en) 2011-03-10
EA022476B1 (ru) 2016-01-29
EP2420489B1 (en) 2014-04-23
MX2010012113A (es) 2010-12-01
AU2009243730A1 (en) 2009-11-12
CN102026971B (zh) 2014-10-29
CA2721644A1 (en) 2009-11-12
JP2011519884A (ja) 2011-07-14
IL208930A (en) 2014-07-31
KR20140061548A (ko) 2014-05-21
IL208930A0 (en) 2011-01-31
HK1154860A1 (en) 2012-05-04
CO6390068A2 (es) 2012-02-29
JP2014193872A (ja) 2014-10-09
CN102026971A (zh) 2011-04-20
CA2721644C (en) 2013-10-15
ZA201007614B (en) 2011-07-27
EP2420489A1 (en) 2012-02-22
KR20110014167A (ko) 2011-02-10
EA201001738A1 (ru) 2011-06-30
WO2009135645A1 (en) 2009-11-12
US8431720B2 (en) 2013-04-30
KR101493554B1 (ko) 2015-02-16
BRPI0912355A2 (pt) 2015-07-28

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